Chemistry towards life sciences

Our Publications

The team gathers four thematic groups with common research interests in the field of molecular and supramolecular chemistry to study, mimic or interact with living systems. Major topics include:

Methodological developments

This axis addresses two major issues: the need for greater chemical diversity and the need for new methodologies allowing the selective functionalization of complex biomolecules.

The first approach aims at developing complexity-oriented synthetic methods by: 1) setting up short and scalable routes to complex or densely functionalized scaffolds notably by transition metal-catalyzed domino sequences and post-(de)functionalization. 2) Generating novel chemical entities by exploring the synthetic potential of organoaluminum reagents. 3) Exploring the chemical space between natural products and synthetic compounds using engineered microorganisms to produce natural-product like new chemical entities in a mutasynthetic approach. And finally 4) widen the chemical space of reactions conducted under kinetic control through flow-chemistry technics.

The second approach concerns biomolecules with the development of post-synthetic methodologies for bi-functionalization of RNAs with reactive groups, affinity purification tags, and fluorescent probes.

RNA directed chemistry

Investigating the biology of RNA is of great interest to better explore living systems at a molecular/supramolecular level. Our goals are to develop: 1) Tools and probes to better understand the biosynthesis and post-transcriptional modifications of RNA by designing analogues of S-adenosyl-L-methionine (SAM), an ubiquitous cofactor acting as a carbon source for methylation or more complex post-transcriptional modifications. We notably focus on RNA methylation by methyltransferases such as TrmK, a bacterial tRNA MTase. And 2) Molecular probes for sensing single-stranded RNA regions. The [2.2]paracyclophane scaffold  that cannot intercalate in classical multi-stranded helices is used for the design of new ligands allowing the specific recognition of non-helical RNA tridimensional motifs through either a fluorimetric response or SERS-based detection (after grafting on gold surfaces). These sensors will be used as reporters to drive the design of small molecules capable of binding to RNA and interfering with its biological activity.

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molecular diversity rna directed chemistry

Nature’s inspired models and concepts

Biomimetic coordination chemistry is a major field devoted to a better understanding of fundamental enzymatic processes. It comprises molecular recognition on the one hand and reactivity and catalysis on the other hand. Our major goals are to: 1) Elaborate efficient and selective receptors for small biological molecules. These are based on the host-guest chemistry of cavity-complexes with the aim to provide probes (either water-soluble or electrode-grafted) with high affinity constants and allowing spectroscopic reporting in a biological context. 2) Obtain new fundamental insights into electron and proton coupled redox processes under the supramolecular control provided by the cavities surrounding the metal ion. This is mainly focused on redox-active cavities (integrating quinone or phenol moieties), which, up to now, have never been exploited in the context of biomimetic coordination chemistry. And 3) Elaborate new catalysts for the activation of small molecules (O2, N2, CO2, H2…). Two levels of studies will be conducted: the first one concerns solution studies of the new complexes, whereas the second one is based on the grafting of the ligands/cavities/metal complexes on electro-active surfaces.

Targets and Drug design

Developing drug design programs and molecular tools for the study of biological targets is also a major priority. We are focusing on: 1) Infectious diseases. The goals are to study and inhibit enzymes involved in the biosynthesis of bacterial peptidoglycan, with different approaches: i) the use of functionalized RNAs, to study the tRNA recognition by amino-acyltransferases of the Fem family. ii) the design and synthesis of inhibitors to study LDts-transpeptidases and MurT/GatD amidotransferase complex. iii) The discovery of new MraY inhibitors through a combination of virtual screening and multi-component synthesis. 2) New antiviral therapy. The goal is to use novel classes of compounds we developed, and able to interfere with the proliferation of the HIV, to discover and study new targets in its replication cycle. 3) Congenital diseases. Novel fluorescent and biotinylated probes are developed to assay, purify and inhibit mammalian Dolichol Linked Oligosaccharide DiPhosphatases (DLODPs) to explore their roles in rare inherited diseases. 4) Cancer. Focal adhesion kinase (FAK) belongs to the most attractive tyrosine kinase targets for cancer chemotherapy. We develop new potent irreversible inhibitors of FAK based on the first crystallographic structure of a covalent complex between FAK and an irreversible inhibitor we recently obtained.

nature inspired models and concepts anti-infectious deseases
Our Publications

Team Leaders

Research Groups

OSBioR

Organic synthesis for biomedical research

NSynC

New synthetic methods for the chemistry/biology interface

CRANPH

Chemistry of RNAs, Nucleosides, Peptides and Heterocycles

SBiC

Supramolecular Bio-inorganic Chemistry

Organic synthesis for biomedical research

The group’s expertise relies on multi-step synthesis of smart molecules for the chemistry-biology interface, methodology in organic synthesis and diversity oriented synthesis. Our objectives span from the development of new methodologies towards privileged structures in medicinal chemistry to the synthesis of enzymes inhibitors and molecular tools for biology. The designed methods are based on step and atom economy concepts and they notably involve domino reactions catalyzed by transition metals. We recently developed a green process based on the iron catalyzed generation of nitrene to perform the aziridination of alkenes. An unprecedented catalytic reductive cleavage of aromatic and heteroaromatic methyl ester functions was also successfully performed with a cheap, non-toxic, and air-stable Cu(OAc)2 catalyst. The diastereoselectivity of uridine-derived aldehyde 5’-alkynylation was investigated and revealed to be highly dependent on uridine protected groups. The synthesis of probes and molecules to study and inhibit enzymes involved in peptidoglycan biosynthesis machinery (MraY transferase, MurT/GatD amidotransferase complex) is a major objective of the group. No marketed drug is targeting these enzymes which are essential for bacteria viability, a key feature to tackle the issue of bacterial resistance to commonly used antibiotics. Complementary in silico approaches involving structure-based and ligand-based drug design are exploited. We are also developing new antiviral therapy to fight replication-cycle of HIV. Molecules resulting from our methodological developments were identified as novel classes of compounds interfering with the proliferation of the HIV with encouraging potency. These new tools will be used to discover and study new targets in the replication cycle of the HIV. Other on-going projects are dedicated to the design and synthesis of chemical tools for a better understanding of some pathologies such as Congenital Disorders of Glycosylation or Cystic Fibrosis. All the projects, at the interface between chemistry and biology, benefit from multi-disciplinary collaboration at the local, national and international levels. Major achievements can be reached thanks to the invaluable contribution of numerous motivated students and to the financial support of funding agencies (ANR, ANRS, VLM, FRM), they are gratefully acknowledged.

Permanent Members

Group leaders

Members

New synthetic methods for the chemistry/biology interface

The interests of the group span a wide range of topics in the fields of synthetic organic chemistry and chemical biology, all of them being grounded on molecular innovation. Our works involve the exploration of new chemical spaces as well as the development of synthetic tools or analytical methods for studying and / or interfering with biological regulatory mechanisms. Our research activities are organized around two main axes:

RNA ligands: chemical spaces, probes and analytical methods

Diversity-oriented-synthesis of cyclic polyamines

Chiral paracyclophanes

RNA/ligand interactions

Organometallic chemistry and molecular diversity: Synthesis and reactivity of organoaluminum reagents 

Reactivity of Organoaluminum reagents

Permanent Members

Group leader

  • Laurent Micouin, Senior Research Scientist, Chemistry towards life sciences, New synthetic methods for the chemistry/biology interface
    laurent.micouin@-Code to remove to avoid SPAM-parisdescartes.fr, +33 1 42 86 20 40, room R216-2, R216-7

Members

Main publications

(click here for all publications)

1. M.-L. Delcourt, S. Felder, E. Benedetti, L. Micouin Highly Enantioselective Desymmetrization of Centrosymmetric pseudo-para-Diformyl [2.2 ]paracyclophane via Asymmetric Transfer Hydrogenation. ACS Catalysis 2018, 8, 6612-6616
2. H. Guyon, F. Mavré, M. Catala, S. Turcaud, F. Brachet, B. Limoges, C. Tisné, L. Micouin Use of a redox probe for an electrochemical RNA–ligand binding assay in microliter droplets Chem. Commun., 2017, 53, 1140-1143
3. M.-L Delcourt, C. Reynaud, S. Turcaud, L. Favereau, J. Crassous, L. Micouin, E. Benedetti 3D Coumarin Systems Based on [2.2]Paracyclophane: Synthesis, Spectroscopic Characterization, and Chiroptical Properties J. Org. Chem. 2019, 84, 888-899
4. P. Gordillo, P. Clerici, L. Micouin Modular Access to N-subtituted cis 5-amino-3-hydroxypiperidines J. Org. Chem. 2017, 82, 7689-7694
5. T. Zhao, R. Piccardi, L. Micouin Rapid and Effective Synthesis of α-Acyloxy-α-alkynyl-trimethylsilanes Organic Lett. 2018, 20, 5015-5018
6. R. Piccardi, S. Turcaud, E. Benedetti, L. Micouin Synthesis and Reactivity of Mixed Dimethylalkynylaluminum Reagents. Synthesis 2019, 51, 97-106

Chemistry of RNAs, Nucleosides, Peptides and Heterocycles

Our team is specialized in chemistry of nucleosides, nucleotides, peptides and heterocycles, which is used to generate molecules with desired physical or biological properties in order to better understand or inhibit biological processes. More recently, the team has reinforced is expertise in chemistry of nucleic acids to obtain synthetic RNAs and has acquired new expertise in β-lactamine chemistry. The molecules and biomolecules synthesized are used i) to explore the catalytic mechanism of transferases involved in the cell wall synthesis of bacteria  ii) to study transferases involved in epitranscriptomic events, iii) as tools for structural studies of enzymes. The different projects are presented below :

Chemistry of RNAs :

Development of new methodologies for post-functionalization of RNAs. Using our methodologies, we were able to synthesized :

– Peptidyl-RNA conjugates for the study of FmhB of Staphyloccocus Aureus

– Stable aminoacyl-tRNA analogues to explore non ribosomal peptide synthesis processes.

– RNA-SAM cofactor conjugates to study  m6A-RNA methyltransferases.

– Development of Nanospectroscopy for mapping RNA profile in Tumor-educated blood platelets.

Chemistry of Peptides

We  synthezise peptidoglycan fragments to study L,D- transpeptidases enzymes involved in cell wall synthesis of Mycobacterium Tuberculosis.

 

Chemistry of Heterocycles

Development of new chemistry for the synthesis of carbapenem or avibactam analogues in order to inhibit or study the cell wall synthesis of bacteria. Development of selective inhibitors of FAK kinase is also one of our current projects.

All of these projects are at the interface between chemistry and biology and benefit from collaboration at the local, national and international levels.

Permanent Members

Group leader

Members

Main publications

(click here for all publications)

1. Y. S. Polikanov, M. Etheve-Quelquejeu, R. Micura, “Synthesis of Peptidyl-tRNA Mimics for Structural Biology Applications”Accounts of Chemical Research, 2023, doi-org.ezproxy.u-paris.fr/10.1021

2. L. Iannazzo, E. Braud, C. Atdjian,  M. Ethève-Quelquejeu & al., Synthesis of RNA-cofactor conjugates and structural exploration of RNA recognition by an m6A RNA methyltransferase, Nucleic Acids Research, 2022, gkac354, https://doi.org/10.1093/nar/gkac354

3. S. Saidjalolov, E. Braud, L. Iannazzo, M. Etheve-Quelquejeu & al., Click and Release Chemistry for Activity-based Purification of b-lactam targets, Chem. Eur. J., 2021, DOI:10.1002/chem.202100653

4. C. Kitoun, M. Etheve-Quelquejeu, L. Iannazzo & al. Phosphine-Mediated Bioconjugation of 3’-end of RNA,  Org. Lett. 2020, DOI:10.1021/acs.orglett.0c02982.

5. F. Bouchet, H. Atze & al. Diazabicyclooctane functionalization for inhibition of β-lactamases from enterobacteria, Journal of Medicinal Chemistry,  2020, 63, 10, 5257–5273  https://doi.org/10.1021/acs.jmedchem.9b02125

6. C. Atdjian, L. Iannazzo, E. Braud & al. Synthesis of SAM-adenosine conjugates for the study of m6A-RNA methyltransferases Eur. J. Org. Chem., 2018, 4411-4425.

Supramolecular Bio-inorganic Chemistry

 

Context: In the biological world, proteins act as highly efficient and selective receptors. Recognition processes are based on multiple non-covalent interactions. However, many proteins also contain metal ions that can be directly involved in recognition processes or even act as a catalyst leading to the selective transformation of an organic substrate. In enzymes, the control of the metallo-site is due to the structuring of the protein backbone in order to not only preorganize the coordination site for the metal ion, but also provide a cavity and a corridor connecting it to the bulk. All these features lead to remarkable control of the binding of exogenous molecules and the reactivity of the metal ion.

Interest: We are interested in developing supramolecular models that will allow the control of the first and the second coordination spheres as well as the substrate access channel that selects and drives the substrate to the metal center, and expels the product. Our strategies consist in:

i) The covalent linkage of a coordination site, which will reproduce the natural core provided by the amino acid residues found in the enzymes, to a hydrophobic cavity that will protect the metal center and play the role of the enzyme active site pocket;

ii) The encapsulation of simple biomimetic metal complexes within a supramolecular cage.

Goals:

Get key information on Nature’s strategy for controlling the reactivity of a metal ion confined in an organic pocket (active site of enzymes).

Design molecular receptors and redox probes.

Discover new reactive pathways by constraining in a well-defined cavity space the catalyst (metal ion), the reactant (small molecules such as H2O, O2, CO2) and guest substrate.

Obtain selective and efficient supramolecular catalysts.

Control other metal complexes’ properties (e.g. luminescence)

 

Key-words: Biomimetic metal complexes, Host-guest chemistry, Chirality.

Expertise: Supramolecular Chemistry, Coordination Chemistry, Biomimetic Chemistry, Macrocyclic chemistry, Calixarenes and Resorcinarenes.

Tools: Organic synthesis (functionalization of molecular hosts, synthesis of ligands); coordination chemistry of Zn, Cu, Cr; Spectroscopies (NMR, EPR, UV-vis-NIR, fluorescence, IR), mass spectrometry; cyclic voltammetry…

Permanent Members

Group leader

Publications of the team

Journal articles

2025

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Jules Bresson, Katie Burke, Mélanie Ethève‐quelquejeu, Laura Iannazzo, Kevin Cariou. Metal‐Catalyzed Cross‐Coupling for the Synthesis of β‐Lactam Drugs and Related Chemical Probes. ChemMedChem, 2025, 20 (9), pp.e202400960. ⟨10.1002/cmdc.202400960⟩. ⟨hal-05287299⟩
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Katie Burke, Quentin Herail, Ines Zerguine, Catherine Bougault, Michel Arthur, et al.. Optimization of prodrug activation by enzymatic cleavage of the β‐lactam ring of carbapenems. Chemistry - A European Journal, 2025, 31 (46), pp.e01534. ⟨10.1002/chem.202501534⟩. ⟨hal-05287283⟩
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Jianxun Du, Batoul Mahcene, Valerii Martynov, Elisa Frezza, Christelle Vasnier, et al.. Investigation of a squaramide motif as a bioisostere of the amino-acid group of S-adenosyl-L-methionine and its functional impact on RNA methylation. Communications Chemistry, 2025, 8 (1), pp.244. ⟨10.1038/s42004-025-01627-7⟩. ⟨hal-05287286v1⟩
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Jianxun Du, Bastien Felipe, Dylan Coelho, Laura Iannazzo, Alexandre David, et al.. Synthetic approaches to bis-adenosine derivatives as potential bisubstrates of RNA methyltransferases. Organic & Biomolecular Chemistry, 2025, 23 (24), pp.5887-5896. ⟨10.1039/D5OB00758E⟩. ⟨hal-05139585⟩
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Cécilia Hognon, Ameni Ben Abdeljaoued, Pierre Hardouin, Mélanie Etheve-Quelquejeu, Bruno Sargueil, et al.. A multiscale study to characterize SHAPE probe/ RNA molecules pre-reactive complex and its role in initiating the SHAPE reaction. Journal of Chemical Information and Modeling, 2025, ⟨10.1021/acs.jcim.5c00812⟩. ⟨hal-05226372⟩
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Laura Iannazzo, Emmanuelle Braud, Matthieu Fonvielle, Mélanie Etheve-Quelquejeu. Synthesis of RNA conjugates as bisubstrates for the study of transferases. Comptes Rendus. Chimie, 2025, 28 (G1), pp.111-129. ⟨10.5802/crchim.356⟩. ⟨hal-05287289⟩
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Hichem Ichou, Kevin Telliez, Sonia Lajnef, Fabienne Peyrot, Benjamin Doistau, et al.. Anion-mediated properties of a metal complex in a hexameric resorcin[4]arene cage: chirality induction, kinetics and reactivity. Inorganic Chemistry Frontiers, 2025, 12 (3), pp.1028-1039. ⟨10.1039/d4qi02896a⟩. ⟨hal-05158345⟩
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Catherine Laurent, Gabrielle Poncet, Tristan Herskovits, Rodolphe Alves de Sousa, Laurent Le Corre, et al.. Inhibition of the Parkinson’s Disease-Related Protein DJ-1 by Endogenous Neurotoxins of the 1,2,3,4-Tetrahydroisoquinoline Family. ACS Chemical Neuroscience, 2025, 16 (6), pp.1034-1042. ⟨10.1021/acschemneuro.4c00559⟩. ⟨hal-05291792⟩
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Nicolas Mathas, Emmanuelle Braud, Erwan Galardon, Lucie Larigot, Mélanie Etheve-Quelquejeu, et al.. Park7 (DJ-1), a Parkinson-associated glyoxalase/deglycase: characterization of enzymatic activity in biological samples using fluorescence-based liquid chromatography. Biochimie, 2025, 235, pp.113-121. ⟨10.1016/j.biochi.2025.06.005⟩. ⟨hal-05139644⟩
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Riccardo Piccardi, Laurent Micouin. An Overview of the Direct Preparation of Organoaluminum Compounds. Synthesis: Journal of Synthetic Organic Chemistry, In press, ⟨10.1055/a-2669-5996⟩. ⟨hal-05302402⟩
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2024

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Erica Benedetti, Laurent Micouin. Have spirocyclic scaffolds been properly utilized in recent drug discovery efforts?. Expert Opinion on Drug Discovery, 2024, 19 (3), pp.263-266. ⟨10.1080/17460441.2024.2305735⟩. ⟨hal-04736219⟩
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Jules Brom, Antoine Maruani, Serge Turcaud, Sonia Lajnef, Fabienne Peyrot, et al.. [2.2]Paracyclophane-based coumarins: effective organo-photocatalysts for light-induced desulfonylation processes. Organic & Biomolecular Chemistry, 2024, ⟨10.1039/D3OB01711G⟩. ⟨hal-04335222⟩
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Margaux Cescato, Laurence Cuisset, Laurent Le Corre, Mathieu Rodero, Sophie Georgin-Lavialle. Diagnosis traps for patients with acquired NLRP3 mutation. European Journal of Internal Medicine, 2024, 125 (16), pp.129-131. ⟨10.1016/j.ejim.2024.01.028⟩. ⟨hal-05073743⟩
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Margaux Cescato, Yixiang y J Zhu, Laurent Le Corre, Bénédicte F Py, Sophie Georgin-Lavialle, et al.. Implication of the LRR Domain in the Regulation and Activation of the NLRP3 Inflammasome. Cells, 2024, 13 (16), pp.1365. ⟨10.3390/cells13161365⟩. ⟨hal-04695751⟩
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Hugo Esteves, Tania Xavier, Sonia Lajnef, Fabienne Peyrot, Guillaume Lefèvre, et al.. Iron-Catalyzed Intramolecular C(sp 3 )-H Lactonization of Hydroxamate Derivatives Promoted by a 1,5-HAT. ACS Catalysis, 2024, 14 (6), pp.4329-4339. ⟨10.1021/acscatal.3c04900⟩. ⟨hal-04778122⟩
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Claire Fleurisson, Nessrine Graidia, Jihed Azzouz, Audrey Di Giorgio, Marc Gaysinski, et al.. Design and Evaluation of Azaspirocycles as RNA binders. Chemistry - A European Journal, 2024, 31 (5), pp.e202403518. ⟨10.1002/chem.202403518⟩. ⟨hal-05302366⟩
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Hadrien Flichot, Annika Sickinger, Jules Brom, Bertrand Lefeuvre, Vincent Dorcet, et al.. Magneto-structural correlation in lanthanide luminescent [2.2]Paracyclophane-based Single-Molecule Magnets. Dalton Transactions, 2024, 53 (19), pp.8191-8201. ⟨10.1039/d4dt00536h⟩. ⟨hal-04571100⟩
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Zhendong Peng, Laurent Royon, Yun Luo, Philippe Decorse, Sarra Gam Derouich, et al.. Eradication of planktonic bacteria by shape-tailored gold nanoparticle photothermia. Materials Advances, 2024, 21, ⟨10.1039/d4ma00821a⟩. ⟨hal-04724709⟩
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Shiqi Wu, Laurent Micouin, Erica Benedetti. Synthesis of Three-Dimensional Benzophenone Analogues Based on a [2.2]Paracyclophane Scaffold. SYNLETT, 2024, ⟨10.1055/a-2284-4984⟩. ⟨hal-04578271⟩
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Shiqi Wu, Simon Felder, Jules Brom, Fabrice Pointillart, Olivier Maury, et al.. [2.2]Paracyclophanes: From Selective Functionalization to Optical Properties. Advanced Optical Materials, 2024, 12 (21), pp.2400934. ⟨10.1002/adom.202400934⟩. ⟨hal-04614001⟩
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Tuan Zhao, Emmanuelle Sachon, Laurent Micouin, Riccardo Piccardi. α‐Silylated Diazoalkynes: New Tools for Bioconjugation of Proteins. Chemistry - A European Journal, 2024, 30 (19), pp.2042-2048. ⟨10.1002/chem.202302807⟩. ⟨hal-04762411⟩
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2023

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Leeroy Baron, Justine Hadjerci, Leishemba Thoidingjam, Marina Plays, Romain Bucci, et al.. PSL Chemical Biology Symposia Third Edition: A Branch of Science in its Explosive Phase. ChemBioChem, 2023, 24 (8), pp.e202300093. ⟨10.1002/cbic.202300093⟩. ⟨hal-04092530⟩
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Jules Brom, Antoine Maruani, Laurent Micouin, Erica Benedetti. Light-Driven Reductive Cleavage of Sulfonamides Promoted by Thiourea Organophotosensitizers. Journal of Organic Chemistry, 2023, 88 (9), pp.5923-5935. ⟨10.1021/acs.joc.3c00296⟩. ⟨hal-04267371⟩
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Dylan Coelho, Laurent Le Corre, Karolina Bartosik, Laura Iannazzo, Emmanuelle Braud, et al.. Synthesis of Bisubstrate Analogues for RNA Methylation Studies using two Transition‐Metal‐Catalyzed Reactions. Chemistry - A European Journal, 2023, 29 (44), ⟨10.1002/chem.202301134⟩. ⟨hal-04246592⟩
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Ivan Corbeski, Pablo Andrés Vargas-Rosales, Rajiv Kumar Bedi, Jiahua Deng, Dylan Coelho, et al.. The catalytic mechanism of the RNA methyltransferase METTL3. eLife, 2023, ⟨10.7554/eLife.92537.1⟩. ⟨hal-05287291⟩
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Antoine Fayand, Margaux Cescato, Laurent Le Corre, Alexandre Terré, Margaux Wacheux, et al.. Pathogenic variants in the NLRP3 LRR domain at position 861 are responsible for a boost-dependent atypical CAPS phenotype.. Journal of Allergy and Clinical Immunology, 2023, 152 (5), pp.1303-1311.e1. ⟨10.1016/j.jaci.2023.07.006⟩. ⟨hal-04182567⟩
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Antoine Fayand, Véronique Hentgen, Céline Posseme, Carole Lacout, Capucine Picard, et al.. Successful treatment of JAK1 associated inflammatory disease. Journal of Allergy and Clinical Immunology, 2023, 152 (4), pp.972-983. ⟨10.1016/j.jaci.2023.06.004⟩. ⟨hal-04137977⟩
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Simon Felder, Marie-Leonie Delcourt, Damian Contant, Rafael Rodríguez, Ludovic Favereau, et al.. Compact CPL emitters based on a [2.2]paracyclophane scaffold: recent developments and future perspectives. Journal of Materials Chemistry C, 2023, 11, pp.2053-2062. ⟨10.1039/d2tc04885j⟩. ⟨hal-04011240⟩
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Claire Fleurisson, Nessrine Graidia, Yann Foricher, Erica Benedetti, Laurent Micouin. Intramolecular Buchwald–Hartwig N -arylation of bicyclic hydrazines: practical access to spiro[indoline-2,3′-piperidines]. Organic & Biomolecular Chemistry, 2023, 21 (17), pp.3542-3546. ⟨10.1039/D3OB00406F⟩. ⟨hal-04267385⟩
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2022

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Mélanie Faria da Cunha, Iwona Pranke, Ali Sassi, Christiane Schreiweis, Stéphanie Moriceau, et al.. Systemic bis-phosphinic acid derivative restores chloride transport in Cystic Fibrosis mice. Scientific Reports, 2022, 12 (1), pp.6132. ⟨10.1038/s41598-022-09678-9⟩. ⟨hal-03662932⟩
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Simon Felder, Marie-Leonie Delcourt, Manon Bousquet, Denis Jacquemin, Rafael Rodriguez, et al.. Planar Chiral Analogues of PRODAN Based on a [2.2]Paracyclophane Scaffold: Synthesis and Photophysical Studies. Journal of Organic Chemistry, 2022, 87 (1), pp.147-158. ⟨10.1021/acs.joc.1c02071⟩. ⟨hal-03512519⟩
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Simon Felder, Corinne Sagné, Erica Benedetti, Laurent Micouin. Small-Molecule 3D Ligand for RNA Recognition: Tuning Selectivity through Scaffold Hopping. ACS Chemical Biology, 2022, 17 (11), pp.3069-3076. ⟨10.1021/acschembio.2c00171⟩. ⟨hal-04035021⟩
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Chiara Figazzolo, Frédéric Bonhomme, Saidbakhrom Saidjalolov, Mélanie Ethève-Quelquejeu, Marcel Hollenstein. Enzymatic synthesis of vancomycin-modified DNA. Molecules, 2022, 27 (24), pp.8927. ⟨10.3390/molecules27248927⟩. ⟨hal-03927068⟩
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Ivona Krošl, Ena Otković, Ivana Nikšić-Franjić, Benoît Colasson, Olivia Reinaud, et al.. Impact of positive charge and ring-size on the interactions of calixarenes with DNA, RNA and nucleotides. New Journal of Chemistry, 2022, 46 (15), pp.6860-6869. ⟨10.1039/D2NJ00061J⟩. ⟨hal-03627557⟩
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Vincent Meynier, Laura Iannazzo, Marjorie Catala, Stephanie Oerum, Emmanuelle Braud, et al.. Synthesis of RNA-cofactor conjugates and structural exploration of RNA recognition by an m6A RNA methyltransferase. Nucleic Acids Research, 2022, ⟨10.1093/nar/gkac354⟩. ⟨hal-03689976⟩
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Khawla Nouri, Nicolas Pietrancosta, Laurent Le Corre, Patrick Dansette, Daniel Mansuy, et al.. Human Orphan Cytochrome P450 2U1 Catalyzes the ω-Hydroxylation of Leukotriene B4. International Journal of Molecular Sciences, 2022, 23 (23), pp.14615. ⟨10.3390/ijms232314615⟩. ⟨hal-03957648⟩
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Martin Oliver, Laurent Le Corre, Mélanie Poinsot, Michaël Bosco, Hongwei Wan, et al.. A Sub-Micromolar MraYAA Inhibitor with an Aminoribosyl Uridine Structure and a (S,S)-Tartaric Diamide: Synthesis, Biological Evaluation and Molecular Modeling. Molecules, 2022, 27 (6), pp.1769. ⟨10.3390/molecules27061769⟩. ⟨hal-03632451⟩
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Lauriane Rietmeyer, Inès Li de la Sierra-Gallay, Guy Schepers, Delphine Dorchêne, Laura Iannazzo, et al.. Amino-acyl tXNA as inhibitors or amino acid donors in peptide synthesis. Nucleic Acids Research, 2022, ⟨10.1093/nar/gkac1023⟩. ⟨hal-03879768⟩
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Célia Sahli, Sergio Moya, John Lomas, Christine Gravier-Pelletier, Romain Briandet, et al.. Recent advances in nanotechnology for eradicating bacterial biofilm. Theranostics, 2022, 12 (5), pp.2383-2405. ⟨10.7150/thno.67296⟩. ⟨hal-03607522⟩
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Hongwei Wan, Raja Ben Othman, Laurent Le Corre, Mélanie Poinsot, Martin Oliver, et al.. New MraYAA Inhibitors with an Aminoribosyl Uridine Structure and an Oxadiazole. Antibiotics, 2022, 11 (9), pp.1189. ⟨10.3390/antibiotics11091189⟩. ⟨hal-03805942⟩
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2021

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Emmanuelle Bardin, Alexandra Pastor, Michaela Semeraro, Anita Golec, Kate Hayes, et al.. Modulators of CFTR. Updates on clinical development and future directions. European Journal of Medicinal Chemistry, 2021, 213, pp.113195. ⟨10.1016/j.ejmech.2021.113195⟩. ⟨hal-03445073⟩
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Anais Biscotti, François Estour, Berthe-Sandra Sembo-Backonly, Sebastien Balieu, Michaël Bosco, et al.. Gd3+ Complexes Conjugated to Cyclodextrins: Hydroxyl Functions Influence the Relaxation Properties. Processes, 2021, 9 (2), pp.269. ⟨10.3390/pr9020269⟩. ⟨hal-03127005⟩
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Sara Bitam, Ahmad Elbahnsi, Geordie Creste, Iwona Pranke, Benoit Chevalier, et al.. New insights into structure and function of bis-phosphinic acid derivatives and implications for CFTR modulation. Scientific Reports, 2021, 11 (1), ⟨10.1038/s41598-021-83240-x⟩. ⟨hal-03184333⟩
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Flavie Bouchet, Heiner Atze, Michel Arthur, Mélanie Ethève-Quelquejeu, Laura Iannazzo. Traceless Staudinger Ligation To Introduce Chemical Diversity on β-Lactamase Inhibitors of Second Generation. Organic Letters, 2021, 23 (20), pp.7755-7758. ⟨10.1021/acs.orglett.1c02741⟩. ⟨hal-03647098⟩
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Alessandra Corio, Christine Gravier-Pelletier, Patricia Busca. Regioselective Functionalization of Quinolines through C-H Activation: A Comprehensive Review. Molecules, 2021, 26 (18), pp.5467. ⟨10.3390/molecules26185467⟩. ⟨hal-03445072⟩
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Aurore Dumond, Etienne Brachet, Jérôme Durivault, Valérie Vial, Anna Puszko, et al.. Neuropilin 1 and Neuropilin 2 gene invalidation or pharmacological inhibition reveals their relevance for the treatment of metastatic renal cell carcinoma. Journal of experimental & clinical cancer research, 2021, 40, pp.33. ⟨10.1186/s13046-021-01832-x⟩. ⟨hal-03132345⟩
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Simon Felder, Laurent Micouin, Erica Benedetti. Para‐Functionalization of N‐Substituted 4‐amino[2.2]paracyclophanes by Regioselective Formylation. European Journal of Organic Chemistry, 2021, pp.4015. ⟨10.1002/ejoc.202100288⟩. ⟨hal-03297447⟩
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Simon Felder, Shiqi Wu, Jules Brom, Laurent Micouin, Erica Benedetti. Enantiopure planar chiral [2.2]paracyclophanes: Synthesis and applications in asymmetric organocatalysis. Chirality, 2021, 33 (9), pp.506-527. ⟨10.1002/chir.23335⟩. ⟨hal-03366196⟩
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Georgina Kirby, Laurence Grimaud, Maxime Vitale, Guillaume Prestat, Farouk Berhal. Iron(II)-catalyzed intermolecular aziridination of alkenes employing hydroxylamine derivatives as clean nitrene sources. Green Chemistry, 2021, 23 (23), pp.9428-9432. ⟨10.1039/d1gc03495b⟩. ⟨hal-03588341⟩
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Camélia Kitoun, Matthieu Fonvielle, Michel Arthur, Mélanie Etheve‐quelquejeu, Laura Iannazzo. Traceless Staudinger Ligation for Bioconjugation of RNA. Current Protocols, 2021, 1 (2), ⟨10.1002/cpz1.42⟩. ⟨hal-03647120⟩
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Martin Oliver, Laurent Le Corre, Mélanie Poinsot, Alessandra Corio, Léa Madegard, et al.. Synthesis, biological evaluation and molecular modeling of urea-containing MraY inhibitors. Organic & Biomolecular Chemistry, 2021, 19 (26), pp.5844-5866. ⟨10.1039/D1OB00710F⟩. ⟨hal-03432617⟩
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Claire Pujol, Anne Legrand, Livia Parodi, Priscilla Thomas, Fanny Mochel, et al.. Implication of folate deficiency in CYP2U1 loss of function. Journal of Experimental Medicine, 2021, 218 (11), pp.e20210846. ⟨10.1084/jem.20210846⟩. ⟨pasteur-03349041⟩
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Lauriane Rietmeyer, Nicolas Fix-Boulier, Chloé Le Fournis, Laura Iannazzo, Camelia Kitoun, et al.. Partition of tRNAGly isoacceptors between protein and cell-wall peptidoglycan synthesis in Staphylococcus aureus. Nucleic Acids Research, 2021, 49 (2), pp.684-699. ⟨10.1093/nar/gkaa1242⟩. ⟨hal-03201622⟩
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Saidbakhrom Saidjalolov, Zainab Edoo, Matthieu Fonvielle, Louis Mayer, Laura Iannazzo, et al.. Synthesis of carbapenems containing peptidoglycanmimetics and inhibition of the cross-linking activity of a transpeptidase of the L,D specificity. Chemistry - A European Journal, 2021, 27 (10), pp.3542-3551. ⟨10.1002/chem.202004831⟩. ⟨hal-03184204⟩
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Saidbakhrom Saidjalolov, Emmanuelle Braud, Zainab Edoo, Laura Iannazzo, Filippo Rusconi, et al.. Click and Release Chemistry for Activity-Based Purification of β-Lactam Targets. Chemistry - A European Journal, 2021, 27 (28), pp.7687-7695. ⟨10.1002/chem.202100653⟩. ⟨hal-03281379⟩
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Shiqi Wu, Laura Abad Galán, Margaux Roux, François Riobé, Boris Le Guennic, et al.. Tuning the excited state properties of [2.2]paracyclophane-based antennas to ensure efficient sensitization of lanthanide ions or singlet oxygen generation. Inorganic Chemistry, 2021, 60 (60), pp.21. ⟨10.1021/acs.inorgchem.1c01986⟩. ⟨hal-03407500⟩
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Tongtong Zhang, Laurent Le Corre, Olivia Reinaud, Benoit Colasson. A Promising Approach for Controlling the Second Coordination Sphere of Biomimetic Metal Complexes: Encapsulation in a Dynamic Hydrogen‐Bonded Capsule. Chemistry - A European Journal, 2021, 27 (1), pp.434-443. ⟨10.1002/chem.202004370⟩. ⟨hal-03154347⟩
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2020

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Colette Atdjian, Dylan Coelho, Laura Iannazzo, Mélanie Etheve-Quelquejeu, Emmanuelle Braud. Synthesis of triazole-linked SAM-adenosine 2 conjugates: functionalization of adenosine at N-1 or N-6 position without protecting groups. Molecules, 2020, 25 (14), pp.3241. ⟨10.3390/molecules25143241⟩. ⟨hal-02915430⟩
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Céline Aubry, Paolo Clerici, Claude Gerbaud, Laurent Micouin, Jean-Luc Pernodet, et al.. Revised structure of anthelvencin A and characterization of the anthelvencin biosynthetic gene cluster. ACS Chemical Biology, 2020, ⟨10.1021/acschembio.9b00960⟩. ⟨hal-02502312⟩
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Jonah Kailer Aw, Kevin Christopher Boellaard, Teck Kiang Tan, John Yap, Yi Ping Loh, et al.. Interacting with Three-Dimensional Molecular Structures Using an Augmented Reality Mobile App. Journal of Chemical Education, 2020, 97 (10), pp.3877-3881. ⟨10.1021/acs.jchemed.0c00387⟩. ⟨hal-03154348⟩
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Michaël Bosco, Marjorie Damian, Vinay Chauhan, Mélanie Roche, Pierre Guillet, et al.. Biotinylated non-ionic amphipols for GPCR ligands screening. Methods, 2020, 180, pp.69 - 78. ⟨10.1016/j.ymeth.2020.06.001⟩. ⟨hal-03009212v2⟩
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Michaël Bosco, Su-Jin Paik, Patricia Busca, Stuart E H Moore, Christine Gravier-Pelletier. Synthetic Route to Glycosyl β-1C-(phosphino)-phosphonates as Unprecedented Stable Glycosyl Diphosphate Analogs and Their Preliminary Biological Evaluation. Molecules, 2020, 25 (21), pp.4969. ⟨10.3390/molecules25214969⟩. ⟨hal-03030819⟩
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Flavie Bouchet, Heiner Atze, Matthieu Fonvielle, Zainab Edoo, Michel Arthur, et al.. Diazabicyclooctane Functionalization for Inhibition of β-Lactamases from Enterobacteria. Journal of Medicinal Chemistry, 2020, 63 (10), pp.5257-5273. ⟨10.1021/acs.jmedchem.9b02125⟩. ⟨hal-03646829v2⟩
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Sandra Abi Fayssal, Alessandro Giungi, Farouk Berhal, Guillaume Prestat. Iron-Catalyzed Intra-intermolecular Aminoazidation of Alkenes. Organic Process Research and Development, 2020, 24 (5), pp.695-703. ⟨10.1021/acs.oprd.9b00400⟩. ⟨hal-03667879⟩
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Jeanne Fichez, Cathia Soulié, Laurent Le Corre, Sophie Sayon, Stéphane Priet, et al.. Discovery, SAR study and ADME properties of methyl 4-amino-3-cyano-1-(2-benzyloxyphenyl)-1 H -pyrazole-5-carboxylate as an HIV-1 replication inhibitor. RSC Medicinal Chemistry, 2020, 11 (5), pp.577-582. ⟨10.1039/D0MD00025F⟩. ⟨hal-03030936⟩
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Claire Fleurisson, Erica Benedetti, Laurent Micouin. Cyclic cis-1,3-Diamines Derived from Bicyclic Hydrazines: Synthesis and Applications. SYNLETT, 2020, ⟨10.1055/s-0040-1707324⟩. ⟨hal-03003668⟩
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Camelia Kitoun, Matthieu Fonvielle, Nicolas Sakkas, Manon Lefresne, Fabiola Djago, et al.. Phosphine-Mediated Bioconjugation of the 3′-End of RNA. Organic Letters, 2020, 22 (20), pp.8034-8038. ⟨10.1021/acs.orglett.0c02982⟩. ⟨hal-02996863⟩
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Bo Li, Mélanie Etheve-Quelquejeu, Expédite Yen-Pon, Christiane Garbay, Huixiong Chen. Microwave-assisted synthesis of 2,5-disubstituted pyrimidine derivatives via Buchwald-Hartwig amination. Tetrahedron Letters, 2020, 61, pp.151406 -. ⟨10.1016/j.tetlet.2019.151406⟩. ⟨hal-03488531⟩
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Yun Luo, Yu Xiao, Delphine Onidas, Laura Iannazzo, Mélanie Ethève-Quelquejeu, et al.. Raman reporters derived from aryl diazonium salts for SERS encoded-nanoparticles. Chemical Communications, 2020, 56 (50), pp.6822-6825. ⟨10.1039/d0cc02842h⟩. ⟨hal-03411993⟩
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Bruno Mégarbane, Camille Gamblin, Olivier Roussel, Elodie Bouaziz-Amar, Lucie Chevillard, et al.. The neurobehavioral effects of the designer drug naphyrone – an experimental investigation with pharmacokinetics and concentration/effect relationship in mice. Psychopharmacology, 2020, 237 (7), pp.1943-1957. ⟨10.1007/s00213-020-05510-2⟩. ⟨hal-03823023⟩
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Alberto Ongaro, Giovanni Ribaudo, Emmanuelle Braud, Mélanie Ethève-Quelquejeu, Michele de Franco, et al.. Design and synthesis of a peptide derivative of ametantrone targeting the major groove of the d(GGCGCC) 2 palindromic sequence. New Journal of Chemistry, 2020, 44 (9), pp.3624-3631. ⟨10.1039/C9NJ03817E⟩. ⟨hal-03689989⟩
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2019

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Usama Ashraf, Laura Tengo, Laurent Le Corre, Guillaume Fournier, Patricia Busca, et al.. Destabilization of the human RED–SMU1 splicing complex as a basis for host-directed antiinfluenza strategy. Proceedings of the National Academy of Sciences of the United States of America, 2019, 116 (22), pp.10968-10977. ⟨10.1073/pnas.1901214116⟩. ⟨hal-02160991⟩
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Luisa Alessandra Atehortua-Martinez, Cyriaque Masniere, Patrizia Campolongo, Stéphanie Chasseigneaux, Jacques Callebert, et al.. Acute and chronic neurobehavioral effects of the designer drug and bath salt constituent 3,4-methylenedioxypyrovalerone in the rat. Journal of Psychopharmacology, 2019, 33 (3), pp.392-405. ⟨10.1177/0269881118822151⟩. ⟨hal-03860016⟩
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Luisa Alessandra Atehortua-Martinez, Cyriaque Masniere, Patrizia Campolongo, Stéphanie Chasseigneaux, Jacques Callebert, et al.. Acute and chronic neurobehavioral effects of the designer drug and bath salt constituent 3,4-methylenedioxypyrovalerone in the rat. Journal of Psychopharmacology, 2019, 33 (3), pp.392-405. ⟨10.1177/0269881118822151⟩. ⟨hal-02557840⟩
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Luisa Alessandra Atehortua-Martinez, Cyriaque Masniere, Patrizia Campolongo, Stéphanie Chasseigneaux, Jacques Callebert, et al.. Acute and chronic neurobehavioral effects of the designer drug and bath salt constituent 3,4-methylenedioxypyrovalerone in the rat. Journal of Psychopharmacology, 2019, 33 (3), pp.392-405. ⟨10.1177/0269881118822151⟩. ⟨hal-03908457⟩
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Nadia Benturquia, Lucie Chevillard, Christophe Poiré, Olivier Roussel, Camille Cohier, et al.. Is the 3,4-methylendioxypyrovalerone/mephedrone combination responsible for enhanced stimulant effects? A rat study with investigation of the effect/concentration relationships. Psychopharmacology, 2019, 236 (3), pp.891-901. ⟨10.1007/s00213-018-4962-0⟩. ⟨hal-03823031⟩
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Nadia Benturquia, Lucie Chevillard, Christophe Poiré, Olivier Roussel, Camille Cohier, et al.. Is the 3,4-methylendioxypyrovalerone/mephedrone combination responsible for enhanced stimulant effects? A rat study with investigation of the effect/concentration relationships. Psychopharmacology, 2019, 236 (3), pp.891-901. ⟨10.1007/s00213-018-4962-0⟩. ⟨hal-03860105⟩
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Nicholus Bhattacharjee, Sébastien Triboulet, Vincent Dubée, Matthieu Fonvielle, Zainab Edoo, et al.. Negative impact of carbapenem methylation on the reactivity of β-lactams for cysteine acylation revealed by quantum calculations and kinetic analyses. Antimicrobial Agents and Chemotherapy, 2019, 63 (4), pp.e02039-18. ⟨10.1128/AAC.02039-18⟩. ⟨hal-02057268⟩
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Etienne Brachet, Aurore Dumond, Wang-Qing Liu, Marie Fabre, Mohamed Selkti, et al.. Synthesis, 3D-structure and stability analyses of NRPa-308, a new promising anti-cancer agent. Bioorganic and Medicinal Chemistry Letters, 2019, 29 (24), pp.126710. ⟨10.1016/j.bmcl.2019.126710⟩. ⟨hal-02418648⟩
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Benoit Colasson, Alberto Credi, Barbara Ventura. Photoinduced Electron Transfer Involving a Naphthalimide Chromophore in Switchable and Flexible [2]Rotaxanes. Chemistry - A European Journal, 2019, 26 (2), pp.534-542. ⟨10.1002/chem.201904155⟩. ⟨hal-03154349⟩
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Marie-Leonie Delcourt, Simon Felder, Serge Turcaud, Corina Pollok, Christian Merten, et al.. Highly Enantioselective Asymmetric Transfer Hydrogenation: A Practical and Scalable Method To Efficiently Access Planar Chiral [2.2]Paracyclophanes. Journal of Organic Chemistry, 2019, ⟨10.1021/acs.joc.9b00372⟩. ⟨hal-02113386⟩
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Marie-Leonie Delcourt, Corentin Reynaud, Serge Turcaud, Ludovic Favereau, Jeanne Crassous, et al.. 3D Coumarin Systems Based on [2.2]Paracyclophane Synthesis, Spectroscopic Characterization, and Chiroptical Properties. Journal of Organic Chemistry, 2019, 84 (2), pp.888-899. ⟨10.1021/acs.joc.8b02773⟩. ⟨hal-02049506⟩
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Ahmad Massarweh, Michael Bosco, Isabelle Chantret, Thibaut Léger, Layla Jamal, et al.. Bacterial Lipid II Analogs: Novel In Vitro Substrates for Mammalian Oligosaccharyl Diphosphodolichol Diphosphatase (DLODP) Activities. Molecules, 2019, 24 (11), pp.2135. ⟨10.3390/molecules24112135⟩. ⟨hal-02172947⟩
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Stephanie Oerum, Marjorie Catala, Colette Atdjian, Franck Brachet, Luc Ponchon, et al.. Bisubstrate analogues as structural tools to investigate m 6 A methyltransferase active sites. RNA Biology, 2019, 16 (6), pp.798-808. ⟨10.1080/15476286.2019.1589360⟩. ⟨hal-02353503⟩
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Tuan Zhao, Laurent Micouin, Riccardo Piccardi. Synthesis of Organometallic Compounds in Flow. Helvetica Chimica Acta, 2019, 102 (11), ⟨10.1002/hlca.201900172⟩. ⟨hal-02346965⟩
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2018

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Colette Atdjian, Laura Iannazzo, Emmanuelle Braud, Mélanie Ethève-Quelquejeu. Synthesis of SAM-Adenosine Conjugates for the Study of m 6 A-RNA Methyltransferases. European Journal of Organic Chemistry, 2018, 2018 (32), pp.4411-4425. ⟨10.1002/ejoc.201800798⟩. ⟨hal-03647207⟩
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Colette Atdjian, Laura Iannazzo, Emmanuelle Braud, Mélanie Ethève-Quelquejeu. Synthesis of SAM-Adenosine Conjugates for the Study of m 6 A-RNA Methyltransferases. European Journal of Organic Chemistry, 2018, 2018 (32), pp.4411-4425. ⟨10.1002/ejoc.201800798⟩. ⟨hal-02353523⟩
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Colette Atdjian, Laura Iannazzo, Emmanuelle Braud, Mélanie Ethève-Quelquejeu. Synthesis of SAM-Adenosine Conjugates for the Study of m 6 A-RNA Methyltransferases. European Journal of Organic Chemistry, 2018, 2018 (32), pp.4411-4425. ⟨10.1002/ejoc.201800798⟩. ⟨hal-03689993⟩
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Nadia Benturquia, Lucie Chevillard, Christophe Poiré, Olivier Roussel, Camille Cohier, et al.. Is the 3,4-methylendioxypyrovalerone/mephedrone combination responsible for enhanced stimulant effects? A rat study with investigation of the effect/concentration relationships. Psychopharmacology, 2018, ⟨10.1007/s00213-018-4962-0⟩. ⟨hal-01899917⟩
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Aurélie Blond, Serge Turcaud, Thomas Lecourt, Laurent Micouin. Diastereoselective Ring Homologation of Bicyclic Hydrazines: Access to cis -1,3-Diaminocyclohexitols. ACS Omega, 2018, 3 (11), pp.15302-15307. ⟨10.1021/acsomega.8b02910⟩. ⟨hal-02186751⟩
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Marie-Leonie Delcourt, Simon Felder, Erica Benedetti, Laurent Micouin. Highly Enantioselective Desymmetrization of Centrosymmetric pseudo - para -Diformyl[2.2]paracyclophane via Asymmetric Transfer Hydrogenation. ACS Catalysis, 2018, 8 (7), pp.6612-6616. ⟨10.1021/acscatal.8b01872⟩. ⟨hal-02113395⟩
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Zainab Edoo, Laura Iannazzo, Fabrice Compain, Inès Li de La Sierra Gallay, Herman Van Tilbeurgh, et al.. Synthesis of Avibactam Derivatives and Activity on β-Lactamases and Peptidoglycan Biosynthesis Enzymes of Mycobacteria. Chemistry - A European Journal, 2018, 24 (32), pp.8081--8086. ⟨10.1002/chem.201800923⟩. ⟨hal-02177911⟩
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Mickaël Fer, Laurent Le Corre, Nicolas Pietrancosta, Nathalie Evrard-Todeschi, Samir Olatunji, et al.. Bacterial Transferase MraY, a Source of Inspiration towards New Antibiotics. Current Medicinal Chemistry, 2018, 25 (42), pp.6013-6029. ⟨10.2174/0929867325666180330095154⟩. ⟨hal-02364241⟩
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Matthieu Fonvielle, Ahmed Bouhss, Coralie Hoareau, Delphine Patin, Dominique Mengin-Lecreulx, et al.. Synthesis of lipid-carbohydrate-peptidyl-RNA conjugates to explore the limits imposed by the substrate specificity of cell wall enzymes on the acquisition of drug resistance. Chemistry - A European Journal, 2018, 24 (56), pp.14911-14915. ⟨10.1002/chem.201802360⟩. ⟨hal-01962025⟩
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Laura Iannazzo, Matthieu Fonvielle, Emmanuelle Braud, Hubert Hřebabecký, Eliška Procházková, et al.. Synthesis of tRNA analogues containing a terminal ribose locked in the South conformation to study tRNA-dependent enzymes. Organic & Biomolecular Chemistry, 2018, 16 (11), pp.1903-1911. ⟨10.1039/C8OB00019K⟩. ⟨hal-03689994⟩
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Alex Inthasot, Nicolas Le Poul, Michel Luhmer, Benoit Colasson, Ivan Jabin, et al.. Selective EPR Detection of Primary Amines in Water with a Calix[6]azacryptand-Based Copper(II) Funnel Complex. Inorganic Chemistry, 2018, ⟨10.1021/acs.inorgchem.7b02541⟩. ⟨hal-01679879⟩
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Nicolas Le Poul, Benoit Colasson, Grégory Thiabaud, Dany Jeanne Dit Fouque, Claudio Iacobucci, et al.. Gating the electron transfer at a monocopper centre through the supramolecular coordination of water molecules within a protein chamber mimic. Chemical Science, 2018, 9 (43), pp.8282-8290. ⟨10.1039/C8SC03124J⟩. ⟨hal-01874257⟩
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Nicolas Le Poul, Benoit Colasson, Grégory Thiabaud, Dany Jeanne Dit Fouque, Claudio Iacobucci, et al.. Gating the electron transfer at a monocopper centre through the supramolecular coordination of water molecules within a protein chamber mimic. Chemical Science, 2018, 9 (43), pp.8282-8290. ⟨10.1039/C8SC03124J⟩. ⟨hal-03824727⟩
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Anne-Doriane Manick, Sidonie Aubert, Boubacar Yalcouye, Thierry Prangé, Farouk Berhal, et al.. Access to Functionalized Imidazolidin-2-one Derivatives by Iron-Catalyzed Oxyamination of Alkenes. Chemistry - A European Journal, 2018, 24 (44), pp.11485-11492. ⟨10.1002/chem.201802190⟩. ⟨hal-03710267⟩
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Anne-Doriane Manick, Farouk Berhal, Guillaume Prestat. Development of a One-Pot Four C–C Bond-Forming Sequence Based on Palladium/Ruthenium Tandem Catalysis. Organic Letters, 2018, 20 (1), pp.194-197. ⟨10.1021/acs.orglett.7b03556⟩. ⟨hal-03710509⟩
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Cécile Morlot, Daniel Straume, Katharina Peters, Olav A Hegnar, Nolwenn Simon, et al.. Structure of the essential peptidoglycan amidotransferase MurT/GatD complex from Streptococcus pneumoniae. Nature Communications, 2018, 9, pp.3180. ⟨10.1038/s41467-018-05602-w⟩. ⟨hal-01861372⟩
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Flora Ngadjeua, Emmanuelle Braud, Saidbakhrom Saidjalolov, Laura Iannazzo, Dirk Schnappinger, et al.. Critical Impact of Peptidoglycan Precursor Amidation on the Activity of l,d -Transpeptidases from Enterococcus faecium and Mycobacterium tuberculosis. Chemistry - A European Journal, 2018, 24 (22), pp.5743 - 5747. ⟨10.1002/chem.201706082⟩. ⟨hal-01817697⟩
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Flora Ngadjeua, Emmanuelle Braud, Saidbakhrom Saidjalolov, Laura Iannazzo, Dirk Schnappinger, et al.. Critical Impact of Peptidoglycan Precursor Amidation on the Activity of l,d -Transpeptidases from Enterococcus faecium and Mycobacterium tuberculosis. Chemistry - A European Journal, 2018, 24 (22), pp.5743-5747. ⟨10.1002/chem.201706082⟩. ⟨hal-03647180⟩
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Riccardo Piccardi, Serge Turcaud, Erica Benedetti, Laurent Micouin. Synthesis and Reactivity of Mixed Dimethylalkynylaluminum Reagents. Synthesis: Journal of Synthetic Organic Chemistry, 2018, 51 (01), pp.97-106. ⟨10.1055/s-0037-1610392⟩. ⟨hal-02113388⟩
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Giulio Ragazzon, Christian Schäfer, Paola Franchi, Serena Silvi, Benoit Colasson, et al.. Remote electrochemical modulation of pK a in a rotaxane by co-conformational allostery. Proceedings of the National Academy of Sciences of the United States of America, 2018, 115 (38), pp.9385-9390. ⟨10.1073/pnas.1712783115⟩. ⟨hal-03154351⟩
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Expédite Yen-Pon, Bo Li, Marta Acebrón-Garcia-De-Eulate, Céline Tomkiewicz-Raulet, John Dawson, et al.. Structure-Based Design, Synthesis, and Characterization of the First Irreversible Inhibitor of Focal Adhesion Kinase. ACS Chemical Biology, 2018, 13 (8), pp.2067-2073. ⟨10.1021/acschembio.8b00250⟩. ⟨hal-02196326⟩
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Tuan Zhao, Riccardo Piccardi, Laurent Micouin. Rapid and Effective Synthesis of α-Acyloxy-α-alkynyltrimethylsilanes. Organic Letters, 2018, 20 (16), pp.5015-5018. ⟨10.1021/acs.orglett.8b02165⟩. ⟨hal-02113392⟩
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2017

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E. Benedetti, M.-L. Delcourt, B. Gatin-Fraudet, S. Turcaud, L. Micouin. Synthesis and photophysical studies of through-space conjugated [2.2]paracyclophane-based naphthalene fluorophores. RSC Advances, 2017, 7 (80), pp.50472-50476. ⟨10.1039/C7RA10038H⟩. ⟨hal-02113405⟩
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Michaël Bosco, Ahmad Massarweh, Soria Iatmanen-Harbi, Ahmed Bouhss, Isabelle Chantret, et al.. Synthesis and biological evaluation of chemical tools for the study of Dolichol Linked Oligosaccharide Diphosphatase (DLODP).. European Journal of Medicinal Chemistry, 2017, 125, pp.952-964. ⟨10.1016/j.ejmech.2016.10.013⟩. ⟨hal-01440749⟩
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Hélène Guyon, François Mavré, Marjorie Catala, Serge Turcaud, Franck Brachet, et al.. Use of a redox probe for an electrochemical RNA–ligand binding assay in microliter droplets. Chemical Communications, 2017, 53 (6), pp.1140-1143. ⟨10.1039/c6cc07785d⟩. ⟨hal-02185366⟩
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Alex Inthasot, Nicolas Le Poul, Michel Luhmer, Benoit Colasson, Ivan Jabin, et al.. Selective EPR Detection of Primary Amines in Water with a Calix[6]azacryptand-Based Copper(II) Funnel Complex. Inorganic Chemistry, 2017, 57 (7), pp.3646-3655. ⟨10.1021/acs.inorgchem.7b02541⟩. ⟨hal-03154352⟩
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Antoine Joosten, Mélissa Boultadakis-Arapinis, V. Gandon, L. Micouin, Thomas Lecourt. Substitution of the Participating Group of Glycosyl Donors by a Halogen Atom: Influence on the Rearrangement of Transient Orthoesters Formed during Glycosylation Reactions. Journal of Organic Chemistry, 2017, 82 (6), pp.3291-3297. ⟨10.1021/acs.joc.6b03088⟩. ⟨hal-02046285⟩
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Sophie Letort, Michaël Bosco, Benedetta Cornelio, Frédérique Brégier, Sébastien Daulon, et al.. Structure-efficiency relationships of cyclodextrin scavengers in the hydrolytic degradation of organophosphorus compounds. Beilstein Journal of Organic Chemistry, 2017, 13, pp.417-427. ⟨10.3762/bjoc.13.45⟩. ⟨hal-02046294⟩
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Zhongyi Mao, Elisabetta Martini, Guillaume Prestat, Julie Oble, Pei-Qiang Huang, et al.. Analogues of the 2-carboxyl-6-hydroxyoctahydroindole (CHOI) unit from diverging Pd-catalyzed allylations: Selectivity as a function of the double bond position. Tetrahedron Letters, 2017, 58 (44), pp.4174-4178. ⟨10.1016/j.tetlet.2017.09.046⟩. ⟨hal-01675514⟩
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Giulio Ragazzon, Alberto Credi, Benoit Colasson. Thermodynamic Insights on a Bistable Acid-Base Switchable Molecular Shuttle with Strongly Shifted Co-conformational Equilibria. Chemistry - A European Journal, 2017, 23 (9), pp.2149-2156. ⟨10.1002/chem.201604783⟩. ⟨hal-03154354⟩
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Manal Sarkis, Maria Miteva, Maria Chiara Dasso Lang, Maryse Jaouen, Marie-Agnès Sari, et al.. Insights into the interaction of high potency inhibitor IRC-083864 with phosphatase CDC25. Proteins: Structure, Function, and Bioinformatics, 2017, 85 (4), pp.593-601. ⟨10.1002/prot.25236⟩. ⟨hal-03684762⟩
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Manal Sarkis, Maria Miteva, Maria Chiara Dasso Lang, Maryse Jaouen, Marie-Agnès Sari, et al.. Insights into the interaction of high potency inhibitor IRC-083864 with phosphatase CDC25. Proteins: Structure, Function, and Bioinformatics, 2017, 85 (4), pp.593-601. ⟨10.1002/prot.25236⟩. ⟨hal-03689998⟩
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2016

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Karen Amirbekyan, Nicolas Duchemin, Erica Benedetti, Rinah Joseph, Aude Colon, et al.. Design, Synthesis, and Binding Affinity Evaluation of Hoechst 33258 Derivatives for the Development of Sequence-Specific DNA-Based Asymmetric Catalysts. ACS Catalysis, 2016, 6 (5), pp.3096-3105. ⟨10.1021/acscatal.6b00495⟩. ⟨hal-02197253⟩
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Benoit Colasson, Alberto Credi, Giulio Ragazzon. Light-driven molecular machines based on ruthenium(II) polypyridine complexes: Strategies and recent advances. Coordination Chemistry Reviews, 2016, 325, pp.125-134. ⟨10.1016/j.ccr.2016.02.012⟩. ⟨hal-03154358⟩
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Thibaut Courant, Rahul Kumar, Serge Turcaud, Laurent Micouin. Rhodium(II)-Alkynyl Carbenoids Insertion into Si–H bonds: An Entry to Propargylic Geminal Bis(silanes). Organic Letters, 2016, 18 (19), pp.4818-4820. ⟨10.1021/acs.orglett.6b02264⟩. ⟨hal-02186746⟩
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Nicolas Duchemin, Erica Benedetti, Lucas Bethge, Stefan Vonhoff, Sven Klussmann, et al.. Expanding biohybrid-mediated asymmetric catalysis into the realm of RNA. Chemical Communications, 2016, 52 (55), pp.8604-8607. ⟨10.1039/c6cc03540j⟩. ⟨hal-02197262⟩
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Matthieu Fonvielle, Nicolas Sakkas, Laura Iannazzo, Chloé Le fournis, Delphine Patin, et al.. Electrophilic RNA for Peptidyl-RNA Synthesis and Site-Specific Cross-Linking with tRNA-Binding Enzymes.. Angewandte Chemie International Edition, 2016, 55 (43), pp.13553-13557. ⟨10.1002/anie.201606843⟩. ⟨hal-01440830⟩
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Alex Inthasot, Emilio Brunetti, Manuel Lejeune, Nicolas Menard, Thierry Prangé, et al.. Kinetic and Thermodynamic Stabilization of Metal Complexes by Introverted Coordination in a Calix[6]azacryptand. Chemistry - A European Journal, 2016, 22 (14), pp.4855-4862. ⟨10.1002/chem.201505057⟩. ⟨hal-03154357⟩
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Ahmad Massarweh, Michaël Bosco, Soria Iatmanen-Harbi, Clarice Tessier, Nicolas Auberger, et al.. Demonstration of an oligosaccharide-diphosphodolichol diphosphatase activity whose subcellular localization is different than those of dolichyl-phosphate-dependent enzymes of the dolichol cycle. Journal of Lipid Research, 2016, 57 (6), pp.1029-1042. ⟨10.1194/jlr.M067330⟩. ⟨hal-02997964⟩
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Riccardo Piccardi, Anaïs Coffinet, Erica Benedetti, Serge Turcaud, Laurent Micouin. Continuous Flow Synthesis of Dimethylalkynylaluminum Reagents. Synthesis: Journal of Synthetic Organic Chemistry, 2016, 48 (19), pp.3272-3278. ⟨10.1055/s-0035-1561484⟩. ⟨hal-02134269⟩
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Christian Schäfer, Giulio Ragazzon, Benoit Colasson, Marcello La rosa, Serena Silvi, et al.. An Artificial Molecular Transporter. ChemistryOpen, 2016, 5 (2), pp.120-124. ⟨10.1002/open.201500217⟩. ⟨hal-03154356⟩
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2015

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Erica Benedetti, Nicolas Duchemin, Lucas Bethge, Stefan Vonhoff, Sven Klussmann, et al.. DNA-cellulose: an economical, fully recyclable and highly effective chiral biomaterial for asymmetric catalysis. Chemical Communications, 2015, 51 (28), pp.6076-6079. ⟨10.1039/C4CC10190A⟩. ⟨hal-03554623⟩
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Pierre-Edouard Danjou, Gael de Leener, Damien Cornut, Steven Moerkerke, Samir Mameri, et al.. Supramolecular Assistance for the Selective Demethylation of Calixarene-Based Receptors. Journal of Organic Chemistry, 2015, 80 (10), pp.5084-5091. ⟨10.1021/acs.joc.5b00464⟩. ⟨hal-02865837⟩
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P. Dao, N. Smith, Daniel Scott-Algara, C. Garbay, J.P. Herbeuval, et al.. Restoration of TRAIL-induced apoptosis in resistant human pancreatic cancer cells by a novel FAK inhibitor, PH11. Cancer Letters, 2015, 360 (1), pp.48-59. ⟨10.1016/j.canlet.2015.02.016⟩. ⟨pasteur-02573704⟩
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Mickaël J Fer, Ahmed Bouhss, Mariana Patrão, Laurent Le Corre, Nicolas Pietrancosta, et al.. 5'-Methylene-triazole-substituted-aminoribosyl uridines as MraY inhibitors: synthesis, biological evaluation and molecular modeling.. Organic & Biomolecular Chemistry, 2015, 13 (26), pp.7193-222. ⟨10.1039/c5ob00707k⟩. ⟨hal-01433063⟩
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Laura Iannazzo, Erica Benedetti, Marjorie Catala, Mélanie Etheve-Quelquejeu, Carine Tisné, et al.. Monitoring of reversible boronic acid–diol interactions by fluorine NMR spectroscopy in aqueous media. Organic & Biomolecular Chemistry, 2015, 13 (33), pp.8817-8821. ⟨10.1039/c5ob01362c⟩. ⟨hal-03544508⟩
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Nicolas Le Poul, Benoit Colasson. Electrochemically and Chemically Induced Redox Processes in Molecular Machines. ChemElectroChem, 2015, 2 (4), pp.475. ⟨10.1002/celc.201402399⟩. ⟨hal-01171145⟩
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Jean-Noël Rebilly, Benoit Colasson, Olivia Bistri, Diana Over, Olivia Reinaud. Biomimetic cavity-based metal complexes. Chemical Society Reviews, 2015, 44 (2), pp.467-489. ⟨10.1039/c4cs00211c⟩. ⟨hal-03154360⟩
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Zsófia Sólyom, Peixiang Ma, Melanie Schwarten, Michaël Bosco, Ange Polidori, et al.. The Disordered Region of the HCV Protein NS5A: Conformational Dynamics, SH3 Binding, and Phosphorylation.. Biophysical Journal, 2015, 109 (7), pp.1483-96. ⟨10.1016/j.bpj.2015.06.040⟩. ⟨hal-01229755⟩
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2014

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Renaud Barbeyron, Erica Benedetti, Janine Cossy, Jean-Jacques Vasseur, Stellios Arseniyadis, et al.. Recent developments in alkyne borylations.. Tetrahedron, 2014, 70 (45), pp.8431-8452. ⟨10.1016/j.tet.2014.06.026⟩. ⟨hal-01078195⟩
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Mélissa Boultadakis-Arapinis, Vincent Gandon, Elise Prost, Laurent Micouin, Thomas Lecourt. Electronic Effects in Carbene-Mediated C H Bond Functionalization: An Experimental and Theoretical Study. Advanced Synthesis and Catalysis, 2014, 356 (11-12), pp.2493-2450. ⟨10.1002/adsc.201300984⟩. ⟨hal-01141166⟩
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Elodie Goldwaser, Benoit de Courcy, Luc Demange, Christiane Garbay, Françoise Raynaud, et al.. Conformational analysis of a polyconjugated protein-binding ligand by joint quantum chemistry and polarizable molecular mechanics. Addressing the issues of anisotropy, conjugation, polarization, and multipole transferability. Journal of Molecular Modeling, 2014, 20 (11), ⟨10.1007/s00894-014-2472-5⟩. ⟨hal-02126794⟩
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Claire Kammerer, Guillaume Prestat, David Madec, Giovanni Poli. Synthesis of γ-Lactams and γ-Lactones via Intramolecular Pd-Catalyzed Allylic Alkylations. Accounts of Chemical Research, 2014, 47 (12), pp.3439--3447. ⟨10.1021/ar500178n⟩. ⟨hal-01712373⟩
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Rahul Kumar, Serge Turcaud, Laurent Micouin. The Reaction of Dimethylalkynylaluminum Reagents with Trimethylsilyldiazomethane: Original Reactivity Leading to New α-Silylated Alkynyl Hydrazones. Organic Letters, 2014, 16 (23), pp.6192-6195. ⟨10.1021/ol503113d⟩. ⟨hal-02185384⟩
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Wang-Qing Liu, Valentino Megale, Lucia Borriello, Bertrand Leforban, Matthieu Montes, et al.. Synthesis and structure–activity relationship of non-peptidic antagonists of neuropilin-1 receptor. Bioorganic and Medicinal Chemistry Letters, 2014, 24 (17), pp.4254-4259. ⟨10.1016/j.bmcl.2014.07.028⟩. ⟨hal-02126861⟩
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Laetitia Mistico, Emel Ay, Vaizanne Huynh, Aurelie Bourderioux, Fabrice Chemla, et al.. Reactivity of tert-butanesulfinamides in palladium-catalyzed allylic substitutions. Journal of Organometallic Chemistry, 2014, 760, pp.124--129. ⟨10.1016/j.jorganchem.2013.11.026⟩. ⟨hal-01712367⟩
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Milena Opacié, Gregory Durand, Michaël Bosco, Ange Polidori, Jean-Luc Popot. Amphipols and photosynthetic light-harvesting pigment-protein complexes.. Journal of Membrane Biology, 2014, ⟨10.1007/s00232-014-9712-6⟩. ⟨hal-01332956⟩
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Jamshid Rajabi, Mélanie M. Lorion, Vu Linh Ly, Frédéric Liron, Julie Oble, et al.. Dormant versus Evolving Aminopalladated Intermediates: Toward a Unified Mechanistic Scenario in Pd ^\textrmII -Catalyzed Aminations. Chemistry - A European Journal, 2014, 20 (6), pp.1539--1546. ⟨10.1002/chem.201302744⟩. ⟨hal-01712369⟩
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Micol Rigamonti, Guillaume Prestat, Gianluigi Broggini, Giovanni Poli. Synthesis of 1,4-benzodiazepinones via palladium-catalysed allene carbopalladation/amination domino sequence. Journal of Organometallic Chemistry, 2014, 760, pp.149--155. ⟨10.1016/j.jorganchem.2013.11.010⟩. ⟨hal-01712374⟩
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2013

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Aurélie Blond, Paul Dockerty, Raquel Alvarez, Serge Turcaud, Thomas Lecourt, et al.. Modular Access to N-Substituted cis -3,5-Diaminopiperidines. Journal of Organic Chemistry, 2013, 78 (23), pp.12236-12242. ⟨10.1021/jo401994y⟩. ⟨hal-02186757⟩
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Mélissa Boultadakis-Arapinis, Elise Prost, Vincent Gandon, Pascale Lemoine, Serge Turcaud, et al.. Carbene-Mediated Functionalization of the Anomeric C-H Bond of Carbohydrates: Scope and Limitations. Chemistry - A European Journal, 2013, 19 (19), pp.6052-6066. ⟨10.1002/chem.201203725⟩. ⟨hal-02185449⟩
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Eric Leclerc, Xavier Pannecoucke, Mélanie Etheve-Quelquejeu, M. Sollogoub. Fluoro-C-glycosides and fluoro-carbasugars, hydrolytically stable and synthetically challenging glycomimetics. Chemical Society Reviews, 2013, 42 (10), pp.4270-4283. ⟨10.1039/c2cs35403a⟩. ⟨hal-00825637⟩
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Nicolas Menard, Yohann Heriot, Yves Le Mest, Olivia Reinaud, Nicolas Le Poul, et al.. Electrochemically Driven Cup-and-Ball Cu-I and Cu-II Complexes. Chemistry - A European Journal, 2013, 19 (32), pp.10611--10618. ⟨10.1002/chem.201301141⟩. ⟨hal-01175765⟩
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Sébastien Triboulet, Vincent Dubée, Lauriane Lecoq, Catherine M Bougault, Jean-Luc Mainardi, et al.. Kinetic features of L,D-transpeptidase inactivation critical for β-lactam antibacterial activity.. PLoS ONE, 2013, 8 (7), pp.e67831. ⟨10.1371/journal.pone.0067831⟩. ⟨hal-01321589⟩
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2012

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Erica Benedetti, Michela Lomazzi, Francesco Tibiletti, Jean-Philippe Goddard, Louis Fensterbank, et al.. Synthesis of Nitrogen-Containing Heterocycles via Ring-Closing Ene-Ene and Ene-Yne Metathesis Reactions: An Easy Access to 1-and 2-Benzazepine Scaffolds and Five- and Six-Membered Lactams. Synthesis: Journal of Synthetic Organic Chemistry, 2012, 44 (22), pp.3523-3533. ⟨10.1055/s-0032-1317352⟩. ⟨hal-01397631⟩
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Aurelie Jonquoy, Emilie Mugniery, Catherine Benoist-Lasselin, Nabil Kaci, Laurent Le Corre, et al.. A novel tyrosine kinase inhibitor restores chondrocyte differentiation and promotes bone growth in a gain-of-function Fgfr3 mouse model. Human Molecular Genetics, 2012, 21 (4), pp.841-851. ⟨10.1093/hmg/ddr514⟩. ⟨hal-01019795⟩
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Thomas Lombès, Roba Moumné, Valéry Larue, Elise Prost, Marjorie Catala, et al.. Investigation of RNA-Ligand Interactions by (19) F NMR Spectroscopy Using Fluorinated Probes.. Angewandte Chemie International Edition, 2012, 51 (38), pp.9530-9534. ⟨10.1002/anie.201204083⟩. ⟨hal-00724894⟩
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Roba Moumné, Marjorie Catala, Valéry Larue, Laurent Micouin, Carine Tisné. Fragment-based design of small RNA binders: promising developments and contribution of NMR.. Biochimie, 2012, 94 (7), pp.1607-1619. ⟨10.1016/j.biochi.2012.02.002⟩. ⟨hal-00692356⟩
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Eric Rose, Nicolas Raoul, Mélanie Etheve-Quelquejeu, Emma Gallo, Bernard Boitrel, et al.. Crystal structure of a chiral binaphthyl porphyrin. Journal of Porphyrins and Phthalocyanines, 2012, 16 (3), pp.324-330. ⟨10.1142/S1088424612500393⟩. ⟨hal-00863134⟩
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Grégory Thiabaud, Andrea Brugnara, Michaël Carboni, Nicolas Le Poul, Benoit Colasson, et al.. Synthesis and Studies of a Water-Soluble and Air-Stable Cu-I/Cu-II Open-Shell Funnel Complex. Organic Letters, 2012, 14 (10), pp.2500--2503. ⟨10.1021/ol3007875⟩. ⟨hal-01175768⟩
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2011

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Nicolas Auberger, Rok Frlan, Bayan Al-Dabbagh, Ahmed Bouhss, Muriel Crouvoisier, et al.. Synthesis and biological evaluation of potential new inhibitors of the bacterial transferase MraY with a β-ketophosphonate structure. Organic & Biomolecular Chemistry, 2011, 9 (24), pp.8301. ⟨10.1039/c1ob06124k⟩. ⟨hal-02188360⟩
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Tatiana Besset, Emmanuelle Braud, Rafika Jarray, Christiane Garbay, Stephanie Kolb, et al.. Preparation and evaluation of a set of bis(methoxycarbonylmethylthio) heteroquinones as CDC25B phosphatase inhibitors. Central European Journal of Chemistry, 2011, 2 (4), pp.433-440. ⟨10.5155/eurjchem.2.4.433-440.400⟩. ⟨hal-02541860⟩
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A. Blond,, Roba Moumné, G. Begis,, M. Pasco, Thomas Lecourt, et al.. Rhodium(II) carbene-mediated modification of 2-deoxystreptamine surrogates. Journal of Organic Chemistry, 2011, 52 (25), pp.3201-3203. ⟨hal-00649113⟩
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Benoit Colasson, Nicolas Le Poul, Yves Le Mest, Olivia Reinaud. Tris(triazolyl) Calix[6]arene-Based Zinc and Copper Funnel Complexes: Imidazole-like or Pyridine-like? A Comparative Study. Inorganic Chemistry, 2011, 50 (21), pp.10985--10993. ⟨10.1021/ic201540x⟩. ⟨hal-01175770⟩
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Benoît Gautier, Maria Miteva, Victor Goncalves, Florent Huguenot, Pascale Coric, et al.. Targeting the Proangiogenic VEGF-VEGFR Protein-Protein Interface with Drug-like Compounds by In Silico and In Vitro Screening. Chemistry and Biology, 2011, 18 (12), pp.1631-1639. ⟨10.1016/j.chembiol.2011.10.016⟩. ⟨hal-01061760⟩
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Olivier Jackowski, Thomas Lecourt, Laurent Micouin. Direct Synthesis of Polysubstituted Aluminoisoxazoles and Pyrazoles by a Metalative Cyclization. Organic Letters, 2011, 13 (20), pp.5664-5667. ⟨10.1021/ol202389u⟩. ⟨hal-02185376⟩
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Morgane Pasco, Roba Moumné, Thomas Lecourt, Laurent Micouin. Stereoselective synthesis of fluorinated 1,3-cis-diaminocyclopentanes.. Journal of Organic Chemistry, 2011, 76 (12), pp.5137-42. ⟨10.1021/jo2001512⟩. ⟨hal-00649119⟩
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Morgane Pasco, Roba Moumné, Thomas Lecourt, Laurent Micouin. Stereoselective Synthesis of Fluorinated 1,3- cis -Diaminocyclopentanes. Journal of Organic Chemistry, 2011, 76 (12), pp.5137-5142. ⟨10.1021/jo2001512⟩. ⟨hal-02186896⟩
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2010

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Xavier Bantreil, David Madec, Giovanni Poli, Guillaume Prestat, Guillaume Maitro, et al.. Palladium-catalyzed intramolecular allylic alkylation of -sulfinyl carbanions: a new asymmetric route to enantiopure -lactams. Tetrahedron Letters, 2010, 51, pp.1459-1461. ⟨hal-00458722⟩
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Elise Bernoud, Gaetan Le Duc, Xavier Bantreil, Guillaume Prestat, Giovanni Poli, et al.. Aryl sulfoxides from allyl sulfoxides via [2,3]-sigmatropic rearrangement and domino Pd-catalyzed generation / arylation of sulfenate anions. Organic Letters, 2010, 12, pp.320-323. ⟨10.1002/chin.201023082⟩. ⟨hal-00458700⟩
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Benoit Colasson, Nicolas Le Poul, Yves Le Mest, Olivia Reinaud. Electrochemically Triggered Double Translocation of Two Different Metal Ions with a Ditopic Calix[6]arene Ligand. Journal of the American Chemical Society, 2010, 132 (12), pp.4393--4398. ⟨10.1021/ja910676z⟩. ⟨hal-01175771⟩
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B. de Courcy, J. P. Piquemal, C. Garbay, N. Gresh. Polarizable water molecules in ligand-macromolecule recognition. Impact on the relative affinities of competing pyrrolopyrimidine inhibitors for FAK kinase.. Journal of the American Chemical Society, 2010, 132, pp.3312. ⟨hal-00494585⟩
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Réda Hadj-Slimane, Perayot Pamonsinlapatham, Jean-Philippe Herbeuval, Christiane Garbay, Yves Lepelletier, et al.. Rasv12 induces survivin/auroraB pathway conferring tumor cell apoptosis resistance. Cellular Signalling, 2010, 22 (8), pp.1214-1221. ⟨10.1016/j.cellsig.2010.03.013⟩. ⟨hal-00473108⟩
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Réda Hadj-Slimane, Perayot Pamonsinlapatham, Jean-Philippe Herbeuval, Christiane Garbay, Yves Lepelletier, et al.. RasV12 induces Survivin/AuroraB pathway conferring tumor cell apoptosis resistance. Cellular Signalling, 2010, 22 (8), pp.1214-1221. ⟨10.1016/j.cellsig.2010.03.013⟩. ⟨hal-04250005⟩
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Roba Moumné, Morgane Pasco, Elise Prost, Thomas Lecourt, Laurent Micouin, et al.. Fluorinated diaminocyclopentanes as chiral sensitive NMR probes of RNA structure.. Journal of the American Chemical Society, 2010, 132 (38), pp.13111-3. ⟨10.1021/ja1037885⟩. ⟨hal-00614591⟩
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Roba Moumné, Valéry Larue, Bili Seijo, Thomas Lecourt, Laurent Micouin, et al.. Tether influence on the binding properties of tRNALys3 ligands designed by a fragment-based approach.. Organic & Biomolecular Chemistry, 2010, 8 (5), pp.1154-9. ⟨10.1039/b921232a⟩. ⟨hal-00596199⟩
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Yuhan Zhou, Thomas Lecourt, Laurent Micouin. Direct Synthesis of 1,4-Disubstituted-5-alumino-1,2,3-triazoles: Copper-Catalyzed Cycloaddition of Organic Azides and Mixed Aluminum Acetylides. Angewandte Chemie International Edition, 2010, 49 (14), pp.2607-2610. ⟨10.1002/anie.200907016⟩. ⟨hal-02185392⟩
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2009

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Nicolas Auberger, Christine Gravier-Pelletier, Yves Le Merrer. Synthesis of a β-Ketophosphonate Bioisostere of UDP- N -acetylglucosamine. European Journal of Organic Chemistry, 2009, 2009 (20), pp.3323-3326. ⟨10.1002/ejoc.200900399⟩. ⟨hal-02188351⟩
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Christophe Decroos, Yun Li, Gildas Bertho, Yves Frapart, Daniel Mansuy, et al.. Synthetic studies towards diazepanone scaffolds. Tetrahedron: Asymmetry, 2009, 20 (20), pp.2320-2330. ⟨10.1016/j.tetasy.2009.09.022⟩. ⟨hal-03685013⟩
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Romain Duval, S. Kolb, E. Braud, D. Genest, C. Garbay. Rapid discovery of Triazolobenzylidene-Thiazolopyrimidines (TBTP) as CDC25 phosphatase inhibitors by parallel click chemistry and in situ screening. Journal of Combinatorial Chemistry, 2009, 11 (6), pp.947-950. ⟨10.1021/cc900140f⟩. ⟨hal-04504305⟩
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P. Pamonsinlapatham, R. Hadj-Slimane, F. Raynaud, M. Bickle, C. Corneloup, et al.. A RasGAP peptide aptamer inhibits RasGAP-Aurora interaction and induces caspase-independent tumor cell death.. PLoS ONE, 2009, 3, pp.e2902. ⟨hal-00422287⟩
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P. Pamonsinlapatham, R. Hadj-Slimane, Y. Lepelletier, B. Allain, M. Toccafondi, et al.. P120-Ras GTPase activating protein (RasGAP): a multi-interacting protein in downstream signaling.. Biochimie, 2009, 91, pp.320-328. ⟨hal-00397954⟩
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G. Thiabaud, G. Guillemot, Isabelle Schmitz-Afonso, B. Colasson, O. Reinaud. Solid-state chemistry at an isolated copper(I) center with O2. Angewandte Chemie International Edition, 2009, 48 (40), pp.7383-7386. ⟨10.1002/anie.200902691⟩. ⟨hal-00469664⟩
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2008

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Michaël Bosco, Sophie Le Gall, Christophe Rihouey, Samuel Couve-Bonnaire, Muriel Bardor, et al.. 6-Azido d-galactose transfer to N-acetyl-d-glucosamine derivative using commercially available β-1,4-galactosyltransferase. Tetrahedron Letters, 2008, 49 (14), pp.2294-2297. ⟨10.1016/j.tetlet.2008.02.018⟩. ⟨hal-02384444⟩
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Chloée Bournaud, Thomas Lecourt, Laurent Micouin, Catherine Méliet, Francine Agbossou-Niedercorn. Desymmetrization of meso-Bicyclic Hydrazines by Rhodium-Catalyzed Enantioselective Hydroformylation. European Journal of Organic Chemistry, 2008, 2008 (13), pp.2298-2302. ⟨10.1002/ejoc.200800116⟩. ⟨hal-02185573⟩
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C. Courme, S. Gillon, N. Gresh, M. Vidal, C. Garbay, et al.. Terminal alkyne-functionalized triazine by Sonogashira coupling : synthesis of a potential cell signalling inhibitor via click chemistry. Tetrahedron Letters, 2008, 49, pp.4542-4545. ⟨hal-00323801⟩
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Thomas Lombès, Guillaume Bégis, Frédérique Maurice, Serge Turcaud, Thomas Lecourt, et al.. NMR-Guided Fragment-Based Approach for the Design of AAC(6′)-Ib Ligands. ChemBioChem, 2008, 9 (9), pp.1368-1371. ⟨10.1002/cbic.200700677⟩. ⟨hal-02185444⟩
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Perayot Pamonsinlapatham, Réda Hadj-Slimane, Françoise Raynaud, Marc Bickle, Claudine Corneloup, et al.. A RasGAP SH3 peptide aptamer inhibits RasGAP-Aurora interaction and induces caspase-independent tumor cell death. PLoS ONE, 2008, 3 (8), pp.e2902. ⟨10.1371/journal.pone.0002902⟩. ⟨hal-00416049⟩
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P. Pamonsinlapatham, R. Hadj-Slimane, Y. Lepelletier, B. Allain, M. Toccafondi, et al.. P120-Ras GTPase activating protein (RasGAO): A multi-interacting protein in downstream signaling.. Biochimie, 2008, ?, pp.?-?. ⟨hal-00356306⟩
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P. Pamonsinlapatham, R. Hadj-Slimane, F. Raynaud, M. Bickle, C. Corneloup, et al.. A RasGAP SH3 peptide aptamer inhibits RASGAP-Aurora interaction and induces caspase-independent tumor cell death.. PLoS ONE, 2008, 3, pp.2902-2914. ⟨hal-00356308⟩
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2007

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Florence Chung, Carine Tisné, Thomas Lecourt, Frédéric Dardel, Laurent Micouin. NMR-guided fragment-based approach for the design of tRNA(Lys3) ligands.. Angewandte Chemie International Edition, 2007, 46 (24), pp.4489-91. ⟨10.1002/anie.200605201⟩. ⟨hal-00218344⟩
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Jennifer Dourlat, Wang-Qing Liu, Nohad Gresh, Christiane Garbay. Novel 1,4-benzodiazepine derivatives with antiproliferative properties on tumor cell lines.. Bioorganic and Medicinal Chemistry Letters, 2007, 17 (9), pp.2527-30. ⟨10.1016/j.bmcl.2007.02.016⟩. ⟨inserm-00168656⟩
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Jennifer Dourlat, Bruno Valentin, Wang-Qing Liu, Christiane Garbay. New syntheses of tetrazolylmethylphenylalanine and O-malonyltyrosine as pTyr mimetics for the design of STAT3 dimerization inhibitors.. Bioorganic and Medicinal Chemistry Letters, 2007, 17 (14), pp.3943-6. ⟨10.1016/j.bmcl.2007.04.107⟩. ⟨inserm-00168682⟩
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Victor Goncalves, Benoît Gautier, Anne Regazzetti, Pascale Coric, Serge Bouaziz, et al.. On-resin cyclization of peptide ligands of the Vascular Endothelial Growth Factor Receptor 1 by copper(I)-catalyzed 1,3-dipolar azide–alkyne cycloaddition. Bioorganic and Medicinal Chemistry Letters, 2007, 17 (20), pp.5590-5594. ⟨10.1016/j.bmcl.2007.07.087⟩. ⟨hal-02122521⟩
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Victor Goncalves, Benoît Gautier, Pascale Coric, Serge Bouaziz, Christine Lenoir, et al.. Rational Design, Structure, and Biological Evaluation of Cyclic Peptides Mimicking the Vascular Endothelial Growth Factor. Journal of Medicinal Chemistry, 2007, 50 (21), pp.5135-5146. ⟨10.1021/jm0706970⟩. ⟨hal-02122518⟩
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Victor Goncalves, Benoit Gautier, Christiane Garbay, Michel Vidal, Nicolas Inguimbert. Development of a chemiluminescent screening assay for detection of vascular endothelial growth factor receptor 1 ligands.. Analytical Biochemistry, 2007, 366 (1), pp.108-10. ⟨10.1016/j.ab.2007.03.027⟩. ⟨inserm-00168674⟩
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Brunilde Gril, Michel Vidal, Franck Assayag, Marie-France Poupon, Wang-Qing Liu, et al.. Grb2-SH3 ligand inhibits the growth of HER2+ cancer cells and has antitumor effects in human cancer xenografts alone and in combination with docetaxel.. International Journal of Cancer, 2007, 121 (2), pp.407-15. ⟨10.1002/ijc.22674⟩. ⟨inserm-00168667⟩
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R. Hadj-Slimane, Y. Lepelletier, N. Lopez, C. Garbay, F. Raynaud. Short interfering RNA (siRNA), a novel therapeutic tool acting on angiogenesis.. Biochimie, 2007, 89, pp.1234-1244. ⟨hal-00172570⟩
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Vincent Leroux, Nohad Gresh, Wang-Qing Liu, Christiane Garbay, Bernard Maigret. Role of water molecules for binding inhibitors in the SH2 domain of Grb2: a molecular dynamics study. Journal of Molecular Structure: THEOCHEM, 2007, 806 (1-3), pp.51-66. ⟨inria-00188596⟩
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Olivier Monasson, Maryon Ginisty, Gildas Bertho, Christine Gravier-Pelletier, Yves Le Merrer. Efficient synthesis of polyfunctionalised enantiopure diazepanone scaffolds. Tetrahedron Letters, 2007, 48 (46), pp.8149-8152. ⟨10.1016/j.tetlet.2007.09.098⟩. ⟨hal-03685046⟩
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Hiba Noureddine, Claudine Schmitt, Wangqing Liu, Christiane Garbay, Jean Massoulié, et al.. Assembly of acetylcholinesterase tetramers by peptidic motifs from the proline-rich membrane anchor, PRiMA: competition between degradation and secretion pathways of heteromeric complexes.. Journal of Biological Chemistry, 2007, 282 (6), pp.3487-97. ⟨10.1074/jbc.M607221200⟩. ⟨hal-00140001⟩
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Giuseppe Paladino, David Madec, Guillaume Prestat, Guillaume Maitro, Giovanni Poli, et al.. Oxidative Addition of Ligand-Chelated Palladium(0) to Aryl Halides: Comparison between 1,2-Bisthioethers and 1,2-Bisphosphines. Organometallics, 2007, 26 (2), pp.455. ⟨10.1021/om060846x⟩. ⟨hal-00158052⟩
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Régis Villet, Matthieu Fonvielle, Patricia Busca, Maryline Chemama, Antoine P. Maillard, et al.. Idiosyncratic features in tRNAs participating in bacterial cell wall synthesis. Nucleic Acids Research, 2007, 35 (20), pp.6870-6883. ⟨10.1093/nar/gkm778⟩. ⟨hal-02331010⟩
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2006

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Martine Bonin, Laurent Micouin, Ariane Chauveau. Asymmetric 1,3-Dipolar Cycloadditions of Cyclic Stabilized Ylides Derived from Chiral 1,2-Amino Alcohols. SYNLETT, 2006, 2006 (15), pp.2349-2363. ⟨10.1055/s-2006-949626⟩. ⟨hal-02185347⟩
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Frédérique Maurice, Guillaume Bégis, Laurent Micouin, Frédéric Dardel. NMR identification of ligands of aminoglycoside resistance enzymes. Comptes Rendus. Chimie, 2006, 9, pp.413-419. ⟨hal-00021873⟩
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2005

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Marie-Priscille Brun, Emmanuelle Braud, Delphine Angotti, Odile Mondésert, Muriel Quaranta, et al.. Design, synthesis, and biological evaluation of novel naphthoquinone derivatives with CDC25 phosphatase inhibitory activity.. Bioorganic and Medicinal Chemistry, 2005, 13 (16), pp.4871-9. ⟨10.1016/j.bmc.2005.05.005⟩. ⟨hal-00317419⟩
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Christiane Dietrich-Buchecker, Benoit Colasson, Damien Jouvenot, Jean-Pierre Sauvage. Synthesis of Multi-1,10-phenanthroline Ligands with 1,3-Phenylene Linkers and Their Lithium Complexes. Chemistry - A European Journal, 2005, 11 (15), pp.4374 - 4386. ⟨10.1002/chem.200401264⟩. ⟨hal-01689666⟩
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Stéphanie Gobert Gosse, Caroline Bourgin, Wang Qing Liu, Christiane Garbay, Guy Mouchiroud. M-CSF stimulated differentiation requires persistent MEK activity and MAPK phosphorylation independent of Grb2-Sos association and phosphatidylinositol 3-kinase activity.. Cellular Signalling, 2005, 17 (11), pp.1352-62. ⟨10.1016/j.cellsig.2005.02.002⟩. ⟨hal-00192857⟩
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S. Gobert-Gosse, C. Bourgin, Liu W. Q., C. Garbay, G. Mouchiroud. GM-CSF stimulated differentiation requires persistent MEK activity and MAPK phosphorylation independant of Grb2-Sos association and phosphatidylinositol 3-kinase activity.. Cellular Signalling, 2005, 17, pp.1352-1632. ⟨hal-00150766⟩
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2004

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Virginie Binet, Carole Brajon, Laurent Le Corre, Francine Acher, Jean-Philippe Pin, et al.. The heptahelical domain of GABA(B2) is activated directly by CGP7930, a positive allosteric modulator of the GABA(B) receptor.. Journal of Biological Chemistry, 2004, 279 (28), pp.29085-91. ⟨10.1074/jbc.M400930200⟩. ⟨inserm-00318926⟩
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Marie-Priscille Brun, Laurent Bischoff, Christiane Garbay. A Very Short Route to Enantiomerically Pure Coumarin-Bearing Fluorescent Amino Acids. Angewandte Chemie International Edition, 2004, 43 (26), pp.3432-3436. ⟨10.1002/anie.200454116⟩. ⟨hal-02385514⟩
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Christophe Feuvrie, Jérôme Blanchet, Martine Bonin, Laurent Micouin. Synthesis and reactivity of mixed alkynylalanes by direct triethylamine-catalyzed alumination of terminal alkynes.. Organic Letters, 2004, 6 (14), pp.2333-6. ⟨10.1021/ol049346v⟩. ⟨hal-00909871⟩
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Yen Vo-Hoang, Cécile Gasse, Michel Vidal, Christiane Garbay, Hervé Galons. Efficient synthesis of N-benzyl-3-aminopyrrolidine-2,5-dione and N-benzyl-3-aminopyrrolidin-2-one. Tetrahedron Letters, 2004, 45 (18), pp.3603-3605. ⟨10.1016/j.tetlet.2004.03.052⟩. ⟨hal-03531874⟩
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2003

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Marie-Priscille Brun, Anne-Sophie Martin, Christiane Garbay, Laurent Bischoff. An alternative route to the proline derivative (2S,5R)-5-ethoxycarbonylmethyl-pyrrolidine-2-carboxylic acid from protected glutamic acid. Tetrahedron Letters, 2003, 44 (37), pp.7011-7013. ⟨10.1016/S0040-4039(03)01792-1⟩. ⟨hal-02385515⟩
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S. Cutri, A. Chiaroni, M. Bonin, L. Micouin, H.-P. Husson. Practical Asymmetric Synthesis of 1,2-Diamines in the 3-Aminoazepane Series. Journal of Organic Chemistry, 2003, 68 (7), pp.2645-2651. ⟨10.1021/jo026711s⟩. ⟨hal-02186903⟩
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Yen Vo-Hoang, Laurent Micouin, Catherine Ronet, Gabriel Gachelin, Martine Bonin. Total Enantioselective Synthesis and In Vivo Biological Evaluation of a Novel Fluorescent BODIPY α-Galactosylceramide. ChemBioChem, 2003, 4 (1), pp.27-33. ⟨10.1002/cbic.200390009⟩. ⟨hal-03531886⟩
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2002

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Jerome Blanchet, M. Bonin, L. Micouin. Recent progress in the asymmetric synthesis of α-substituted propargylamines. Organic Preparations and Procedures International : The New Journal for Organic Synthesis, 2002, 34 (5), pp.467-492. ⟨10.1080/00304940209355765⟩. ⟨hal-02328004⟩
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Jérôme Blanchet, Martine Bonin, Laurent Micouin, Henri-Philippe Husson. Isomerization of Chiral Non-Racemic α-Substituted Propargylic Amines to Terminal Acetylenes. European Journal of Organic Chemistry, 2002, 2002 (15), pp.2598-2602. ⟨10.1002/1099-0690(200208)2002:15<2598::AID-EJOC2598>3.0.CO;2-V⟩. ⟨hal-02185592⟩
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Wang-Qing Liu, Catherine Olszowy, Laurent Bischoff, Christiane Garbay. Enantioselective synthesis of (2S)-2-(4-phosphonophenylmethyl)-3-aminopropanoic acid suitably protected for peptide synthesis. Tetrahedron Letters, 2002, 43 (8), pp.1417-1419. ⟨10.1016/S0040-4039(02)00004-7⟩. ⟨hal-02385516⟩
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Pierre Nioche, Wang-Qing Liu, Isabelle Broutin, Franck Charbonnier, Marie-Thérèse Latreille, et al.. Crystal structures of the SH2 domain of grb2: highlight on the binding of a new high-affinity inhibitor. Journal of Molecular Biology, 2002, 315 (5), pp.1167-1177. ⟨10.1006/jmbi.2001.5299⟩. ⟨hal-02520104⟩
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A. Pérez Luna, M.-A Ceschi, M. Bonin, L. Micouin, H.-P. Husson, et al.. Enantioselective Desymmetrization of Meso Bicyclic Hydrazines: A Novel Approach to the Asymmetric Synthesis of Polysubstituted Amino Cyclopentanic Cores. Journal of Organic Chemistry, 2002, 67 (10), ⟨10.1021/jo011190e⟩. ⟨hal-02186763⟩
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Alejandro Pérez Luna, Martine Bonin, Laurent Micouin, Henri-Philippe Husson. Reversal of Enantioselectivity in the Asymmetric Rhodium- versus Iridium-Catalyzed Hydroboration of Meso Substrates. Journal of the American Chemical Society, 2002, 124 (41), pp.12098-12099. ⟨10.1021/ja026714m⟩. ⟨hal-02185596⟩
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Jordi Piró, Pilar Forns, Jérôme Blanchet, Martine Bonin, Laurent Micouin, et al.. Asymmetric synthesis of β-pseudopeptides from chiral 3,4-aziridinolactams. Tetrahedron: Asymmetry, 2002, 13 (9), pp.995-1004. ⟨10.1016/S0957-4166(02)00221-5⟩. ⟨hal-02328007⟩
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2001

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Valérie Alezra, Martine Bonin, Laurent Micouin, Clotilde Policar, Henri-Philippe Husson. The Origin of Chemical and Configurational Stability of Chiral Nonracemic Tert-Butyl Aziridinecarboxylate Anions. European Journal of Organic Chemistry, 2001, 2001 (13), pp.2589-2594. ⟨10.1002/1099-0690(200107)2001:13<2589::AID-EJOC2589>3.0.CO;2-Y⟩. ⟨hal-02011971⟩
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Jérôme Blanchet, Martine Bonin, Laurent Micouin, Henri-Philippe Husson. Asymmetric synthesis of α-substituted propynyl amines. Application to the preparation of a polysubstituted dihydroisoindoline framework. Tetrahedron Letters, 2001, 42 (18), pp.3171-3173. ⟨10.1016/S0040-4039(01)00356-2⟩. ⟨hal-02328009⟩
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Katia Cailliau, Edith Browaeys-Poly, Isabelle Broutin-L'Hermite, Pierre Nioche, Christiane Garbay, et al.. Grb2 promotes reinitiation of meiosis in Xenopus oocytes. Cellular Signalling, 2001, 13 (1), pp.51-55. ⟨10.1016/s0898-6568(00)00138-8⟩. ⟨hal-02520116⟩
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2000

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B Bellier, M. Million, S Danascimento, H. Meudal, S Kellou, et al.. Replacement of glycine with dicarbonyl and related moieties in analogues of the C-terminal pentapeptide of cholecystokinin: CCK(2) agonists displaying a novel binding mode.. Journal of Medicinal Chemistry, 2000, 43 (20), pp.3614-23. ⟨hal-02122170⟩
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Jérôme Blanchet, Martine Bonin, Laurent Micouin, Henri-Philippe Husson. [2,3]-Meisenheimer rearrangement of N-allyl phenylglycinol derivatives. NC versus CC chirality transfer. Tetrahedron Letters, 2000, 41 (43), pp.8279-8283. ⟨10.1016/S0040-4039(00)01460-X⟩. ⟨hal-02328033⟩
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J. Blanchet, M. Bonin, L. Micouin, H. P. Husson. Synthesis of enantiomerically pure alpha-substituted propargylic amines by reaction of organoaluminum reagents with oxazolidines.. Journal of Organic Chemistry, 2000, 65 (20), pp.6423-6. ⟨hal-00909874⟩
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Jerome Blanchet, M. Bonin, L. Micouin, H.-P. Husson. Synthesis of Enantiomerically Pure α-Substituted Propargylic Amines by Reaction of Organoaluminum Reagents with Oxazolidines. Journal of Organic Chemistry, 2000, 65 (20), pp.6423-6426. ⟨10.1021/jo0003706⟩. ⟨hal-02328014⟩
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Marie-France Carlier, Pierre Nioche, Isabelle Broutin-L'Hermite, Rajaa Boujemaa, Christophe Le Clainche, et al.. GRB2 Links Signaling to Actin Assembly by Enhancing Interaction of Neural Wiskott-Aldrich Syndrome Protein (N-WASp) with Actin-related Protein (ARP2/3) Complex. Journal of Biological Chemistry, 2000, 275 (29), pp.21946-21952. ⟨10.1074/jbc.M000687200⟩. ⟨hal-02520338⟩
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1999

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Jérôme Blanchet, Martine Bonin, Angèle Chiaroni, Laurent Micouin, Claude Riche, et al.. Diastereoselective alkynylation of chiral non-racemic oxazolidines with mixed organoaluminum compounds. Tetrahedron Letters, 1999, 40 (15), pp.2935-2938. ⟨10.1016/S0040-4039(99)00328-7⟩. ⟨hal-02328037⟩
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1998

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B Bellier, S da Nascimento, H. Meudal, E. Gincel, B.P Roques, et al.. Novel constrained CCK-B dipeptoid antagonists derived from pipecolic acid.. Bioorganic and Medicinal Chemistry Letters, 1998, 8 (11), pp.1419-24. ⟨hal-02122133⟩
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1997

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Bruno Bellier, Isabelle Mccort, Bertrand Ducos, Sophie Danascimento, Hervé Meudal, et al.. Synthesis and Biological Properties of New Constrained CCK-B Antagonists: Discrimination of Two Affinity States of the CCK-B Receptor on Transfected CHO Cells. Journal of Medicinal Chemistry, 1997, 40 (24), pp.3947-3956. ⟨10.1021/jm970439a⟩. ⟨hal-02122116⟩
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Conference papers

2023

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Miryana Hemadi, Romain Briandet, Christine Gravier-Pelletier, John Lomas, Laurent Royon. Nanoparticules métalliques fonctionnalisées pour l'éradication de biofilm à la surface de condenseurs d'eau de rosée. CNRIUT 2023 Saint Pierre - La Réunion, IUT de Saint Pierre, Jun 2023, Saint Pierre (La Réunion), La Réunion. ⟨hal-04326928⟩
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Book sections

2025

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L. Micouin, R. Piccardi. Organoaluminum Reagents. Comprehensive Organic Synthesis, Elsevier; Elsevier, pp.45-69, 2025, ⟨10.1016/B978-0-323-96025-0.00041-7⟩. ⟨hal-05304382⟩
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2016

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Riccardo Piccardi, Laurent Micouin, Olivier Jackowski. The Chemistry of Alkynylaluminum Species. Marek, Ilan. PATAI'S Chemistry of Functional Groups, John Wiley & Sons, Ltd, pp.1--47, 2016, 978-0-470-68253-1. ⟨10.1002/9780470682531.pat0832⟩. ⟨hal-02891076⟩
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Françoise Schaefers, Tobias A. M. Gulder, Cyril Bressy, Michaël Smietana, Erica Benedetti, et al.. Polyketides. Zografos A. From Biosynthesis to Total Synthesis: Strategies and Tactics for Natural Products, Wiley, pp.21-129, 2016, ⟨10.1002/9781118754085.ch2⟩. ⟨hal-01415109⟩
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2014

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Fabrice Chemla, Franck Ferreira, Olivier Jackowski, Laurent Micouin, Alejandro Perez-Luna. Carbon\textendashCarbon Bond Forming Reactions Mediated by Organozinc Reagents. de Meijere, Armin and Bräse, Stefan and Oestreich, Martin. Metal-Catalyzed Cross-Coupling Reactions and More, Wiley-VCH Verlag GmbH & Co. KGaA, pp.279--364, 2014, 978-3-527-65558-8. ⟨10.1002/9783527655588.ch4⟩. ⟨hal-02891142⟩
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Fabrice Chemla, Franck Ferreira, Alejandro Perez-Luna, Laurent Micouin, Olivier Jackowski. Carbon\textendashCarbon Bond-Forming Reactions Mediated by Organomagnesium Reagents. de Meijere, Armin and Bräse, Stefan and Oestreich, Martin. Metal-Catalyzed Cross-Coupling Reactions and More, Wiley-VCH Verlag GmbH & Co. KGaA, pp.365--422, 2014, 978-3-527-65558-8. ⟨10.1002/9783527655588.ch5⟩. ⟨hal-02891143⟩
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Patents

2019

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François Estour, Michaël Bosco. Nouveaux dimères de cyclodextrines et leurs utilisations comme épurateurs chimiques. France, N° de brevet: FR1910022. 2019. ⟨hal-02376085⟩
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Poster communications

2024

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Michaël Bosco, Nolwenn Periaux-Becquey, Finn Tlatlik, Stéphanie Pradeau, Isabelle Chantret, et al.. Synthesis Of Fluorescent And Fluorogenic Probes To Characterize Lost, The Lysosomal Oligosaccharide Transporter. XXVIII EFMC International Symposium on Medicinal Chemistry, Sep 2024, Rome, Italy. ⟨hal-04773375⟩
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2023

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Michaël Bosco, Younès Bouzidi, Haifei Gao, Stéphanie Pradeau, Isabelle Chantret, et al.. Synthèse de N-acétylchitooligosaccharides fluorescents : Applications à la caractérisation du transport lysosomal d’oligosaccharides (LOST). 3èmes Journées du GDR ChemBio, Jun 2023, Strasbourg, France. ⟨hal-04784597⟩
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2022

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Michaël Bosco, Younès Bouzidi, Haifei Gao, Isabelle Chantret, Sébastien Fort, et al.. Chemical tools for the identification of Lysosomal OligoSaccharide Transporter (LOST). Journées de Chimie Organique de la SFC 2022, Nov 2022, Palaiseau, France. ⟨hal-04784650⟩
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2018

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Céline Aubry, Paolo Clerici, Laurent Micouin, Jean-Luc Pernodet, Sylvie Lautru. COMBINATORIAL BIOSYNTHESIS OF NON-RIBOSOMAL PEPTIDES, THE EXAMPLE OF PYRROLAMIDES. 5èmes journées du GDR MufoPAM, Oct 2018, Paris, France. ⟨hal-02367767⟩
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Journal articles

2024

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Hugo Esteves, Tania Xavier, Sonia Lajnef, Fabienne Peyrot, Guillaume Lefèvre, et al.. Iron-Catalyzed Intramolecular C(sp 3 )-H Lactonization of Hydroxamate Derivatives Promoted by a 1,5-HAT. ACS Catalysis, 2024, 14 (6), pp.4329-4339. ⟨10.1021/acscatal.3c04900⟩. ⟨hal-04778122⟩
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Zhendong Peng, Laurent Royon, Yun Luo, Philippe Decorse, Sarra Gam Derouich, et al.. Eradication of planktonic bacteria by shape-tailored gold nanoparticle photothermia. Materials Advances, 2024, 21, ⟨10.1039/d4ma00821a⟩. ⟨hal-04724709⟩
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2023

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Georgina Kirby, Guillaume Prestat, Farouk Berhal. Iron-catalyzed intermolecular oxyamination of terminal alkenes promoted by HFIP using hydroxylamine derivatives. Journal of Organic Chemistry, 2023, 88 (7), pp.4720-4729. ⟨10.1021/acs.joc.3c00198⟩. ⟨hal-04266179⟩
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2022

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Mélanie Faria da Cunha, Iwona Pranke, Ali Sassi, Christiane Schreiweis, Stéphanie Moriceau, et al.. Systemic bis-phosphinic acid derivative restores chloride transport in Cystic Fibrosis mice. Scientific Reports, 2022, 12 (1), pp.6132. ⟨10.1038/s41598-022-09678-9⟩. ⟨hal-03662932⟩
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Martin Oliver, Laurent Le Corre, Mélanie Poinsot, Michaël Bosco, Hongwei Wan, et al.. A Sub-Micromolar MraYAA Inhibitor with an Aminoribosyl Uridine Structure and a (S,S)-Tartaric Diamide: Synthesis, Biological Evaluation and Molecular Modeling. Molecules, 2022, 27 (6), pp.1769. ⟨10.3390/molecules27061769⟩. ⟨hal-03632451⟩
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Célia Sahli, Sergio Moya, John Lomas, Christine Gravier-Pelletier, Romain Briandet, et al.. Recent advances in nanotechnology for eradicating bacterial biofilm. Theranostics, 2022, 12 (5), pp.2383-2405. ⟨10.7150/thno.67296⟩. ⟨hal-03607522⟩
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Hongwei Wan, Raja Ben Othman, Laurent Le Corre, Mélanie Poinsot, Martin Oliver, et al.. New MraYAA Inhibitors with an Aminoribosyl Uridine Structure and an Oxadiazole. Antibiotics, 2022, 11 (9), pp.1189. ⟨10.3390/antibiotics11091189⟩. ⟨hal-03805942⟩
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2021

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Emmanuelle Bardin, Alexandra Pastor, Michaela Semeraro, Anita Golec, Kate Hayes, et al.. Modulators of CFTR. Updates on clinical development and future directions. European Journal of Medicinal Chemistry, 2021, 213, pp.113195. ⟨10.1016/j.ejmech.2021.113195⟩. ⟨hal-03445073⟩
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Anais Biscotti, François Estour, Berthe-Sandra Sembo-Backonly, Sebastien Balieu, Michaël Bosco, et al.. Gd3+ Complexes Conjugated to Cyclodextrins: Hydroxyl Functions Influence the Relaxation Properties. Processes, 2021, 9 (2), pp.269. ⟨10.3390/pr9020269⟩. ⟨hal-03127005⟩
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Sara Bitam, Ahmad Elbahnsi, Geordie Creste, Iwona Pranke, Benoit Chevalier, et al.. New insights into structure and function of bis-phosphinic acid derivatives and implications for CFTR modulation. Scientific Reports, 2021, 11 (1), ⟨10.1038/s41598-021-83240-x⟩. ⟨hal-03184333⟩
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Alessandra Corio, Christine Gravier-Pelletier, Patricia Busca. Regioselective Functionalization of Quinolines through C-H Activation: A Comprehensive Review. Molecules, 2021, 26 (18), pp.5467. ⟨10.3390/molecules26185467⟩. ⟨hal-03445072⟩
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Georgina Kirby, Laurence Grimaud, Maxime Vitale, Guillaume Prestat, Farouk Berhal. Iron(II)-catalyzed intermolecular aziridination of alkenes employing hydroxylamine derivatives as clean nitrene sources. Green Chemistry, 2021, 23 (23), pp.9428-9432. ⟨10.1039/d1gc03495b⟩. ⟨hal-03588341⟩
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Martin Oliver, Laurent Le Corre, Mélanie Poinsot, Alessandra Corio, Léa Madegard, et al.. Synthesis, biological evaluation and molecular modeling of urea-containing MraY inhibitors. Organic & Biomolecular Chemistry, 2021, 19 (26), pp.5844-5866. ⟨10.1039/D1OB00710F⟩. ⟨hal-03432617⟩
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2020

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Michaël Bosco, Su-Jin Paik, Patricia Busca, Stuart E H Moore, Christine Gravier-Pelletier. Synthetic Route to Glycosyl β-1C-(phosphino)-phosphonates as Unprecedented Stable Glycosyl Diphosphate Analogs and Their Preliminary Biological Evaluation. Molecules, 2020, 25 (21), pp.4969. ⟨10.3390/molecules25214969⟩. ⟨hal-03030819⟩
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Michaël Bosco, Marjorie Damian, Vinay Chauhan, Mélanie Roche, Pierre Guillet, et al.. Biotinylated non-ionic amphipols for GPCR ligands screening. Methods, 2020, 180, pp.69 - 78. ⟨10.1016/j.ymeth.2020.06.001⟩. ⟨hal-03009212v2⟩
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Sandra Abi Fayssal, Alessandro Giungi, Farouk Berhal, Guillaume Prestat. Iron-Catalyzed Intra-intermolecular Aminoazidation of Alkenes. Organic Process Research and Development, 2020, 24 (5), pp.695-703. ⟨10.1021/acs.oprd.9b00400⟩. ⟨hal-03667879⟩
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https://hal.science/hal-03667879/file/Manuscript_GPFB_Iron.pdf BibTex
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Jeanne Fichez, Cathia Soulié, Laurent Le Corre, Sophie Sayon, Stéphane Priet, et al.. Discovery, SAR study and ADME properties of methyl 4-amino-3-cyano-1-(2-benzyloxyphenyl)-1 H -pyrazole-5-carboxylate as an HIV-1 replication inhibitor. RSC Medicinal Chemistry, 2020, 11 (5), pp.577-582. ⟨10.1039/D0MD00025F⟩. ⟨hal-03030936⟩
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2019

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Usama Ashraf, Laura Tengo, Laurent Le Corre, Guillaume Fournier, Patricia Busca, et al.. Destabilization of the human RED–SMU1 splicing complex as a basis for host-directed antiinfluenza strategy. Proceedings of the National Academy of Sciences of the United States of America, 2019, 116 (22), pp.10968-10977. ⟨10.1073/pnas.1901214116⟩. ⟨hal-02160991⟩
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Ahmad Massarweh, Michael Bosco, Isabelle Chantret, Thibaut Léger, Layla Jamal, et al.. Bacterial Lipid II Analogs: Novel In Vitro Substrates for Mammalian Oligosaccharyl Diphosphodolichol Diphosphatase (DLODP) Activities. Molecules, 2019, 24 (11), pp.2135. ⟨10.3390/molecules24112135⟩. ⟨hal-02172947⟩
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2018

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Mickaël Fer, Laurent Le Corre, Nicolas Pietrancosta, Nathalie Evrard-Todeschi, Samir Olatunji, et al.. Bacterial Transferase MraY, a Source of Inspiration towards New Antibiotics. Current Medicinal Chemistry, 2018, 25 (42), pp.6013-6029. ⟨10.2174/0929867325666180330095154⟩. ⟨hal-02364241⟩
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Anne-Doriane Manick, Farouk Berhal, Guillaume Prestat. Development of a One-Pot Four C–C Bond-Forming Sequence Based on Palladium/Ruthenium Tandem Catalysis. Organic Letters, 2018, 20 (1), pp.194-197. ⟨10.1021/acs.orglett.7b03556⟩. ⟨hal-03710509⟩
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Anne-Doriane Manick, Sidonie Aubert, Boubacar Yalcouye, Thierry Prangé, Farouk Berhal, et al.. Access to Functionalized Imidazolidin-2-one Derivatives by Iron-Catalyzed Oxyamination of Alkenes. Chemistry - A European Journal, 2018, 24 (44), pp.11485-11492. ⟨10.1002/chem.201802190⟩. ⟨hal-03710267⟩
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Cécile Morlot, Daniel Straume, Katharina Peters, Olav A Hegnar, Nolwenn Simon, et al.. Structure of the essential peptidoglycan amidotransferase MurT/GatD complex from Streptococcus pneumoniae. Nature Communications, 2018, 9, pp.3180. ⟨10.1038/s41467-018-05602-w⟩. ⟨hal-01861372⟩
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2017

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Michaël Bosco, Ahmad Massarweh, Soria Iatmanen-Harbi, Ahmed Bouhss, Isabelle Chantret, et al.. Synthesis and biological evaluation of chemical tools for the study of Dolichol Linked Oligosaccharide Diphosphatase (DLODP).. European Journal of Medicinal Chemistry, 2017, 125, pp.952-964. ⟨10.1016/j.ejmech.2016.10.013⟩. ⟨hal-01440749⟩
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Sophie Letort, Michaël Bosco, Benedetta Cornelio, Frédérique Brégier, Sébastien Daulon, et al.. Structure-efficiency relationships of cyclodextrin scavengers in the hydrolytic degradation of organophosphorus compounds. Beilstein Journal of Organic Chemistry, 2017, 13, pp.417-427. ⟨10.3762/bjoc.13.45⟩. ⟨hal-02046294⟩
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Zhongyi Mao, Elisabetta Martini, Guillaume Prestat, Julie Oble, Pei-Qiang Huang, et al.. Analogues of the 2-carboxyl-6-hydroxyoctahydroindole (CHOI) unit from diverging Pd-catalyzed allylations: Selectivity as a function of the double bond position. Tetrahedron Letters, 2017, 58 (44), pp.4174-4178. ⟨10.1016/j.tetlet.2017.09.046⟩. ⟨hal-01675514⟩
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2016

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Ahmad Massarweh, Michaël Bosco, Soria Iatmanen-Harbi, Clarice Tessier, Nicolas Auberger, et al.. Demonstration of an oligosaccharide-diphosphodolichol diphosphatase activity whose subcellular localization is different than those of dolichyl-phosphate-dependent enzymes of the dolichol cycle. Journal of Lipid Research, 2016, 57 (6), pp.1029-1042. ⟨10.1194/jlr.M067330⟩. ⟨hal-02997964⟩
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2015

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Mickaël J Fer, Ahmed Bouhss, Mariana Patrão, Laurent Le Corre, Nicolas Pietrancosta, et al.. 5'-Methylene-triazole-substituted-aminoribosyl uridines as MraY inhibitors: synthesis, biological evaluation and molecular modeling.. Organic & Biomolecular Chemistry, 2015, 13 (26), pp.7193-222. ⟨10.1039/c5ob00707k⟩. ⟨hal-01433063⟩
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Zsófia Sólyom, Peixiang Ma, Melanie Schwarten, Michaël Bosco, Ange Polidori, et al.. The Disordered Region of the HCV Protein NS5A: Conformational Dynamics, SH3 Binding, and Phosphorylation.. Biophysical Journal, 2015, 109 (7), pp.1483-96. ⟨10.1016/j.bpj.2015.06.040⟩. ⟨hal-01229755⟩
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2014

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Claire Kammerer, Guillaume Prestat, David Madec, Giovanni Poli. Synthesis of γ-Lactams and γ-Lactones via Intramolecular Pd-Catalyzed Allylic Alkylations. Accounts of Chemical Research, 2014, 47 (12), pp.3439--3447. ⟨10.1021/ar500178n⟩. ⟨hal-01712373⟩
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Laetitia Mistico, Emel Ay, Vaizanne Huynh, Aurelie Bourderioux, Fabrice Chemla, et al.. Reactivity of tert-butanesulfinamides in palladium-catalyzed allylic substitutions. Journal of Organometallic Chemistry, 2014, 760, pp.124--129. ⟨10.1016/j.jorganchem.2013.11.026⟩. ⟨hal-01712367⟩
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Milena Opacié, Gregory Durand, Michaël Bosco, Ange Polidori, Jean-Luc Popot. Amphipols and photosynthetic light-harvesting pigment-protein complexes.. Journal of Membrane Biology, 2014, ⟨10.1007/s00232-014-9712-6⟩. ⟨hal-01332956⟩
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Jamshid Rajabi, Mélanie M. Lorion, Vu Linh Ly, Frédéric Liron, Julie Oble, et al.. Dormant versus Evolving Aminopalladated Intermediates: Toward a Unified Mechanistic Scenario in Pd ^\textrmII -Catalyzed Aminations. Chemistry - A European Journal, 2014, 20 (6), pp.1539--1546. ⟨10.1002/chem.201302744⟩. ⟨hal-01712369⟩
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Micol Rigamonti, Guillaume Prestat, Gianluigi Broggini, Giovanni Poli. Synthesis of 1,4-benzodiazepinones via palladium-catalysed allene carbopalladation/amination domino sequence. Journal of Organometallic Chemistry, 2014, 760, pp.149--155. ⟨10.1016/j.jorganchem.2013.11.010⟩. ⟨hal-01712374⟩
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2011

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Nicolas Auberger, Rok Frlan, Bayan Al-Dabbagh, Ahmed Bouhss, Muriel Crouvoisier, et al.. Synthesis and biological evaluation of potential new inhibitors of the bacterial transferase MraY with a β-ketophosphonate structure. Organic & Biomolecular Chemistry, 2011, 9 (24), pp.8301. ⟨10.1039/c1ob06124k⟩. ⟨hal-02188360⟩
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2010

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Xavier Bantreil, David Madec, Giovanni Poli, Guillaume Prestat, Guillaume Maitro, et al.. Palladium-catalyzed intramolecular allylic alkylation of -sulfinyl carbanions: a new asymmetric route to enantiopure -lactams. Tetrahedron Letters, 2010, 51, pp.1459-1461. ⟨hal-00458722⟩
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Elise Bernoud, Gaetan Le Duc, Xavier Bantreil, Guillaume Prestat, Giovanni Poli, et al.. Aryl sulfoxides from allyl sulfoxides via [2,3]-sigmatropic rearrangement and domino Pd-catalyzed generation / arylation of sulfenate anions. Organic Letters, 2010, 12, pp.320-323. ⟨10.1002/chin.201023082⟩. ⟨hal-00458700⟩
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2009

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Nicolas Auberger, Christine Gravier-Pelletier, Yves Le Merrer. Synthesis of a β-Ketophosphonate Bioisostere of UDP- N -acetylglucosamine. European Journal of Organic Chemistry, 2009, 2009 (20), pp.3323-3326. ⟨10.1002/ejoc.200900399⟩. ⟨hal-02188351⟩
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Christophe Decroos, Yun Li, Gildas Bertho, Yves Frapart, Daniel Mansuy, et al.. Synthetic studies towards diazepanone scaffolds. Tetrahedron: Asymmetry, 2009, 20 (20), pp.2320-2330. ⟨10.1016/j.tetasy.2009.09.022⟩. ⟨hal-03685013⟩
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2008

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Michaël Bosco, Sophie Le Gall, Christophe Rihouey, Samuel Couve-Bonnaire, Muriel Bardor, et al.. 6-Azido d-galactose transfer to N-acetyl-d-glucosamine derivative using commercially available β-1,4-galactosyltransferase. Tetrahedron Letters, 2008, 49 (14), pp.2294-2297. ⟨10.1016/j.tetlet.2008.02.018⟩. ⟨hal-02384444⟩
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2007

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Olivier Monasson, Maryon Ginisty, Gildas Bertho, Christine Gravier-Pelletier, Yves Le Merrer. Efficient synthesis of polyfunctionalised enantiopure diazepanone scaffolds. Tetrahedron Letters, 2007, 48 (46), pp.8149-8152. ⟨10.1016/j.tetlet.2007.09.098⟩. ⟨hal-03685046⟩
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Giuseppe Paladino, David Madec, Guillaume Prestat, Guillaume Maitro, Giovanni Poli, et al.. Oxidative Addition of Ligand-Chelated Palladium(0) to Aryl Halides: Comparison between 1,2-Bisthioethers and 1,2-Bisphosphines. Organometallics, 2007, 26 (2), pp.455. ⟨10.1021/om060846x⟩. ⟨hal-00158052⟩
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Conference papers

2023

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Miryana Hemadi, Romain Briandet, Christine Gravier-Pelletier, John Lomas, Laurent Royon. Nanoparticules métalliques fonctionnalisées pour l'éradication de biofilm à la surface de condenseurs d'eau de rosée. CNRIUT 2023 Saint Pierre - La Réunion, IUT de Saint Pierre, Jun 2023, Saint Pierre (La Réunion), La Réunion. ⟨hal-04326928⟩
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Patents

2019

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François Estour, Michaël Bosco. Nouveaux dimères de cyclodextrines et leurs utilisations comme épurateurs chimiques. France, N° de brevet: FR1910022. 2019. ⟨hal-02376085⟩
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Poster communications

2024

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Michaël Bosco, Nolwenn Periaux-Becquey, Finn Tlatlik, Stéphanie Pradeau, Isabelle Chantret, et al.. Synthesis Of Fluorescent And Fluorogenic Probes To Characterize Lost, The Lysosomal Oligosaccharide Transporter. XXVIII EFMC International Symposium on Medicinal Chemistry, Sep 2024, Rome, Italy. ⟨hal-04773375⟩
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2023

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Michaël Bosco, Younès Bouzidi, Haifei Gao, Stéphanie Pradeau, Isabelle Chantret, et al.. Synthèse de N-acétylchitooligosaccharides fluorescents : Applications à la caractérisation du transport lysosomal d’oligosaccharides (LOST). 3èmes Journées du GDR ChemBio, Jun 2023, Strasbourg, France. ⟨hal-04784597⟩
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2022

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Michaël Bosco, Younès Bouzidi, Haifei Gao, Isabelle Chantret, Sébastien Fort, et al.. Chemical tools for the identification of Lysosomal OligoSaccharide Transporter (LOST). Journées de Chimie Organique de la SFC 2022, Nov 2022, Palaiseau, France. ⟨hal-04784650⟩
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Journal articles

2025

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Riccardo Piccardi, Laurent Micouin. An Overview of the Direct Preparation of Organoaluminum Compounds. Synthesis: Journal of Synthetic Organic Chemistry, In press, ⟨10.1055/a-2669-5996⟩. ⟨hal-05302402⟩
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2024

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Erica Benedetti, Laurent Micouin. Have spirocyclic scaffolds been properly utilized in recent drug discovery efforts?. Expert Opinion on Drug Discovery, 2024, 19 (3), pp.263-266. ⟨10.1080/17460441.2024.2305735⟩. ⟨hal-04736219⟩
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Jules Brom, Antoine Maruani, Serge Turcaud, Sonia Lajnef, Fabienne Peyrot, et al.. [2.2]Paracyclophane-based coumarins: effective organo-photocatalysts for light-induced desulfonylation processes. Organic & Biomolecular Chemistry, 2024, ⟨10.1039/D3OB01711G⟩. ⟨hal-04335222⟩
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Claire Fleurisson, Nessrine Graidia, Jihed Azzouz, Audrey Di Giorgio, Marc Gaysinski, et al.. Design and Evaluation of Azaspirocycles as RNA binders. Chemistry - A European Journal, 2024, 31 (5), pp.e202403518. ⟨10.1002/chem.202403518⟩. ⟨hal-05302366⟩
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ref_biblio
Hadrien Flichot, Annika Sickinger, Jules Brom, Bertrand Lefeuvre, Vincent Dorcet, et al.. Magneto-structural correlation in lanthanide luminescent [2.2]Paracyclophane-based Single-Molecule Magnets. Dalton Transactions, 2024, 53 (19), pp.8191-8201. ⟨10.1039/d4dt00536h⟩. ⟨hal-04571100⟩
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Shiqi Wu, Laurent Micouin, Erica Benedetti. Synthesis of Three-Dimensional Benzophenone Analogues Based on a [2.2]Paracyclophane Scaffold. SYNLETT, 2024, ⟨10.1055/a-2284-4984⟩. ⟨hal-04578271⟩
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Shiqi Wu, Simon Felder, Jules Brom, Fabrice Pointillart, Olivier Maury, et al.. [2.2]Paracyclophanes: From Selective Functionalization to Optical Properties. Advanced Optical Materials, 2024, 12 (21), pp.2400934. ⟨10.1002/adom.202400934⟩. ⟨hal-04614001⟩
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Tuan Zhao, Emmanuelle Sachon, Laurent Micouin, Riccardo Piccardi. α‐Silylated Diazoalkynes: New Tools for Bioconjugation of Proteins. Chemistry - A European Journal, 2024, 30 (19), pp.2042-2048. ⟨10.1002/chem.202302807⟩. ⟨hal-04762411⟩
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2023

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Jules Brom, Antoine Maruani, Laurent Micouin, Erica Benedetti. Light-Driven Reductive Cleavage of Sulfonamides Promoted by Thiourea Organophotosensitizers. Journal of Organic Chemistry, 2023, 88 (9), pp.5923-5935. ⟨10.1021/acs.joc.3c00296⟩. ⟨hal-04267371⟩
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Simon Felder, Marie-Leonie Delcourt, Damian Contant, Rafael Rodríguez, Ludovic Favereau, et al.. Compact CPL emitters based on a [2.2]paracyclophane scaffold: recent developments and future perspectives. Journal of Materials Chemistry C, 2023, 11, pp.2053-2062. ⟨10.1039/d2tc04885j⟩. ⟨hal-04011240⟩
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Claire Fleurisson, Nessrine Graidia, Yann Foricher, Erica Benedetti, Laurent Micouin. Intramolecular Buchwald–Hartwig N -arylation of bicyclic hydrazines: practical access to spiro[indoline-2,3′-piperidines]. Organic & Biomolecular Chemistry, 2023, 21 (17), pp.3542-3546. ⟨10.1039/D3OB00406F⟩. ⟨hal-04267385⟩
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2022

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Simon Felder, Marie-Leonie Delcourt, Manon Bousquet, Denis Jacquemin, Rafael Rodriguez, et al.. Planar Chiral Analogues of PRODAN Based on a [2.2]Paracyclophane Scaffold: Synthesis and Photophysical Studies. Journal of Organic Chemistry, 2022, 87 (1), pp.147-158. ⟨10.1021/acs.joc.1c02071⟩. ⟨hal-03512519⟩
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Simon Felder, Corinne Sagné, Erica Benedetti, Laurent Micouin. Small-Molecule 3D Ligand for RNA Recognition: Tuning Selectivity through Scaffold Hopping. ACS Chemical Biology, 2022, 17 (11), pp.3069-3076. ⟨10.1021/acschembio.2c00171⟩. ⟨hal-04035021⟩
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2021

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Simon Felder, Laurent Micouin, Erica Benedetti. Para‐Functionalization of N‐Substituted 4‐amino[2.2]paracyclophanes by Regioselective Formylation. European Journal of Organic Chemistry, 2021, pp.4015. ⟨10.1002/ejoc.202100288⟩. ⟨hal-03297447⟩
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Simon Felder, Shiqi Wu, Jules Brom, Laurent Micouin, Erica Benedetti. Enantiopure planar chiral [2.2]paracyclophanes: Synthesis and applications in asymmetric organocatalysis. Chirality, 2021, 33 (9), pp.506-527. ⟨10.1002/chir.23335⟩. ⟨hal-03366196⟩
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Shiqi Wu, Laura Abad Galán, Margaux Roux, François Riobé, Boris Le Guennic, et al.. Tuning the excited state properties of [2.2]paracyclophane-based antennas to ensure efficient sensitization of lanthanide ions or singlet oxygen generation. Inorganic Chemistry, 2021, 60 (60), pp.21. ⟨10.1021/acs.inorgchem.1c01986⟩. ⟨hal-03407500⟩
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2020

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Céline Aubry, Paolo Clerici, Claude Gerbaud, Laurent Micouin, Jean-Luc Pernodet, et al.. Revised structure of anthelvencin A and characterization of the anthelvencin biosynthetic gene cluster. ACS Chemical Biology, 2020, ⟨10.1021/acschembio.9b00960⟩. ⟨hal-02502312⟩
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Claire Fleurisson, Erica Benedetti, Laurent Micouin. Cyclic cis-1,3-Diamines Derived from Bicyclic Hydrazines: Synthesis and Applications. SYNLETT, 2020, ⟨10.1055/s-0040-1707324⟩. ⟨hal-03003668⟩
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2019

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Marie-Leonie Delcourt, Corentin Reynaud, Serge Turcaud, Ludovic Favereau, Jeanne Crassous, et al.. 3D Coumarin Systems Based on [2.2]Paracyclophane Synthesis, Spectroscopic Characterization, and Chiroptical Properties. Journal of Organic Chemistry, 2019, 84 (2), pp.888-899. ⟨10.1021/acs.joc.8b02773⟩. ⟨hal-02049506⟩
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Marie-Leonie Delcourt, Simon Felder, Serge Turcaud, Corina Pollok, Christian Merten, et al.. Highly Enantioselective Asymmetric Transfer Hydrogenation: A Practical and Scalable Method To Efficiently Access Planar Chiral [2.2]Paracyclophanes. Journal of Organic Chemistry, 2019, ⟨10.1021/acs.joc.9b00372⟩. ⟨hal-02113386⟩
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Tuan Zhao, Laurent Micouin, Riccardo Piccardi. Synthesis of Organometallic Compounds in Flow. Helvetica Chimica Acta, 2019, 102 (11), ⟨10.1002/hlca.201900172⟩. ⟨hal-02346965⟩
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2018

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Aurélie Blond, Serge Turcaud, Thomas Lecourt, Laurent Micouin. Diastereoselective Ring Homologation of Bicyclic Hydrazines: Access to cis -1,3-Diaminocyclohexitols. ACS Omega, 2018, 3 (11), pp.15302-15307. ⟨10.1021/acsomega.8b02910⟩. ⟨hal-02186751⟩
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Marie-Leonie Delcourt, Simon Felder, Erica Benedetti, Laurent Micouin. Highly Enantioselective Desymmetrization of Centrosymmetric pseudo - para -Diformyl[2.2]paracyclophane via Asymmetric Transfer Hydrogenation. ACS Catalysis, 2018, 8 (7), pp.6612-6616. ⟨10.1021/acscatal.8b01872⟩. ⟨hal-02113395⟩
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Riccardo Piccardi, Serge Turcaud, Erica Benedetti, Laurent Micouin. Synthesis and Reactivity of Mixed Dimethylalkynylaluminum Reagents. Synthesis: Journal of Synthetic Organic Chemistry, 2018, 51 (01), pp.97-106. ⟨10.1055/s-0037-1610392⟩. ⟨hal-02113388⟩
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Tuan Zhao, Riccardo Piccardi, Laurent Micouin. Rapid and Effective Synthesis of α-Acyloxy-α-alkynyltrimethylsilanes. Organic Letters, 2018, 20 (16), pp.5015-5018. ⟨10.1021/acs.orglett.8b02165⟩. ⟨hal-02113392⟩
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2017

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E. Benedetti, M.-L. Delcourt, B. Gatin-Fraudet, S. Turcaud, L. Micouin. Synthesis and photophysical studies of through-space conjugated [2.2]paracyclophane-based naphthalene fluorophores. RSC Advances, 2017, 7 (80), pp.50472-50476. ⟨10.1039/C7RA10038H⟩. ⟨hal-02113405⟩
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Hélène Guyon, François Mavré, Marjorie Catala, Serge Turcaud, Franck Brachet, et al.. Use of a redox probe for an electrochemical RNA–ligand binding assay in microliter droplets. Chemical Communications, 2017, 53 (6), pp.1140-1143. ⟨10.1039/c6cc07785d⟩. ⟨hal-02185366⟩
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Antoine Joosten, Mélissa Boultadakis-Arapinis, V. Gandon, L. Micouin, Thomas Lecourt. Substitution of the Participating Group of Glycosyl Donors by a Halogen Atom: Influence on the Rearrangement of Transient Orthoesters Formed during Glycosylation Reactions. Journal of Organic Chemistry, 2017, 82 (6), pp.3291-3297. ⟨10.1021/acs.joc.6b03088⟩. ⟨hal-02046285⟩
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2016

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Karen Amirbekyan, Nicolas Duchemin, Erica Benedetti, Rinah Joseph, Aude Colon, et al.. Design, Synthesis, and Binding Affinity Evaluation of Hoechst 33258 Derivatives for the Development of Sequence-Specific DNA-Based Asymmetric Catalysts. ACS Catalysis, 2016, 6 (5), pp.3096-3105. ⟨10.1021/acscatal.6b00495⟩. ⟨hal-02197253⟩
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Thibaut Courant, Rahul Kumar, Serge Turcaud, Laurent Micouin. Rhodium(II)-Alkynyl Carbenoids Insertion into Si–H bonds: An Entry to Propargylic Geminal Bis(silanes). Organic Letters, 2016, 18 (19), pp.4818-4820. ⟨10.1021/acs.orglett.6b02264⟩. ⟨hal-02186746⟩
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Nicolas Duchemin, Erica Benedetti, Lucas Bethge, Stefan Vonhoff, Sven Klussmann, et al.. Expanding biohybrid-mediated asymmetric catalysis into the realm of RNA. Chemical Communications, 2016, 52 (55), pp.8604-8607. ⟨10.1039/c6cc03540j⟩. ⟨hal-02197262⟩
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Riccardo Piccardi, Anaïs Coffinet, Erica Benedetti, Serge Turcaud, Laurent Micouin. Continuous Flow Synthesis of Dimethylalkynylaluminum Reagents. Synthesis: Journal of Synthetic Organic Chemistry, 2016, 48 (19), pp.3272-3278. ⟨10.1055/s-0035-1561484⟩. ⟨hal-02134269⟩
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2015

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Erica Benedetti, Nicolas Duchemin, Lucas Bethge, Stefan Vonhoff, Sven Klussmann, et al.. DNA-cellulose: an economical, fully recyclable and highly effective chiral biomaterial for asymmetric catalysis. Chemical Communications, 2015, 51 (28), pp.6076-6079. ⟨10.1039/C4CC10190A⟩. ⟨hal-03554623⟩
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Laura Iannazzo, Erica Benedetti, Marjorie Catala, Mélanie Etheve-Quelquejeu, Carine Tisné, et al.. Monitoring of reversible boronic acid–diol interactions by fluorine NMR spectroscopy in aqueous media. Organic & Biomolecular Chemistry, 2015, 13 (33), pp.8817-8821. ⟨10.1039/c5ob01362c⟩. ⟨hal-03544508⟩
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2014

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Renaud Barbeyron, Erica Benedetti, Janine Cossy, Jean-Jacques Vasseur, Stellios Arseniyadis, et al.. Recent developments in alkyne borylations.. Tetrahedron, 2014, 70 (45), pp.8431-8452. ⟨10.1016/j.tet.2014.06.026⟩. ⟨hal-01078195⟩
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Mélissa Boultadakis-Arapinis, Vincent Gandon, Elise Prost, Laurent Micouin, Thomas Lecourt. Electronic Effects in Carbene-Mediated C H Bond Functionalization: An Experimental and Theoretical Study. Advanced Synthesis and Catalysis, 2014, 356 (11-12), pp.2493-2450. ⟨10.1002/adsc.201300984⟩. ⟨hal-01141166⟩
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Rahul Kumar, Serge Turcaud, Laurent Micouin. The Reaction of Dimethylalkynylaluminum Reagents with Trimethylsilyldiazomethane: Original Reactivity Leading to New α-Silylated Alkynyl Hydrazones. Organic Letters, 2014, 16 (23), pp.6192-6195. ⟨10.1021/ol503113d⟩. ⟨hal-02185384⟩
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2013

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Aurélie Blond, Paul Dockerty, Raquel Alvarez, Serge Turcaud, Thomas Lecourt, et al.. Modular Access to N-Substituted cis -3,5-Diaminopiperidines. Journal of Organic Chemistry, 2013, 78 (23), pp.12236-12242. ⟨10.1021/jo401994y⟩. ⟨hal-02186757⟩
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Mélissa Boultadakis-Arapinis, Elise Prost, Vincent Gandon, Pascale Lemoine, Serge Turcaud, et al.. Carbene-Mediated Functionalization of the Anomeric C-H Bond of Carbohydrates: Scope and Limitations. Chemistry - A European Journal, 2013, 19 (19), pp.6052-6066. ⟨10.1002/chem.201203725⟩. ⟨hal-02185449⟩
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2012

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Erica Benedetti, Michela Lomazzi, Francesco Tibiletti, Jean-Philippe Goddard, Louis Fensterbank, et al.. Synthesis of Nitrogen-Containing Heterocycles via Ring-Closing Ene-Ene and Ene-Yne Metathesis Reactions: An Easy Access to 1-and 2-Benzazepine Scaffolds and Five- and Six-Membered Lactams. Synthesis: Journal of Synthetic Organic Chemistry, 2012, 44 (22), pp.3523-3533. ⟨10.1055/s-0032-1317352⟩. ⟨hal-01397631⟩
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Thomas Lombès, Roba Moumné, Valéry Larue, Elise Prost, Marjorie Catala, et al.. Investigation of RNA-Ligand Interactions by (19) F NMR Spectroscopy Using Fluorinated Probes.. Angewandte Chemie International Edition, 2012, 51 (38), pp.9530-9534. ⟨10.1002/anie.201204083⟩. ⟨hal-00724894⟩
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Roba Moumné, Marjorie Catala, Valéry Larue, Laurent Micouin, Carine Tisné. Fragment-based design of small RNA binders: promising developments and contribution of NMR.. Biochimie, 2012, 94 (7), pp.1607-1619. ⟨10.1016/j.biochi.2012.02.002⟩. ⟨hal-00692356⟩
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2011

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A. Blond,, Roba Moumné, G. Begis,, M. Pasco, Thomas Lecourt, et al.. Rhodium(II) carbene-mediated modification of 2-deoxystreptamine surrogates. Journal of Organic Chemistry, 2011, 52 (25), pp.3201-3203. ⟨hal-00649113⟩
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Olivier Jackowski, Thomas Lecourt, Laurent Micouin. Direct Synthesis of Polysubstituted Aluminoisoxazoles and Pyrazoles by a Metalative Cyclization. Organic Letters, 2011, 13 (20), pp.5664-5667. ⟨10.1021/ol202389u⟩. ⟨hal-02185376⟩
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Morgane Pasco, Roba Moumné, Thomas Lecourt, Laurent Micouin. Stereoselective synthesis of fluorinated 1,3-cis-diaminocyclopentanes.. Journal of Organic Chemistry, 2011, 76 (12), pp.5137-42. ⟨10.1021/jo2001512⟩. ⟨hal-00649119⟩
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Morgane Pasco, Roba Moumné, Thomas Lecourt, Laurent Micouin. Stereoselective Synthesis of Fluorinated 1,3- cis -Diaminocyclopentanes. Journal of Organic Chemistry, 2011, 76 (12), pp.5137-5142. ⟨10.1021/jo2001512⟩. ⟨hal-02186896⟩
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2010

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Roba Moumné, Morgane Pasco, Elise Prost, Thomas Lecourt, Laurent Micouin, et al.. Fluorinated diaminocyclopentanes as chiral sensitive NMR probes of RNA structure.. Journal of the American Chemical Society, 2010, 132 (38), pp.13111-3. ⟨10.1021/ja1037885⟩. ⟨hal-00614591⟩
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Roba Moumné, Valéry Larue, Bili Seijo, Thomas Lecourt, Laurent Micouin, et al.. Tether influence on the binding properties of tRNALys3 ligands designed by a fragment-based approach.. Organic & Biomolecular Chemistry, 2010, 8 (5), pp.1154-9. ⟨10.1039/b921232a⟩. ⟨hal-00596199⟩
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Yuhan Zhou, Thomas Lecourt, Laurent Micouin. Direct Synthesis of 1,4-Disubstituted-5-alumino-1,2,3-triazoles: Copper-Catalyzed Cycloaddition of Organic Azides and Mixed Aluminum Acetylides. Angewandte Chemie International Edition, 2010, 49 (14), pp.2607-2610. ⟨10.1002/anie.200907016⟩. ⟨hal-02185392⟩
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2008

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Chloée Bournaud, Thomas Lecourt, Laurent Micouin, Catherine Méliet, Francine Agbossou-Niedercorn. Desymmetrization of meso-Bicyclic Hydrazines by Rhodium-Catalyzed Enantioselective Hydroformylation. European Journal of Organic Chemistry, 2008, 2008 (13), pp.2298-2302. ⟨10.1002/ejoc.200800116⟩. ⟨hal-02185573⟩
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Thomas Lombès, Guillaume Bégis, Frédérique Maurice, Serge Turcaud, Thomas Lecourt, et al.. NMR-Guided Fragment-Based Approach for the Design of AAC(6′)-Ib Ligands. ChemBioChem, 2008, 9 (9), pp.1368-1371. ⟨10.1002/cbic.200700677⟩. ⟨hal-02185444⟩
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2007

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Florence Chung, Carine Tisné, Thomas Lecourt, Frédéric Dardel, Laurent Micouin. NMR-guided fragment-based approach for the design of tRNA(Lys3) ligands.. Angewandte Chemie International Edition, 2007, 46 (24), pp.4489-91. ⟨10.1002/anie.200605201⟩. ⟨hal-00218344⟩
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2006

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Martine Bonin, Laurent Micouin, Ariane Chauveau. Asymmetric 1,3-Dipolar Cycloadditions of Cyclic Stabilized Ylides Derived from Chiral 1,2-Amino Alcohols. SYNLETT, 2006, 2006 (15), pp.2349-2363. ⟨10.1055/s-2006-949626⟩. ⟨hal-02185347⟩
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Frédérique Maurice, Guillaume Bégis, Laurent Micouin, Frédéric Dardel. NMR identification of ligands of aminoglycoside resistance enzymes. Comptes Rendus. Chimie, 2006, 9, pp.413-419. ⟨hal-00021873⟩
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2004

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Christophe Feuvrie, Jérôme Blanchet, Martine Bonin, Laurent Micouin. Synthesis and reactivity of mixed alkynylalanes by direct triethylamine-catalyzed alumination of terminal alkynes.. Organic Letters, 2004, 6 (14), pp.2333-6. ⟨10.1021/ol049346v⟩. ⟨hal-00909871⟩
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2003

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S. Cutri, A. Chiaroni, M. Bonin, L. Micouin, H.-P. Husson. Practical Asymmetric Synthesis of 1,2-Diamines in the 3-Aminoazepane Series. Journal of Organic Chemistry, 2003, 68 (7), pp.2645-2651. ⟨10.1021/jo026711s⟩. ⟨hal-02186903⟩
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Yen Vo-Hoang, Laurent Micouin, Catherine Ronet, Gabriel Gachelin, Martine Bonin. Total Enantioselective Synthesis and In Vivo Biological Evaluation of a Novel Fluorescent BODIPY α-Galactosylceramide. ChemBioChem, 2003, 4 (1), pp.27-33. ⟨10.1002/cbic.200390009⟩. ⟨hal-03531886⟩
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2002

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Jerome Blanchet, M. Bonin, L. Micouin. Recent progress in the asymmetric synthesis of α-substituted propargylamines. Organic Preparations and Procedures International : The New Journal for Organic Synthesis, 2002, 34 (5), pp.467-492. ⟨10.1080/00304940209355765⟩. ⟨hal-02328004⟩
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Jérôme Blanchet, Martine Bonin, Laurent Micouin, Henri-Philippe Husson. Isomerization of Chiral Non-Racemic α-Substituted Propargylic Amines to Terminal Acetylenes. European Journal of Organic Chemistry, 2002, 2002 (15), pp.2598-2602. ⟨10.1002/1099-0690(200208)2002:15<2598::AID-EJOC2598>3.0.CO;2-V⟩. ⟨hal-02185592⟩
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Alejandro Pérez Luna, Martine Bonin, Laurent Micouin, Henri-Philippe Husson. Reversal of Enantioselectivity in the Asymmetric Rhodium- versus Iridium-Catalyzed Hydroboration of Meso Substrates. Journal of the American Chemical Society, 2002, 124 (41), pp.12098-12099. ⟨10.1021/ja026714m⟩. ⟨hal-02185596⟩
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A. Pérez Luna, M.-A Ceschi, M. Bonin, L. Micouin, H.-P. Husson, et al.. Enantioselective Desymmetrization of Meso Bicyclic Hydrazines: A Novel Approach to the Asymmetric Synthesis of Polysubstituted Amino Cyclopentanic Cores. Journal of Organic Chemistry, 2002, 67 (10), ⟨10.1021/jo011190e⟩. ⟨hal-02186763⟩
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Jordi Piró, Pilar Forns, Jérôme Blanchet, Martine Bonin, Laurent Micouin, et al.. Asymmetric synthesis of β-pseudopeptides from chiral 3,4-aziridinolactams. Tetrahedron: Asymmetry, 2002, 13 (9), pp.995-1004. ⟨10.1016/S0957-4166(02)00221-5⟩. ⟨hal-02328007⟩
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2001

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Valérie Alezra, Martine Bonin, Laurent Micouin, Clotilde Policar, Henri-Philippe Husson. The Origin of Chemical and Configurational Stability of Chiral Nonracemic Tert-Butyl Aziridinecarboxylate Anions. European Journal of Organic Chemistry, 2001, 2001 (13), pp.2589-2594. ⟨10.1002/1099-0690(200107)2001:13<2589::AID-EJOC2589>3.0.CO;2-Y⟩. ⟨hal-02011971⟩
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Jérôme Blanchet, Martine Bonin, Laurent Micouin, Henri-Philippe Husson. Asymmetric synthesis of α-substituted propynyl amines. Application to the preparation of a polysubstituted dihydroisoindoline framework. Tetrahedron Letters, 2001, 42 (18), pp.3171-3173. ⟨10.1016/S0040-4039(01)00356-2⟩. ⟨hal-02328009⟩
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2000

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Jérôme Blanchet, Martine Bonin, Laurent Micouin, Henri-Philippe Husson. [2,3]-Meisenheimer rearrangement of N-allyl phenylglycinol derivatives. NC versus CC chirality transfer. Tetrahedron Letters, 2000, 41 (43), pp.8279-8283. ⟨10.1016/S0040-4039(00)01460-X⟩. ⟨hal-02328033⟩
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J. Blanchet, M. Bonin, L. Micouin, H. P. Husson. Synthesis of enantiomerically pure alpha-substituted propargylic amines by reaction of organoaluminum reagents with oxazolidines.. Journal of Organic Chemistry, 2000, 65 (20), pp.6423-6. ⟨hal-00909874⟩
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Jerome Blanchet, M. Bonin, L. Micouin, H.-P. Husson. Synthesis of Enantiomerically Pure α-Substituted Propargylic Amines by Reaction of Organoaluminum Reagents with Oxazolidines. Journal of Organic Chemistry, 2000, 65 (20), pp.6423-6426. ⟨10.1021/jo0003706⟩. ⟨hal-02328014⟩
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1999

ref_biblio
Jérôme Blanchet, Martine Bonin, Angèle Chiaroni, Laurent Micouin, Claude Riche, et al.. Diastereoselective alkynylation of chiral non-racemic oxazolidines with mixed organoaluminum compounds. Tetrahedron Letters, 1999, 40 (15), pp.2935-2938. ⟨10.1016/S0040-4039(99)00328-7⟩. ⟨hal-02328037⟩
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Book sections

2025

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L. Micouin, R. Piccardi. Organoaluminum Reagents. Comprehensive Organic Synthesis, Elsevier; Elsevier, pp.45-69, 2025, ⟨10.1016/B978-0-323-96025-0.00041-7⟩. ⟨hal-05304382⟩
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2016

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Riccardo Piccardi, Laurent Micouin, Olivier Jackowski. The Chemistry of Alkynylaluminum Species. Marek, Ilan. PATAI'S Chemistry of Functional Groups, John Wiley & Sons, Ltd, pp.1--47, 2016, 978-0-470-68253-1. ⟨10.1002/9780470682531.pat0832⟩. ⟨hal-02891076⟩
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Françoise Schaefers, Tobias A. M. Gulder, Cyril Bressy, Michaël Smietana, Erica Benedetti, et al.. Polyketides. Zografos A. From Biosynthesis to Total Synthesis: Strategies and Tactics for Natural Products, Wiley, pp.21-129, 2016, ⟨10.1002/9781118754085.ch2⟩. ⟨hal-01415109⟩
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2014

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Fabrice Chemla, Franck Ferreira, Olivier Jackowski, Laurent Micouin, Alejandro Perez-Luna. Carbon\textendashCarbon Bond Forming Reactions Mediated by Organozinc Reagents. de Meijere, Armin and Bräse, Stefan and Oestreich, Martin. Metal-Catalyzed Cross-Coupling Reactions and More, Wiley-VCH Verlag GmbH & Co. KGaA, pp.279--364, 2014, 978-3-527-65558-8. ⟨10.1002/9783527655588.ch4⟩. ⟨hal-02891142⟩
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Fabrice Chemla, Franck Ferreira, Alejandro Perez-Luna, Laurent Micouin, Olivier Jackowski. Carbon\textendashCarbon Bond-Forming Reactions Mediated by Organomagnesium Reagents. de Meijere, Armin and Bräse, Stefan and Oestreich, Martin. Metal-Catalyzed Cross-Coupling Reactions and More, Wiley-VCH Verlag GmbH & Co. KGaA, pp.365--422, 2014, 978-3-527-65558-8. ⟨10.1002/9783527655588.ch5⟩. ⟨hal-02891143⟩
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Poster communications

2018

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Céline Aubry, Paolo Clerici, Laurent Micouin, Jean-Luc Pernodet, Sylvie Lautru. COMBINATORIAL BIOSYNTHESIS OF NON-RIBOSOMAL PEPTIDES, THE EXAMPLE OF PYRROLAMIDES. 5èmes journées du GDR MufoPAM, Oct 2018, Paris, France. ⟨hal-02367767⟩
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Journal articles

2025

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Jules Bresson, Katie Burke, Mélanie Ethève‐quelquejeu, Laura Iannazzo, Kevin Cariou. Metal‐Catalyzed Cross‐Coupling for the Synthesis of β‐Lactam Drugs and Related Chemical Probes. ChemMedChem, 2025, 20 (9), pp.e202400960. ⟨10.1002/cmdc.202400960⟩. ⟨hal-05287299⟩
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Katie Burke, Quentin Herail, Ines Zerguine, Catherine Bougault, Michel Arthur, et al.. Optimization of prodrug activation by enzymatic cleavage of the β‐lactam ring of carbapenems. Chemistry - A European Journal, 2025, 31 (46), pp.e01534. ⟨10.1002/chem.202501534⟩. ⟨hal-05287283⟩
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Jianxun Du, Batoul Mahcene, Valerii Martynov, Elisa Frezza, Christelle Vasnier, et al.. Investigation of a squaramide motif as a bioisostere of the amino-acid group of S-adenosyl-L-methionine and its functional impact on RNA methylation. Communications Chemistry, 2025, 8 (1), pp.244. ⟨10.1038/s42004-025-01627-7⟩. ⟨hal-05287286v1⟩
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Jianxun Du, Bastien Felipe, Dylan Coelho, Laura Iannazzo, Alexandre David, et al.. Synthetic approaches to bis-adenosine derivatives as potential bisubstrates of RNA methyltransferases. Organic & Biomolecular Chemistry, 2025, 23 (24), pp.5887-5896. ⟨10.1039/D5OB00758E⟩. ⟨hal-05139585⟩
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Cécilia Hognon, Ameni Ben Abdeljaoued, Pierre Hardouin, Mélanie Etheve-Quelquejeu, Bruno Sargueil, et al.. A multiscale study to characterize SHAPE probe/ RNA molecules pre-reactive complex and its role in initiating the SHAPE reaction. Journal of Chemical Information and Modeling, 2025, ⟨10.1021/acs.jcim.5c00812⟩. ⟨hal-05226372⟩
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Laura Iannazzo, Emmanuelle Braud, Matthieu Fonvielle, Mélanie Etheve-Quelquejeu. Synthesis of RNA conjugates as bisubstrates for the study of transferases. Comptes Rendus. Chimie, 2025, 28 (G1), pp.111-129. ⟨10.5802/crchim.356⟩. ⟨hal-05287289⟩
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Catherine Laurent, Gabrielle Poncet, Tristan Herskovits, Rodolphe Alves de Sousa, Laurent Le Corre, et al.. Inhibition of the Parkinson’s Disease-Related Protein DJ-1 by Endogenous Neurotoxins of the 1,2,3,4-Tetrahydroisoquinoline Family. ACS Chemical Neuroscience, 2025, 16 (6), pp.1034-1042. ⟨10.1021/acschemneuro.4c00559⟩. ⟨hal-05291792⟩
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Nicolas Mathas, Emmanuelle Braud, Erwan Galardon, Lucie Larigot, Mélanie Etheve-Quelquejeu, et al.. Park7 (DJ-1), a Parkinson-associated glyoxalase/deglycase: characterization of enzymatic activity in biological samples using fluorescence-based liquid chromatography. Biochimie, 2025, 235, pp.113-121. ⟨10.1016/j.biochi.2025.06.005⟩. ⟨hal-05139644⟩
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2024

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Margaux Cescato, Laurence Cuisset, Laurent Le Corre, Mathieu Rodero, Sophie Georgin-Lavialle. Diagnosis traps for patients with acquired NLRP3 mutation. European Journal of Internal Medicine, 2024, 125 (16), pp.129-131. ⟨10.1016/j.ejim.2024.01.028⟩. ⟨hal-05073743⟩
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2023

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Leeroy Baron, Justine Hadjerci, Leishemba Thoidingjam, Marina Plays, Romain Bucci, et al.. PSL Chemical Biology Symposia Third Edition: A Branch of Science in its Explosive Phase. ChemBioChem, 2023, 24 (8), pp.e202300093. ⟨10.1002/cbic.202300093⟩. ⟨hal-04092530⟩
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Dylan Coelho, Laurent Le Corre, Karolina Bartosik, Laura Iannazzo, Emmanuelle Braud, et al.. Synthesis of Bisubstrate Analogues for RNA Methylation Studies using two Transition‐Metal‐Catalyzed Reactions. Chemistry - A European Journal, 2023, 29 (44), ⟨10.1002/chem.202301134⟩. ⟨hal-04246592⟩
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Ivan Corbeski, Pablo Andrés Vargas-Rosales, Rajiv Kumar Bedi, Jiahua Deng, Dylan Coelho, et al.. The catalytic mechanism of the RNA methyltransferase METTL3. eLife, 2023, ⟨10.7554/eLife.92537.1⟩. ⟨hal-05287291⟩
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Antoine Fayand, Margaux Cescato, Laurent Le Corre, Alexandre Terré, Margaux Wacheux, et al.. Pathogenic variants in the NLRP3 LRR domain at position 861 are responsible for a boost-dependent atypical CAPS phenotype.. Journal of Allergy and Clinical Immunology, 2023, 152 (5), pp.1303-1311.e1. ⟨10.1016/j.jaci.2023.07.006⟩. ⟨hal-04182567⟩
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Antoine Fayand, Véronique Hentgen, Céline Posseme, Carole Lacout, Capucine Picard, et al.. Successful treatment of JAK1 associated inflammatory disease. Journal of Allergy and Clinical Immunology, 2023, 152 (4), pp.972-983. ⟨10.1016/j.jaci.2023.06.004⟩. ⟨hal-04137977⟩
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Erwan Galardon, Nicolas Mathas, Dominique Padovani, Laurent Le Corre, Gabrielle Poncet, et al.. Persulfidation of DJ-1: Mechanism and Consequences. Biomolecules, 2023, 13 (1), pp.27. ⟨10.3390/biom13010027⟩. ⟨hal-03920432⟩
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Camélia Kitoun, Saidbakhrom Saidjalolov, Delphine Bouquet, Fabiola Djago, Quentin Blancart-Remaury, et al.. Traceless Staudinger Ligation to Access Stable Aminoacyl- or Peptidyl-Dinucleotide. ACS Omega, 2023, 8 (4), pp.3850-3860. ⟨10.1021/acsomega.2c06135⟩. ⟨hal-04294940⟩
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Laurent Le Corre, Dominique Padovani. Mechanism-based and computational modeling of hydrogen sulfide biogenesis inhibition: interfacial inhibition. Scientific Reports, 2023, 13 (1), pp.7287. ⟨10.1038/s41598-023-34405-3⟩. ⟨hal-04285208⟩
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2022

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Chiara Figazzolo, Frédéric Bonhomme, Saidbakhrom Saidjalolov, Mélanie Ethève-Quelquejeu, Marcel Hollenstein. Enzymatic synthesis of vancomycin-modified DNA. Molecules, 2022, 27 (24), pp.8927. ⟨10.3390/molecules27248927⟩. ⟨hal-03927068⟩
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Vincent Meynier, Laura Iannazzo, Marjorie Catala, Stephanie Oerum, Emmanuelle Braud, et al.. Synthesis of RNA-cofactor conjugates and structural exploration of RNA recognition by an m6A RNA methyltransferase. Nucleic Acids Research, 2022, ⟨10.1093/nar/gkac354⟩. ⟨hal-03689976⟩
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Khawla Nouri, Nicolas Pietrancosta, Laurent Le Corre, Patrick Dansette, Daniel Mansuy, et al.. Human Orphan Cytochrome P450 2U1 Catalyzes the ω-Hydroxylation of Leukotriene B4. International Journal of Molecular Sciences, 2022, 23 (23), pp.14615. ⟨10.3390/ijms232314615⟩. ⟨hal-03957648⟩
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Martin Oliver, Laurent Le Corre, Mélanie Poinsot, Michaël Bosco, Hongwei Wan, et al.. A Sub-Micromolar MraYAA Inhibitor with an Aminoribosyl Uridine Structure and a (S,S)-Tartaric Diamide: Synthesis, Biological Evaluation and Molecular Modeling. Molecules, 2022, 27 (6), pp.1769. ⟨10.3390/molecules27061769⟩. ⟨hal-03632451⟩
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Lauriane Rietmeyer, Inès Li de la Sierra-Gallay, Guy Schepers, Delphine Dorchêne, Laura Iannazzo, et al.. Amino-acyl tXNA as inhibitors or amino acid donors in peptide synthesis. Nucleic Acids Research, 2022, ⟨10.1093/nar/gkac1023⟩. ⟨hal-03879768⟩
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Hongwei Wan, Raja Ben Othman, Laurent Le Corre, Mélanie Poinsot, Martin Oliver, et al.. New MraYAA Inhibitors with an Aminoribosyl Uridine Structure and an Oxadiazole. Antibiotics, 2022, 11 (9), pp.1189. ⟨10.3390/antibiotics11091189⟩. ⟨hal-03805942⟩
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2021

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Flavie Bouchet, Heiner Atze, Michel Arthur, Mélanie Ethève-Quelquejeu, Laura Iannazzo. Traceless Staudinger Ligation To Introduce Chemical Diversity on β-Lactamase Inhibitors of Second Generation. Organic Letters, 2021, 23 (20), pp.7755-7758. ⟨10.1021/acs.orglett.1c02741⟩. ⟨hal-03647098⟩
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Aurore Dumond, Etienne Brachet, Jérôme Durivault, Valérie Vial, Anna Puszko, et al.. Neuropilin 1 and Neuropilin 2 gene invalidation or pharmacological inhibition reveals their relevance for the treatment of metastatic renal cell carcinoma. Journal of experimental & clinical cancer research, 2021, 40, pp.33. ⟨10.1186/s13046-021-01832-x⟩. ⟨hal-03132345⟩
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Camélia Kitoun, Matthieu Fonvielle, Michel Arthur, Mélanie Etheve‐quelquejeu, Laura Iannazzo. Traceless Staudinger Ligation for Bioconjugation of RNA. Current Protocols, 2021, 1 (2), ⟨10.1002/cpz1.42⟩. ⟨hal-03647120⟩
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Martin Oliver, Laurent Le Corre, Mélanie Poinsot, Alessandra Corio, Léa Madegard, et al.. Synthesis, biological evaluation and molecular modeling of urea-containing MraY inhibitors. Organic & Biomolecular Chemistry, 2021, 19 (26), pp.5844-5866. ⟨10.1039/D1OB00710F⟩. ⟨hal-03432617⟩
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Claire Pujol, Anne Legrand, Livia Parodi, Priscilla Thomas, Fanny Mochel, et al.. Implication of folate deficiency in CYP2U1 loss of function. Journal of Experimental Medicine, 2021, 218 (11), pp.e20210846. ⟨10.1084/jem.20210846⟩. ⟨pasteur-03349041⟩
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Lauriane Rietmeyer, Nicolas Fix-Boulier, Chloé Le Fournis, Laura Iannazzo, Camelia Kitoun, et al.. Partition of tRNAGly isoacceptors between protein and cell-wall peptidoglycan synthesis in Staphylococcus aureus. Nucleic Acids Research, 2021, 49 (2), pp.684-699. ⟨10.1093/nar/gkaa1242⟩. ⟨hal-03201622⟩
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Saidbakhrom Saidjalolov, Zainab Edoo, Matthieu Fonvielle, Louis Mayer, Laura Iannazzo, et al.. Synthesis of carbapenems containing peptidoglycanmimetics and inhibition of the cross-linking activity of a transpeptidase of the L,D specificity. Chemistry - A European Journal, 2021, 27 (10), pp.3542-3551. ⟨10.1002/chem.202004831⟩. ⟨hal-03184204⟩
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Saidbakhrom Saidjalolov, Emmanuelle Braud, Zainab Edoo, Laura Iannazzo, Filippo Rusconi, et al.. Click and Release Chemistry for Activity-Based Purification of β-Lactam Targets. Chemistry - A European Journal, 2021, 27 (28), pp.7687-7695. ⟨10.1002/chem.202100653⟩. ⟨hal-03281379⟩
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Tongtong Zhang, Laurent Le Corre, Olivia Reinaud, Benoit Colasson. A Promising Approach for Controlling the Second Coordination Sphere of Biomimetic Metal Complexes: Encapsulation in a Dynamic Hydrogen‐Bonded Capsule. Chemistry - A European Journal, 2021, 27 (1), pp.434-443. ⟨10.1002/chem.202004370⟩. ⟨hal-03154347⟩
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2020

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Colette Atdjian, Dylan Coelho, Laura Iannazzo, Mélanie Etheve-Quelquejeu, Emmanuelle Braud. Synthesis of triazole-linked SAM-adenosine 2 conjugates: functionalization of adenosine at N-1 or N-6 position without protecting groups. Molecules, 2020, 25 (14), pp.3241. ⟨10.3390/molecules25143241⟩. ⟨hal-02915430⟩
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Flavie Bouchet, Heiner Atze, Matthieu Fonvielle, Zainab Edoo, Michel Arthur, et al.. Diazabicyclooctane Functionalization for Inhibition of β-Lactamases from Enterobacteria. Journal of Medicinal Chemistry, 2020, 63 (10), pp.5257-5273. ⟨10.1021/acs.jmedchem.9b02125⟩. ⟨hal-03646829v2⟩
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Jeanne Fichez, Cathia Soulié, Laurent Le Corre, Sophie Sayon, Stéphane Priet, et al.. Discovery, SAR study and ADME properties of methyl 4-amino-3-cyano-1-(2-benzyloxyphenyl)-1 H -pyrazole-5-carboxylate as an HIV-1 replication inhibitor. RSC Medicinal Chemistry, 2020, 11 (5), pp.577-582. ⟨10.1039/D0MD00025F⟩. ⟨hal-03030936⟩
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Camelia Kitoun, Matthieu Fonvielle, Nicolas Sakkas, Manon Lefresne, Fabiola Djago, et al.. Phosphine-Mediated Bioconjugation of the 3′-End of RNA. Organic Letters, 2020, 22 (20), pp.8034-8038. ⟨10.1021/acs.orglett.0c02982⟩. ⟨hal-02996863⟩
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Bo Li, Mélanie Etheve-Quelquejeu, Expédite Yen-Pon, Christiane Garbay, Huixiong Chen. Microwave-assisted synthesis of 2,5-disubstituted pyrimidine derivatives via Buchwald-Hartwig amination. Tetrahedron Letters, 2020, 61, pp.151406 -. ⟨10.1016/j.tetlet.2019.151406⟩. ⟨hal-03488531⟩
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Yun Luo, Yu Xiao, Delphine Onidas, Laura Iannazzo, Mélanie Ethève-Quelquejeu, et al.. Raman reporters derived from aryl diazonium salts for SERS encoded-nanoparticles. Chemical Communications, 2020, 56 (50), pp.6822-6825. ⟨10.1039/d0cc02842h⟩. ⟨hal-03411993⟩
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Bruno Mégarbane, Camille Gamblin, Olivier Roussel, Elodie Bouaziz-Amar, Lucie Chevillard, et al.. The neurobehavioral effects of the designer drug naphyrone – an experimental investigation with pharmacokinetics and concentration/effect relationship in mice. Psychopharmacology, 2020, 237 (7), pp.1943-1957. ⟨10.1007/s00213-020-05510-2⟩. ⟨hal-03823023⟩
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Alberto Ongaro, Giovanni Ribaudo, Emmanuelle Braud, Mélanie Ethève-Quelquejeu, Michele de Franco, et al.. Design and synthesis of a peptide derivative of ametantrone targeting the major groove of the d(GGCGCC) 2 palindromic sequence. New Journal of Chemistry, 2020, 44 (9), pp.3624-3631. ⟨10.1039/C9NJ03817E⟩. ⟨hal-03689989⟩
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2019

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Usama Ashraf, Laura Tengo, Laurent Le Corre, Guillaume Fournier, Patricia Busca, et al.. Destabilization of the human RED–SMU1 splicing complex as a basis for host-directed antiinfluenza strategy. Proceedings of the National Academy of Sciences of the United States of America, 2019, 116 (22), pp.10968-10977. ⟨10.1073/pnas.1901214116⟩. ⟨hal-02160991⟩
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Luisa Alessandra Atehortua-Martinez, Cyriaque Masniere, Patrizia Campolongo, Stéphanie Chasseigneaux, Jacques Callebert, et al.. Acute and chronic neurobehavioral effects of the designer drug and bath salt constituent 3,4-methylenedioxypyrovalerone in the rat. Journal of Psychopharmacology, 2019, 33 (3), pp.392-405. ⟨10.1177/0269881118822151⟩. ⟨hal-03860016⟩
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Luisa Alessandra Atehortua-Martinez, Cyriaque Masniere, Patrizia Campolongo, Stéphanie Chasseigneaux, Jacques Callebert, et al.. Acute and chronic neurobehavioral effects of the designer drug and bath salt constituent 3,4-methylenedioxypyrovalerone in the rat. Journal of Psychopharmacology, 2019, 33 (3), pp.392-405. ⟨10.1177/0269881118822151⟩. ⟨hal-02557840⟩
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Luisa Alessandra Atehortua-Martinez, Cyriaque Masniere, Patrizia Campolongo, Stéphanie Chasseigneaux, Jacques Callebert, et al.. Acute and chronic neurobehavioral effects of the designer drug and bath salt constituent 3,4-methylenedioxypyrovalerone in the rat. Journal of Psychopharmacology, 2019, 33 (3), pp.392-405. ⟨10.1177/0269881118822151⟩. ⟨hal-03908457⟩
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Nadia Benturquia, Lucie Chevillard, Christophe Poiré, Olivier Roussel, Camille Cohier, et al.. Is the 3,4-methylendioxypyrovalerone/mephedrone combination responsible for enhanced stimulant effects? A rat study with investigation of the effect/concentration relationships. Psychopharmacology, 2019, 236 (3), pp.891-901. ⟨10.1007/s00213-018-4962-0⟩. ⟨hal-03860105⟩
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Nadia Benturquia, Lucie Chevillard, Christophe Poiré, Olivier Roussel, Camille Cohier, et al.. Is the 3,4-methylendioxypyrovalerone/mephedrone combination responsible for enhanced stimulant effects? A rat study with investigation of the effect/concentration relationships. Psychopharmacology, 2019, 236 (3), pp.891-901. ⟨10.1007/s00213-018-4962-0⟩. ⟨hal-03823031⟩
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Nicholus Bhattacharjee, Sébastien Triboulet, Vincent Dubée, Matthieu Fonvielle, Zainab Edoo, et al.. Negative impact of carbapenem methylation on the reactivity of β-lactams for cysteine acylation revealed by quantum calculations and kinetic analyses. Antimicrobial Agents and Chemotherapy, 2019, 63 (4), pp.e02039-18. ⟨10.1128/AAC.02039-18⟩. ⟨hal-02057268⟩
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Etienne Brachet, Aurore Dumond, Wang-Qing Liu, Marie Fabre, Mohamed Selkti, et al.. Synthesis, 3D-structure and stability analyses of NRPa-308, a new promising anti-cancer agent. Bioorganic and Medicinal Chemistry Letters, 2019, 29 (24), pp.126710. ⟨10.1016/j.bmcl.2019.126710⟩. ⟨hal-02418648⟩
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Stephanie Oerum, Marjorie Catala, Colette Atdjian, Franck Brachet, Luc Ponchon, et al.. Bisubstrate analogues as structural tools to investigate m 6 A methyltransferase active sites. RNA Biology, 2019, 16 (6), pp.798-808. ⟨10.1080/15476286.2019.1589360⟩. ⟨hal-02353503⟩
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2018

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Colette Atdjian, Laura Iannazzo, Emmanuelle Braud, Mélanie Ethève-Quelquejeu. Synthesis of SAM-Adenosine Conjugates for the Study of m 6 A-RNA Methyltransferases. European Journal of Organic Chemistry, 2018, 2018 (32), pp.4411-4425. ⟨10.1002/ejoc.201800798⟩. ⟨hal-03689993⟩
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Colette Atdjian, Laura Iannazzo, Emmanuelle Braud, Mélanie Ethève-Quelquejeu. Synthesis of SAM-Adenosine Conjugates for the Study of m 6 A-RNA Methyltransferases. European Journal of Organic Chemistry, 2018, 2018 (32), pp.4411-4425. ⟨10.1002/ejoc.201800798⟩. ⟨hal-02353523⟩
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Colette Atdjian, Laura Iannazzo, Emmanuelle Braud, Mélanie Ethève-Quelquejeu. Synthesis of SAM-Adenosine Conjugates for the Study of m 6 A-RNA Methyltransferases. European Journal of Organic Chemistry, 2018, 2018 (32), pp.4411-4425. ⟨10.1002/ejoc.201800798⟩. ⟨hal-03647207⟩
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Nadia Benturquia, Lucie Chevillard, Christophe Poiré, Olivier Roussel, Camille Cohier, et al.. Is the 3,4-methylendioxypyrovalerone/mephedrone combination responsible for enhanced stimulant effects? A rat study with investigation of the effect/concentration relationships. Psychopharmacology, 2018, ⟨10.1007/s00213-018-4962-0⟩. ⟨hal-01899917⟩
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Zainab Edoo, Laura Iannazzo, Fabrice Compain, Inès Li de La Sierra Gallay, Herman Van Tilbeurgh, et al.. Synthesis of Avibactam Derivatives and Activity on β-Lactamases and Peptidoglycan Biosynthesis Enzymes of Mycobacteria. Chemistry - A European Journal, 2018, 24 (32), pp.8081--8086. ⟨10.1002/chem.201800923⟩. ⟨hal-02177911⟩
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Matthieu Fonvielle, Ahmed Bouhss, Coralie Hoareau, Delphine Patin, Dominique Mengin-Lecreulx, et al.. Synthesis of lipid-carbohydrate-peptidyl-RNA conjugates to explore the limits imposed by the substrate specificity of cell wall enzymes on the acquisition of drug resistance. Chemistry - A European Journal, 2018, 24 (56), pp.14911-14915. ⟨10.1002/chem.201802360⟩. ⟨hal-01962025⟩
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Laura Iannazzo, Matthieu Fonvielle, Emmanuelle Braud, Hubert Hřebabecký, Eliška Procházková, et al.. Synthesis of tRNA analogues containing a terminal ribose locked in the South conformation to study tRNA-dependent enzymes. Organic & Biomolecular Chemistry, 2018, 16 (11), pp.1903-1911. ⟨10.1039/C8OB00019K⟩. ⟨hal-03689994⟩
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Cécile Morlot, Daniel Straume, Katharina Peters, Olav A Hegnar, Nolwenn Simon, et al.. Structure of the essential peptidoglycan amidotransferase MurT/GatD complex from Streptococcus pneumoniae. Nature Communications, 2018, 9, pp.3180. ⟨10.1038/s41467-018-05602-w⟩. ⟨hal-01861372⟩
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Flora Ngadjeua, Emmanuelle Braud, Saidbakhrom Saidjalolov, Laura Iannazzo, Dirk Schnappinger, et al.. Critical Impact of Peptidoglycan Precursor Amidation on the Activity of l,d -Transpeptidases from Enterococcus faecium and Mycobacterium tuberculosis. Chemistry - A European Journal, 2018, 24 (22), pp.5743 - 5747. ⟨10.1002/chem.201706082⟩. ⟨hal-01817697⟩
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Flora Ngadjeua, Emmanuelle Braud, Saidbakhrom Saidjalolov, Laura Iannazzo, Dirk Schnappinger, et al.. Critical Impact of Peptidoglycan Precursor Amidation on the Activity of l,d -Transpeptidases from Enterococcus faecium and Mycobacterium tuberculosis. Chemistry - A European Journal, 2018, 24 (22), pp.5743-5747. ⟨10.1002/chem.201706082⟩. ⟨hal-03647180⟩
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Expédite Yen-Pon, Bo Li, Marta Acebrón-Garcia-De-Eulate, Céline Tomkiewicz-Raulet, John Dawson, et al.. Structure-Based Design, Synthesis, and Characterization of the First Irreversible Inhibitor of Focal Adhesion Kinase. ACS Chemical Biology, 2018, 13 (8), pp.2067-2073. ⟨10.1021/acschembio.8b00250⟩. ⟨hal-02196326⟩
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2017

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Manal Sarkis, Maria Miteva, Maria Chiara Dasso Lang, Maryse Jaouen, Marie-Agnès Sari, et al.. Insights into the interaction of high potency inhibitor IRC-083864 with phosphatase CDC25. Proteins: Structure, Function, and Bioinformatics, 2017, 85 (4), pp.593-601. ⟨10.1002/prot.25236⟩. ⟨hal-03684762⟩
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Manal Sarkis, Maria Miteva, Maria Chiara Dasso Lang, Maryse Jaouen, Marie-Agnès Sari, et al.. Insights into the interaction of high potency inhibitor IRC-083864 with phosphatase CDC25. Proteins: Structure, Function, and Bioinformatics, 2017, 85 (4), pp.593-601. ⟨10.1002/prot.25236⟩. ⟨hal-03689998⟩
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2016

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Matthieu Fonvielle, Nicolas Sakkas, Laura Iannazzo, Chloé Le fournis, Delphine Patin, et al.. Electrophilic RNA for Peptidyl-RNA Synthesis and Site-Specific Cross-Linking with tRNA-Binding Enzymes.. Angewandte Chemie International Edition, 2016, 55 (43), pp.13553-13557. ⟨10.1002/anie.201606843⟩. ⟨hal-01440830⟩
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2015

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P. Dao, N. Smith, Daniel Scott-Algara, C. Garbay, J.P. Herbeuval, et al.. Restoration of TRAIL-induced apoptosis in resistant human pancreatic cancer cells by a novel FAK inhibitor, PH11. Cancer Letters, 2015, 360 (1), pp.48-59. ⟨10.1016/j.canlet.2015.02.016⟩. ⟨pasteur-02573704⟩
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Mickaël J Fer, Ahmed Bouhss, Mariana Patrão, Laurent Le Corre, Nicolas Pietrancosta, et al.. 5'-Methylene-triazole-substituted-aminoribosyl uridines as MraY inhibitors: synthesis, biological evaluation and molecular modeling.. Organic & Biomolecular Chemistry, 2015, 13 (26), pp.7193-222. ⟨10.1039/c5ob00707k⟩. ⟨hal-01433063⟩
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Laura Iannazzo, Erica Benedetti, Marjorie Catala, Mélanie Etheve-Quelquejeu, Carine Tisné, et al.. Monitoring of reversible boronic acid–diol interactions by fluorine NMR spectroscopy in aqueous media. Organic & Biomolecular Chemistry, 2015, 13 (33), pp.8817-8821. ⟨10.1039/c5ob01362c⟩. ⟨hal-03544508⟩
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2014

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Elodie Goldwaser, Benoit de Courcy, Luc Demange, Christiane Garbay, Françoise Raynaud, et al.. Conformational analysis of a polyconjugated protein-binding ligand by joint quantum chemistry and polarizable molecular mechanics. Addressing the issues of anisotropy, conjugation, polarization, and multipole transferability. Journal of Molecular Modeling, 2014, 20 (11), ⟨10.1007/s00894-014-2472-5⟩. ⟨hal-02126794⟩
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Wang-Qing Liu, Valentino Megale, Lucia Borriello, Bertrand Leforban, Matthieu Montes, et al.. Synthesis and structure–activity relationship of non-peptidic antagonists of neuropilin-1 receptor. Bioorganic and Medicinal Chemistry Letters, 2014, 24 (17), pp.4254-4259. ⟨10.1016/j.bmcl.2014.07.028⟩. ⟨hal-02126861⟩
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2013

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Eric Leclerc, Xavier Pannecoucke, Mélanie Etheve-Quelquejeu, M. Sollogoub. Fluoro-C-glycosides and fluoro-carbasugars, hydrolytically stable and synthetically challenging glycomimetics. Chemical Society Reviews, 2013, 42 (10), pp.4270-4283. ⟨10.1039/c2cs35403a⟩. ⟨hal-00825637⟩
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Sébastien Triboulet, Vincent Dubée, Lauriane Lecoq, Catherine M Bougault, Jean-Luc Mainardi, et al.. Kinetic features of L,D-transpeptidase inactivation critical for β-lactam antibacterial activity.. PLoS ONE, 2013, 8 (7), pp.e67831. ⟨10.1371/journal.pone.0067831⟩. ⟨hal-01321589⟩
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2012

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Aurelie Jonquoy, Emilie Mugniery, Catherine Benoist-Lasselin, Nabil Kaci, Laurent Le Corre, et al.. A novel tyrosine kinase inhibitor restores chondrocyte differentiation and promotes bone growth in a gain-of-function Fgfr3 mouse model. Human Molecular Genetics, 2012, 21 (4), pp.841-851. ⟨10.1093/hmg/ddr514⟩. ⟨hal-01019795⟩
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Eric Rose, Nicolas Raoul, Mélanie Etheve-Quelquejeu, Emma Gallo, Bernard Boitrel, et al.. Crystal structure of a chiral binaphthyl porphyrin. Journal of Porphyrins and Phthalocyanines, 2012, 16 (3), pp.324-330. ⟨10.1142/S1088424612500393⟩. ⟨hal-00863134⟩
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2011

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Tatiana Besset, Emmanuelle Braud, Rafika Jarray, Christiane Garbay, Stephanie Kolb, et al.. Preparation and evaluation of a set of bis(methoxycarbonylmethylthio) heteroquinones as CDC25B phosphatase inhibitors. Central European Journal of Chemistry, 2011, 2 (4), pp.433-440. ⟨10.5155/eurjchem.2.4.433-440.400⟩. ⟨hal-02541860⟩
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Benoît Gautier, Maria Miteva, Victor Goncalves, Florent Huguenot, Pascale Coric, et al.. Targeting the Proangiogenic VEGF-VEGFR Protein-Protein Interface with Drug-like Compounds by In Silico and In Vitro Screening. Chemistry and Biology, 2011, 18 (12), pp.1631-1639. ⟨10.1016/j.chembiol.2011.10.016⟩. ⟨hal-01061760⟩
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2010

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B. de Courcy, J. P. Piquemal, C. Garbay, N. Gresh. Polarizable water molecules in ligand-macromolecule recognition. Impact on the relative affinities of competing pyrrolopyrimidine inhibitors for FAK kinase.. Journal of the American Chemical Society, 2010, 132, pp.3312. ⟨hal-00494585⟩
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Réda Hadj-Slimane, Perayot Pamonsinlapatham, Jean-Philippe Herbeuval, Christiane Garbay, Yves Lepelletier, et al.. Rasv12 induces survivin/auroraB pathway conferring tumor cell apoptosis resistance. Cellular Signalling, 2010, 22 (8), pp.1214-1221. ⟨10.1016/j.cellsig.2010.03.013⟩. ⟨hal-00473108⟩
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Réda Hadj-Slimane, Perayot Pamonsinlapatham, Jean-Philippe Herbeuval, Christiane Garbay, Yves Lepelletier, et al.. RasV12 induces Survivin/AuroraB pathway conferring tumor cell apoptosis resistance. Cellular Signalling, 2010, 22 (8), pp.1214-1221. ⟨10.1016/j.cellsig.2010.03.013⟩. ⟨hal-04250005⟩
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2009

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Romain Duval, S. Kolb, E. Braud, D. Genest, C. Garbay. Rapid discovery of Triazolobenzylidene-Thiazolopyrimidines (TBTP) as CDC25 phosphatase inhibitors by parallel click chemistry and in situ screening. Journal of Combinatorial Chemistry, 2009, 11 (6), pp.947-950. ⟨10.1021/cc900140f⟩. ⟨hal-04504305⟩
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P. Pamonsinlapatham, R. Hadj-Slimane, F. Raynaud, M. Bickle, C. Corneloup, et al.. A RasGAP peptide aptamer inhibits RasGAP-Aurora interaction and induces caspase-independent tumor cell death.. PLoS ONE, 2009, 3, pp.e2902. ⟨hal-00422287⟩
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P. Pamonsinlapatham, R. Hadj-Slimane, Y. Lepelletier, B. Allain, M. Toccafondi, et al.. P120-Ras GTPase activating protein (RasGAP): a multi-interacting protein in downstream signaling.. Biochimie, 2009, 91, pp.320-328. ⟨hal-00397954⟩
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2008

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C. Courme, S. Gillon, N. Gresh, M. Vidal, C. Garbay, et al.. Terminal alkyne-functionalized triazine by Sonogashira coupling : synthesis of a potential cell signalling inhibitor via click chemistry. Tetrahedron Letters, 2008, 49, pp.4542-4545. ⟨hal-00323801⟩
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P. Pamonsinlapatham, R. Hadj-Slimane, Y. Lepelletier, B. Allain, M. Toccafondi, et al.. P120-Ras GTPase activating protein (RasGAO): A multi-interacting protein in downstream signaling.. Biochimie, 2008, ?, pp.?-?. ⟨hal-00356306⟩
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Perayot Pamonsinlapatham, Réda Hadj-Slimane, Françoise Raynaud, Marc Bickle, Claudine Corneloup, et al.. A RasGAP SH3 peptide aptamer inhibits RasGAP-Aurora interaction and induces caspase-independent tumor cell death. PLoS ONE, 2008, 3 (8), pp.e2902. ⟨10.1371/journal.pone.0002902⟩. ⟨hal-00416049⟩
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P. Pamonsinlapatham, R. Hadj-Slimane, F. Raynaud, M. Bickle, C. Corneloup, et al.. A RasGAP SH3 peptide aptamer inhibits RASGAP-Aurora interaction and induces caspase-independent tumor cell death.. PLoS ONE, 2008, 3, pp.2902-2914. ⟨hal-00356308⟩
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2007

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Jennifer Dourlat, Bruno Valentin, Wang-Qing Liu, Christiane Garbay. New syntheses of tetrazolylmethylphenylalanine and O-malonyltyrosine as pTyr mimetics for the design of STAT3 dimerization inhibitors.. Bioorganic and Medicinal Chemistry Letters, 2007, 17 (14), pp.3943-6. ⟨10.1016/j.bmcl.2007.04.107⟩. ⟨inserm-00168682⟩
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Jennifer Dourlat, Wang-Qing Liu, Nohad Gresh, Christiane Garbay. Novel 1,4-benzodiazepine derivatives with antiproliferative properties on tumor cell lines.. Bioorganic and Medicinal Chemistry Letters, 2007, 17 (9), pp.2527-30. ⟨10.1016/j.bmcl.2007.02.016⟩. ⟨inserm-00168656⟩
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Victor Goncalves, Benoît Gautier, Anne Regazzetti, Pascale Coric, Serge Bouaziz, et al.. On-resin cyclization of peptide ligands of the Vascular Endothelial Growth Factor Receptor 1 by copper(I)-catalyzed 1,3-dipolar azide–alkyne cycloaddition. Bioorganic and Medicinal Chemistry Letters, 2007, 17 (20), pp.5590-5594. ⟨10.1016/j.bmcl.2007.07.087⟩. ⟨hal-02122521⟩
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Victor Goncalves, Benoît Gautier, Pascale Coric, Serge Bouaziz, Christine Lenoir, et al.. Rational Design, Structure, and Biological Evaluation of Cyclic Peptides Mimicking the Vascular Endothelial Growth Factor. Journal of Medicinal Chemistry, 2007, 50 (21), pp.5135-5146. ⟨10.1021/jm0706970⟩. ⟨hal-02122518⟩
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Victor Goncalves, Benoit Gautier, Christiane Garbay, Michel Vidal, Nicolas Inguimbert. Development of a chemiluminescent screening assay for detection of vascular endothelial growth factor receptor 1 ligands.. Analytical Biochemistry, 2007, 366 (1), pp.108-10. ⟨10.1016/j.ab.2007.03.027⟩. ⟨inserm-00168674⟩
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Brunilde Gril, Michel Vidal, Franck Assayag, Marie-France Poupon, Wang-Qing Liu, et al.. Grb2-SH3 ligand inhibits the growth of HER2+ cancer cells and has antitumor effects in human cancer xenografts alone and in combination with docetaxel.. International Journal of Cancer, 2007, 121 (2), pp.407-15. ⟨10.1002/ijc.22674⟩. ⟨inserm-00168667⟩
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R. Hadj-Slimane, Y. Lepelletier, N. Lopez, C. Garbay, F. Raynaud. Short interfering RNA (siRNA), a novel therapeutic tool acting on angiogenesis.. Biochimie, 2007, 89, pp.1234-1244. ⟨hal-00172570⟩
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Vincent Leroux, Nohad Gresh, Wang-Qing Liu, Christiane Garbay, Bernard Maigret. Role of water molecules for binding inhibitors in the SH2 domain of Grb2: a molecular dynamics study. Journal of Molecular Structure: THEOCHEM, 2007, 806 (1-3), pp.51-66. ⟨inria-00188596⟩
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Hiba Noureddine, Claudine Schmitt, Wangqing Liu, Christiane Garbay, Jean Massoulié, et al.. Assembly of acetylcholinesterase tetramers by peptidic motifs from the proline-rich membrane anchor, PRiMA: competition between degradation and secretion pathways of heteromeric complexes.. Journal of Biological Chemistry, 2007, 282 (6), pp.3487-97. ⟨10.1074/jbc.M607221200⟩. ⟨hal-00140001⟩
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Régis Villet, Matthieu Fonvielle, Patricia Busca, Maryline Chemama, Antoine P. Maillard, et al.. Idiosyncratic features in tRNAs participating in bacterial cell wall synthesis. Nucleic Acids Research, 2007, 35 (20), pp.6870-6883. ⟨10.1093/nar/gkm778⟩. ⟨hal-02331010⟩
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2005

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Marie-Priscille Brun, Emmanuelle Braud, Delphine Angotti, Odile Mondésert, Muriel Quaranta, et al.. Design, synthesis, and biological evaluation of novel naphthoquinone derivatives with CDC25 phosphatase inhibitory activity.. Bioorganic and Medicinal Chemistry, 2005, 13 (16), pp.4871-9. ⟨10.1016/j.bmc.2005.05.005⟩. ⟨hal-00317419⟩
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Stéphanie Gobert Gosse, Caroline Bourgin, Wang Qing Liu, Christiane Garbay, Guy Mouchiroud. M-CSF stimulated differentiation requires persistent MEK activity and MAPK phosphorylation independent of Grb2-Sos association and phosphatidylinositol 3-kinase activity.. Cellular Signalling, 2005, 17 (11), pp.1352-62. ⟨10.1016/j.cellsig.2005.02.002⟩. ⟨hal-00192857⟩
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S. Gobert-Gosse, C. Bourgin, Liu W. Q., C. Garbay, G. Mouchiroud. GM-CSF stimulated differentiation requires persistent MEK activity and MAPK phosphorylation independant of Grb2-Sos association and phosphatidylinositol 3-kinase activity.. Cellular Signalling, 2005, 17, pp.1352-1632. ⟨hal-00150766⟩
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2004

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Virginie Binet, Carole Brajon, Laurent Le Corre, Francine Acher, Jean-Philippe Pin, et al.. The heptahelical domain of GABA(B2) is activated directly by CGP7930, a positive allosteric modulator of the GABA(B) receptor.. Journal of Biological Chemistry, 2004, 279 (28), pp.29085-91. ⟨10.1074/jbc.M400930200⟩. ⟨inserm-00318926⟩
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Marie-Priscille Brun, Laurent Bischoff, Christiane Garbay. A Very Short Route to Enantiomerically Pure Coumarin-Bearing Fluorescent Amino Acids. Angewandte Chemie International Edition, 2004, 43 (26), pp.3432-3436. ⟨10.1002/anie.200454116⟩. ⟨hal-02385514⟩
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Yen Vo-Hoang, Cécile Gasse, Michel Vidal, Christiane Garbay, Hervé Galons. Efficient synthesis of N-benzyl-3-aminopyrrolidine-2,5-dione and N-benzyl-3-aminopyrrolidin-2-one. Tetrahedron Letters, 2004, 45 (18), pp.3603-3605. ⟨10.1016/j.tetlet.2004.03.052⟩. ⟨hal-03531874⟩
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2003

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Marie-Priscille Brun, Anne-Sophie Martin, Christiane Garbay, Laurent Bischoff. An alternative route to the proline derivative (2S,5R)-5-ethoxycarbonylmethyl-pyrrolidine-2-carboxylic acid from protected glutamic acid. Tetrahedron Letters, 2003, 44 (37), pp.7011-7013. ⟨10.1016/S0040-4039(03)01792-1⟩. ⟨hal-02385515⟩
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2002

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Wang-Qing Liu, Catherine Olszowy, Laurent Bischoff, Christiane Garbay. Enantioselective synthesis of (2S)-2-(4-phosphonophenylmethyl)-3-aminopropanoic acid suitably protected for peptide synthesis. Tetrahedron Letters, 2002, 43 (8), pp.1417-1419. ⟨10.1016/S0040-4039(02)00004-7⟩. ⟨hal-02385516⟩
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Pierre Nioche, Wang-Qing Liu, Isabelle Broutin, Franck Charbonnier, Marie-Thérèse Latreille, et al.. Crystal structures of the SH2 domain of grb2: highlight on the binding of a new high-affinity inhibitor. Journal of Molecular Biology, 2002, 315 (5), pp.1167-1177. ⟨10.1006/jmbi.2001.5299⟩. ⟨hal-02520104⟩
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2001

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Katia Cailliau, Edith Browaeys-Poly, Isabelle Broutin-L'Hermite, Pierre Nioche, Christiane Garbay, et al.. Grb2 promotes reinitiation of meiosis in Xenopus oocytes. Cellular Signalling, 2001, 13 (1), pp.51-55. ⟨10.1016/s0898-6568(00)00138-8⟩. ⟨hal-02520116⟩
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2000

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B Bellier, M. Million, S Danascimento, H. Meudal, S Kellou, et al.. Replacement of glycine with dicarbonyl and related moieties in analogues of the C-terminal pentapeptide of cholecystokinin: CCK(2) agonists displaying a novel binding mode.. Journal of Medicinal Chemistry, 2000, 43 (20), pp.3614-23. ⟨hal-02122170⟩
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Marie-France Carlier, Pierre Nioche, Isabelle Broutin-L'Hermite, Rajaa Boujemaa, Christophe Le Clainche, et al.. GRB2 Links Signaling to Actin Assembly by Enhancing Interaction of Neural Wiskott-Aldrich Syndrome Protein (N-WASp) with Actin-related Protein (ARP2/3) Complex. Journal of Biological Chemistry, 2000, 275 (29), pp.21946-21952. ⟨10.1074/jbc.M000687200⟩. ⟨hal-02520338⟩
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1998

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B Bellier, S da Nascimento, H. Meudal, E. Gincel, B.P Roques, et al.. Novel constrained CCK-B dipeptoid antagonists derived from pipecolic acid.. Bioorganic and Medicinal Chemistry Letters, 1998, 8 (11), pp.1419-24. ⟨hal-02122133⟩
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1997

ref_biblio
Bruno Bellier, Isabelle Mccort, Bertrand Ducos, Sophie Danascimento, Hervé Meudal, et al.. Synthesis and Biological Properties of New Constrained CCK-B Antagonists: Discrimination of Two Affinity States of the CCK-B Receptor on Transfected CHO Cells. Journal of Medicinal Chemistry, 1997, 40 (24), pp.3947-3956. ⟨10.1021/jm970439a⟩. ⟨hal-02122116⟩
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Journal articles

2025

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Hichem Ichou, Kevin Telliez, Sonia Lajnef, Fabienne Peyrot, Benjamin Doistau, et al.. Anion-mediated properties of a metal complex in a hexameric resorcin[4]arene cage: chirality induction, kinetics and reactivity. Inorganic Chemistry Frontiers, 2025, 12 (3), pp.1028-1039. ⟨10.1039/d4qi02896a⟩. ⟨hal-05158345⟩
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2022

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Ivona Krošl, Ena Otković, Ivana Nikšić-Franjić, Benoît Colasson, Olivia Reinaud, et al.. Impact of positive charge and ring-size on the interactions of calixarenes with DNA, RNA and nucleotides. New Journal of Chemistry, 2022, 46 (15), pp.6860-6869. ⟨10.1039/D2NJ00061J⟩. ⟨hal-03627557⟩
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2021

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Tongtong Zhang, Laurent Le Corre, Olivia Reinaud, Benoit Colasson. A Promising Approach for Controlling the Second Coordination Sphere of Biomimetic Metal Complexes: Encapsulation in a Dynamic Hydrogen‐Bonded Capsule. Chemistry - A European Journal, 2021, 27 (1), pp.434-443. ⟨10.1002/chem.202004370⟩. ⟨hal-03154347⟩
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2020

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Jonah Kailer Aw, Kevin Christopher Boellaard, Teck Kiang Tan, John Yap, Yi Ping Loh, et al.. Interacting with Three-Dimensional Molecular Structures Using an Augmented Reality Mobile App. Journal of Chemical Education, 2020, 97 (10), pp.3877-3881. ⟨10.1021/acs.jchemed.0c00387⟩. ⟨hal-03154348⟩
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2019

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Benoit Colasson, Alberto Credi, Barbara Ventura. Photoinduced Electron Transfer Involving a Naphthalimide Chromophore in Switchable and Flexible [2]Rotaxanes. Chemistry - A European Journal, 2019, 26 (2), pp.534-542. ⟨10.1002/chem.201904155⟩. ⟨hal-03154349⟩
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2018

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Alex Inthasot, Nicolas Le Poul, Michel Luhmer, Benoit Colasson, Ivan Jabin, et al.. Selective EPR Detection of Primary Amines in Water with a Calix[6]azacryptand-Based Copper(II) Funnel Complex. Inorganic Chemistry, 2018, ⟨10.1021/acs.inorgchem.7b02541⟩. ⟨hal-01679879⟩
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Nicolas Le Poul, Benoit Colasson, Grégory Thiabaud, Dany Jeanne Dit Fouque, Claudio Iacobucci, et al.. Gating the electron transfer at a monocopper centre through the supramolecular coordination of water molecules within a protein chamber mimic. Chemical Science, 2018, 9 (43), pp.8282-8290. ⟨10.1039/C8SC03124J⟩. ⟨hal-03824727⟩
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Nicolas Le Poul, Benoit Colasson, Grégory Thiabaud, Dany Jeanne Dit Fouque, Claudio Iacobucci, et al.. Gating the electron transfer at a monocopper centre through the supramolecular coordination of water molecules within a protein chamber mimic. Chemical Science, 2018, 9 (43), pp.8282-8290. ⟨10.1039/C8SC03124J⟩. ⟨hal-01874257⟩
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Giulio Ragazzon, Christian Schäfer, Paola Franchi, Serena Silvi, Benoit Colasson, et al.. Remote electrochemical modulation of pK a in a rotaxane by co-conformational allostery. Proceedings of the National Academy of Sciences of the United States of America, 2018, 115 (38), pp.9385-9390. ⟨10.1073/pnas.1712783115⟩. ⟨hal-03154351⟩
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2017

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Alex Inthasot, Nicolas Le Poul, Michel Luhmer, Benoit Colasson, Ivan Jabin, et al.. Selective EPR Detection of Primary Amines in Water with a Calix[6]azacryptand-Based Copper(II) Funnel Complex. Inorganic Chemistry, 2017, 57 (7), pp.3646-3655. ⟨10.1021/acs.inorgchem.7b02541⟩. ⟨hal-03154352⟩
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Giulio Ragazzon, Alberto Credi, Benoit Colasson. Thermodynamic Insights on a Bistable Acid-Base Switchable Molecular Shuttle with Strongly Shifted Co-conformational Equilibria. Chemistry - A European Journal, 2017, 23 (9), pp.2149-2156. ⟨10.1002/chem.201604783⟩. ⟨hal-03154354⟩
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2016

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Benoit Colasson, Alberto Credi, Giulio Ragazzon. Light-driven molecular machines based on ruthenium(II) polypyridine complexes: Strategies and recent advances. Coordination Chemistry Reviews, 2016, 325, pp.125-134. ⟨10.1016/j.ccr.2016.02.012⟩. ⟨hal-03154358⟩
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Alex Inthasot, Emilio Brunetti, Manuel Lejeune, Nicolas Menard, Thierry Prangé, et al.. Kinetic and Thermodynamic Stabilization of Metal Complexes by Introverted Coordination in a Calix[6]azacryptand. Chemistry - A European Journal, 2016, 22 (14), pp.4855-4862. ⟨10.1002/chem.201505057⟩. ⟨hal-03154357⟩
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Christian Schäfer, Giulio Ragazzon, Benoit Colasson, Marcello La rosa, Serena Silvi, et al.. An Artificial Molecular Transporter. ChemistryOpen, 2016, 5 (2), pp.120-124. ⟨10.1002/open.201500217⟩. ⟨hal-03154356⟩
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2015

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Pierre-Edouard Danjou, Gael de Leener, Damien Cornut, Steven Moerkerke, Samir Mameri, et al.. Supramolecular Assistance for the Selective Demethylation of Calixarene-Based Receptors. Journal of Organic Chemistry, 2015, 80 (10), pp.5084-5091. ⟨10.1021/acs.joc.5b00464⟩. ⟨hal-02865837⟩
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Nicolas Le Poul, Benoit Colasson. Electrochemically and Chemically Induced Redox Processes in Molecular Machines. ChemElectroChem, 2015, 2 (4), pp.475. ⟨10.1002/celc.201402399⟩. ⟨hal-01171145⟩
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ref_biblio
Jean-Noël Rebilly, Benoit Colasson, Olivia Bistri, Diana Over, Olivia Reinaud. Biomimetic cavity-based metal complexes. Chemical Society Reviews, 2015, 44 (2), pp.467-489. ⟨10.1039/c4cs00211c⟩. ⟨hal-03154360⟩
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https://hal.science/hal-03154360/file/Rev%20JChemSoc%20020914%20sans%20liens%20endnote_revised.pdf BibTex

2013

ref_biblio
Nicolas Menard, Yohann Heriot, Yves Le Mest, Olivia Reinaud, Nicolas Le Poul, et al.. Electrochemically Driven Cup-and-Ball Cu-I and Cu-II Complexes. Chemistry - A European Journal, 2013, 19 (32), pp.10611--10618. ⟨10.1002/chem.201301141⟩. ⟨hal-01175765⟩
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2012

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Grégory Thiabaud, Andrea Brugnara, Michaël Carboni, Nicolas Le Poul, Benoit Colasson, et al.. Synthesis and Studies of a Water-Soluble and Air-Stable Cu-I/Cu-II Open-Shell Funnel Complex. Organic Letters, 2012, 14 (10), pp.2500--2503. ⟨10.1021/ol3007875⟩. ⟨hal-01175768⟩
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2011

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Benoit Colasson, Nicolas Le Poul, Yves Le Mest, Olivia Reinaud. Tris(triazolyl) Calix[6]arene-Based Zinc and Copper Funnel Complexes: Imidazole-like or Pyridine-like? A Comparative Study. Inorganic Chemistry, 2011, 50 (21), pp.10985--10993. ⟨10.1021/ic201540x⟩. ⟨hal-01175770⟩
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2010

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Benoit Colasson, Nicolas Le Poul, Yves Le Mest, Olivia Reinaud. Electrochemically Triggered Double Translocation of Two Different Metal Ions with a Ditopic Calix[6]arene Ligand. Journal of the American Chemical Society, 2010, 132 (12), pp.4393--4398. ⟨10.1021/ja910676z⟩. ⟨hal-01175771⟩
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2009

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G. Thiabaud, G. Guillemot, Isabelle Schmitz-Afonso, B. Colasson, O. Reinaud. Solid-state chemistry at an isolated copper(I) center with O2. Angewandte Chemie International Edition, 2009, 48 (40), pp.7383-7386. ⟨10.1002/anie.200902691⟩. ⟨hal-00469664⟩
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2005

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Christiane Dietrich-Buchecker, Benoit Colasson, Damien Jouvenot, Jean-Pierre Sauvage. Synthesis of Multi-1,10-phenanthroline Ligands with 1,3-Phenylene Linkers and Their Lithium Complexes. Chemistry - A European Journal, 2005, 11 (15), pp.4374 - 4386. ⟨10.1002/chem.200401264⟩. ⟨hal-01689666⟩
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